CA2510223C - Transdermal buprenorphine dosage regimen for analgesia - Google Patents
Transdermal buprenorphine dosage regimen for analgesia Download PDFInfo
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- CA2510223C CA2510223C CA2510223A CA2510223A CA2510223C CA 2510223 C CA2510223 C CA 2510223C CA 2510223 A CA2510223 A CA 2510223A CA 2510223 A CA2510223 A CA 2510223A CA 2510223 C CA2510223 C CA 2510223C
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- buprenorphine
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43342302P | 2002-12-13 | 2002-12-13 | |
| US60/433,423 | 2002-12-13 | ||
| PCT/US2003/039792 WO2004054553A1 (en) | 2002-12-13 | 2003-12-15 | Transdermal buprenorphine dosage regimen for analgesia |
Publications (2)
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|---|---|
| CA2510223A1 CA2510223A1 (en) | 2004-07-01 |
| CA2510223C true CA2510223C (en) | 2017-09-12 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2510223A Expired - Fee Related CA2510223C (en) | 2002-12-13 | 2003-12-15 | Transdermal buprenorphine dosage regimen for analgesia |
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| JP (2) | JP5054893B2 (enExample) |
| AT (1) | ATE400258T1 (enExample) |
| AU (2) | AU2003297073A1 (enExample) |
| CA (1) | CA2510223C (enExample) |
| CY (1) | CY1108384T1 (enExample) |
| DE (1) | DE60322102D1 (enExample) |
| DK (1) | DK1572167T3 (enExample) |
| ES (1) | ES2310262T3 (enExample) |
| IL (1) | IL169056A (enExample) |
| MX (1) | MXPA05006334A (enExample) |
| NZ (1) | NZ539936A (enExample) |
| PT (1) | PT1572167E (enExample) |
| SI (1) | SI1572167T1 (enExample) |
| WO (1) | WO2004054553A1 (enExample) |
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| US5968547A (en) | 1997-02-24 | 1999-10-19 | Euro-Celtique, S.A. | Method of providing sustained analgesia with buprenorphine |
| US7736665B2 (en) * | 2002-05-31 | 2010-06-15 | Titan Pharmaceuticals, Inc. | Implantable polymeric device for sustained release of buprenorphine |
| MXPA05006334A (es) * | 2002-12-13 | 2005-08-26 | Euro Celtique Sa | Dosis de buprenorfina transdermica para analgesia. |
| ATE499100T1 (de) | 2003-03-31 | 2011-03-15 | Titan Pharmaceuticals Inc | Polymeres implantat zur verzögerten freisetzung von dopamin antagonisten |
| US8790689B2 (en) * | 2003-04-30 | 2014-07-29 | Purdue Pharma L.P. | Tamper resistant transdermal dosage form |
| ME00276B (me) * | 2003-04-30 | 2011-05-10 | Purdue Pharma Lp | Transdermalni dozni oblik otporan na promjene koje sadrže komponentu aktivnog sredstva i komponentu suprotnog sredstva na mjestu koji je ispod sloja aktivnog sredstva |
| US20080026042A1 (en) * | 2003-07-25 | 2008-01-31 | Euro-Celtique S.A. | Preoperative Treatment of Post Operative Pain |
| DK1646328T3 (da) | 2003-07-25 | 2008-02-04 | Euro Celtique Sa | Behandling af afhængighedsophör |
| US20060281775A1 (en) * | 2005-06-14 | 2006-12-14 | Applied Pharmacy Services, Inc. | Two-component pharmaceutical composition for the treatment of pain |
| EP1968539A2 (en) * | 2005-12-13 | 2008-09-17 | Biodelivery Sciences International, Inc. | Abuse resistant transmucosal drug delivery device |
| RU2504377C2 (ru) | 2006-07-21 | 2014-01-20 | БайоДеливери Сайенсиз Интэнэшнл, Инк. | Способ трансмукозальной доставки лекарства, средство трансмукозальной доставки лекарства (варианты) и способ лечения боли |
| DE102006054731B4 (de) | 2006-11-21 | 2013-02-28 | Lts Lohmann Therapie-Systeme Ag | Transdermales therapeutisches System zur Verabreichung des Wirkstoffs Buprenorphin und Verwendung desselben in der Schmerztherapie |
| EP1985292A1 (en) | 2007-04-23 | 2008-10-29 | Grünenthal GmbH | Titration of tapentadol |
| WO2009114118A2 (en) * | 2008-03-08 | 2009-09-17 | Theraquest Biosciences, Inc. | Oral pharmaceutical compositions of buprenorphine and method of use |
| US8741930B2 (en) * | 2008-10-24 | 2014-06-03 | Bridge Pharma, Inc. | Treating xerophthalmia with norketotifen |
| WO2010059894A1 (en) * | 2008-11-21 | 2010-05-27 | Bridge Pharma, Inc. | Ocular formulations of norketotifen |
| SG11201401446RA (en) | 2011-08-18 | 2014-09-26 | Biodelivery Sciences Int Inc | Abuse-resistant mucoadhesive devices for delivery of buprenorphine |
| AR089201A1 (es) * | 2011-12-12 | 2014-08-06 | Lohmann Therapie Syst Lts | Sistema de suministro transdermico |
| US9901539B2 (en) | 2011-12-21 | 2018-02-27 | Biodelivery Sciences International, Inc. | Transmucosal drug delivery devices for use in chronic pain relief |
| AU2013205080B2 (en) * | 2012-12-12 | 2016-07-07 | Lts Lohmann Therapie-Systeme Ag | Transdermal Delivery System |
| LT2810646T (lt) | 2013-06-04 | 2016-10-25 | Lts Lohmann Therapie-Systeme Ag | Transderminė tiekimo sistema |
| WO2017148595A1 (en) * | 2016-02-29 | 2017-09-08 | Grünenthal GmbH | Titration of cebranopadol |
| CA3122430A1 (en) * | 2018-12-14 | 2020-06-18 | Pear Therapeutics, Inc. | A digital therapeutic component to optimize induction of buprenorphine-containing products |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA856002B (en) * | 1984-08-10 | 1987-04-29 | Du Pont | Transdermal delivery of opioids |
| US4806341A (en) | 1985-02-25 | 1989-02-21 | Rutgers, The State University Of New Jersey | Transdermal absorption dosage unit for narcotic analgesics and antagonists and process for administration |
| US5026556A (en) * | 1988-11-10 | 1991-06-25 | Norwich Eaton Pharmaceuticals, Inc. | Compositions for the transdermal delivery of pharmaceutical actives |
| US5240711A (en) * | 1989-11-29 | 1993-08-31 | Lts Lohmann Therapie-Systeme Gmbh & Co. Kg | Transdermal therapeutic system comprising as active component buprenorphine |
| US5225199A (en) | 1990-04-24 | 1993-07-06 | Teijin Limited | Pharmaceutical plasters |
| US5069909A (en) * | 1990-06-20 | 1991-12-03 | Cygnus Therapeutic Systems | Transdermal administration of buprenorphine |
| US5149538A (en) * | 1991-06-14 | 1992-09-22 | Warner-Lambert Company | Misuse-resistive transdermal opioid dosage form |
| JP2886021B2 (ja) * | 1993-03-19 | 1999-04-26 | 帝三製薬株式会社 | 安定な貼付剤 |
| US5613958A (en) | 1993-05-12 | 1997-03-25 | Pp Holdings Inc. | Transdermal delivery systems for the modulated administration of drugs |
| JP2837337B2 (ja) * | 1993-08-10 | 1998-12-16 | 帝三製薬株式会社 | 貼付剤 |
| US5968547A (en) * | 1997-02-24 | 1999-10-19 | Euro-Celtique, S.A. | Method of providing sustained analgesia with buprenorphine |
| JP3662388B2 (ja) * | 1997-05-30 | 2005-06-22 | 日東電工株式会社 | 経皮吸収製剤及びその製造方法 |
| ES2305457T3 (es) | 2002-03-20 | 2008-11-01 | Euro-Celtique S.A. | Metodo de administracion de buprenorfina para tratar la depresion. |
| MXPA05006334A (es) * | 2002-12-13 | 2005-08-26 | Euro Celtique Sa | Dosis de buprenorfina transdermica para analgesia. |
| WO2004103317A2 (en) * | 2003-05-15 | 2004-12-02 | Euro-Celtique S.A. | Transdermal buprenorphine dosage regimen for treatment of diarrhea |
| DK1646328T3 (da) | 2003-07-25 | 2008-02-04 | Euro Celtique Sa | Behandling af afhængighedsophör |
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2003
- 2003-12-15 MX MXPA05006334A patent/MXPA05006334A/es active IP Right Grant
- 2003-12-15 AU AU2003297073A patent/AU2003297073A1/en not_active Abandoned
- 2003-12-15 AT AT03813444T patent/ATE400258T1/de active
- 2003-12-15 EP EP03813444A patent/EP1572167B1/en not_active Expired - Lifetime
- 2003-12-15 CA CA2510223A patent/CA2510223C/en not_active Expired - Fee Related
- 2003-12-15 DK DK03813444T patent/DK1572167T3/da active
- 2003-12-15 WO PCT/US2003/039792 patent/WO2004054553A1/en not_active Ceased
- 2003-12-15 NZ NZ539936A patent/NZ539936A/en not_active IP Right Cessation
- 2003-12-15 ES ES03813444T patent/ES2310262T3/es not_active Expired - Lifetime
- 2003-12-15 JP JP2004560867A patent/JP5054893B2/ja not_active Expired - Fee Related
- 2003-12-15 SI SI200331365T patent/SI1572167T1/sl unknown
- 2003-12-15 PT PT03813444T patent/PT1572167E/pt unknown
- 2003-12-15 US US10/736,043 patent/US7270830B2/en not_active Expired - Lifetime
- 2003-12-15 DE DE60322102T patent/DE60322102D1/de not_active Expired - Lifetime
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2005
- 2005-06-07 IL IL169056A patent/IL169056A/en active IP Right Grant
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2008
- 2008-09-30 CY CY20081101079T patent/CY1108384T1/el unknown
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2010
- 2010-04-14 AU AU2010201479A patent/AU2010201479B2/en not_active Ceased
- 2010-08-17 JP JP2010182231A patent/JP2010285457A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| US7270830B2 (en) | 2007-09-18 |
| ATE400258T1 (de) | 2008-07-15 |
| CA2510223A1 (en) | 2004-07-01 |
| DK1572167T3 (da) | 2008-10-13 |
| MXPA05006334A (es) | 2005-08-26 |
| AU2010201479A1 (en) | 2010-05-06 |
| JP5054893B2 (ja) | 2012-10-24 |
| AU2003297073A1 (en) | 2004-07-09 |
| JP2006513184A (ja) | 2006-04-20 |
| NZ539936A (en) | 2007-06-29 |
| EP1572167A1 (en) | 2005-09-14 |
| WO2004054553A1 (en) | 2004-07-01 |
| EP1572167A4 (en) | 2007-01-10 |
| DE60322102D1 (de) | 2008-08-21 |
| PT1572167E (pt) | 2008-10-03 |
| JP2010285457A (ja) | 2010-12-24 |
| WO2004054553A9 (en) | 2005-09-15 |
| AU2010201479B2 (en) | 2012-11-01 |
| SI1572167T1 (sl) | 2008-12-31 |
| CY1108384T1 (el) | 2014-02-12 |
| US20040126416A1 (en) | 2004-07-01 |
| IL169056A (en) | 2012-01-31 |
| ES2310262T3 (es) | 2009-01-01 |
| EP1572167B1 (en) | 2008-07-09 |
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