CA2508297A1 - Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders - Google Patents
Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders Download PDFInfo
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- CA2508297A1 CA2508297A1 CA002508297A CA2508297A CA2508297A1 CA 2508297 A1 CA2508297 A1 CA 2508297A1 CA 002508297 A CA002508297 A CA 002508297A CA 2508297 A CA2508297 A CA 2508297A CA 2508297 A1 CA2508297 A1 CA 2508297A1
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-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Endocrinology (AREA)
- Psychology (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43349102P | 2002-12-13 | 2002-12-13 | |
| US60/433,491 | 2002-12-13 | ||
| US48348203P | 2003-06-27 | 2003-06-27 | |
| US60/483,482 | 2003-06-27 | ||
| PCT/IB2003/005684 WO2004054565A1 (en) | 2002-12-13 | 2003-12-03 | Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2508297A1 true CA2508297A1 (en) | 2004-07-01 |
Family
ID=32600152
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002508297A Abandoned CA2508297A1 (en) | 2002-12-13 | 2003-12-03 | Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20040138305A1 (https=) |
| EP (1) | EP1572187A1 (https=) |
| JP (1) | JP2006511604A (https=) |
| KR (1) | KR100845932B1 (https=) |
| AU (1) | AU2003286300A1 (https=) |
| BR (1) | BR0317263A (https=) |
| CA (1) | CA2508297A1 (https=) |
| MX (1) | MXPA05006209A (https=) |
| PL (1) | PL377662A1 (https=) |
| TW (1) | TW200412939A (https=) |
| WO (1) | WO2004054565A1 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL189872B1 (pl) | 1996-07-24 | 2005-10-31 | Warner Lambert Co | Zastosowanie izobutylogaby i jej pochodnych do wytwarzania leku do leczenia bólu |
| JP2007505095A (ja) * | 2003-09-12 | 2007-03-08 | ワーナー−ランバート カンパニー リミティド ライアビリティー カンパニー | うつ病及び不安障害の治療のためのアルファ−２−デルタリガンド及びｓｓｒｉ及び／又はｓｎｒｉを含む組み合わせ |
| AU2007222112A1 (en) * | 2006-03-06 | 2007-09-13 | Pfizer Products Inc. | Alpha-2-delta ligands for non-restorative sleep |
| EP1857836B1 (en) * | 2006-05-15 | 2009-10-21 | Eldim Sa | Device and method for discriminating cerenkov and scintillation radiation |
| US20080161393A1 (en) * | 2006-12-08 | 2008-07-03 | Barrett Ronald W | Use of prodrugs of GABA analogs for treating disease |
| US7868043B2 (en) | 2008-01-25 | 2011-01-11 | Xenoport, Inc. | Mesophasic forms of (3S)-aminomethyl-5-methyl-hexanoic acid prodrugs and methods of use |
| EP2250148B1 (en) | 2008-01-25 | 2016-08-17 | XenoPort, Inc. | Crystalline form of calcium-salts of (3s)-aminomethyl-5-methyl-hexanoic acids and methods of use |
| ES2601852T3 (es) * | 2008-01-25 | 2017-02-16 | Xenoport, Inc. | Forma cristalina de sales de calcio de ácidos (3S)-aminometil-5-metil-hexanoicos y métodos de uso |
| ES2758554T3 (es) | 2009-12-08 | 2020-05-05 | Univ Case Western Reserve | Aminoácidos gama para tratamiento de trastornos oculares |
| US8580850B2 (en) | 2011-08-11 | 2013-11-12 | Xenoport, Inc. | Anhydrous and hemihydrate crystalline forms of an (R)-baclofen prodrug, methods of synthesis and methods of use |
| ES2961655T3 (es) | 2013-01-18 | 2024-03-13 | Kemphys Ltd | Medicamento para tratamiento de enfermedad neuropática |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2460891C2 (de) * | 1974-12-21 | 1982-09-23 | Gödecke AG, 1000 Berlin | 1-Aminomethyl-1-cycloalkanessigsäuren und deren Ester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
| US4087544A (en) * | 1974-12-21 | 1978-05-02 | Warner-Lambert Company | Treatment of cranial dysfunctions using novel cyclic amino acids |
| US6197819B1 (en) * | 1990-11-27 | 2001-03-06 | Northwestern University | Gamma amino butyric acid analogs and optical isomers |
| US6372792B1 (en) * | 1996-04-26 | 2002-04-16 | Guy Chouinard | Method for treating anxiety, anxiety disorders and insomnia |
| PL189872B1 (pl) * | 1996-07-24 | 2005-10-31 | Warner Lambert Co | Zastosowanie izobutylogaby i jej pochodnych do wytwarzania leku do leczenia bólu |
| WO1998017627A1 (en) * | 1996-10-23 | 1998-04-30 | Warner-Lambert Company | Substituted gamma aminobutyric acids as pharmaceutical agents |
| WO1999008670A1 (en) * | 1997-08-20 | 1999-02-25 | Guglietta, Antonio | Gaba analogs to prevent and treat gastrointestinal damage |
| EP0974351A3 (en) * | 1998-04-24 | 2000-12-13 | Jouveinal | Medicament for preventing and treating gastrointestinal damage |
| EP1082306A1 (en) * | 1998-05-26 | 2001-03-14 | Warner-Lambert Company | Conformationally constrained amino acid compounds having affinity for the alpha2delta subunit of a calcium channel |
| JP2002520277A (ja) * | 1998-07-09 | 2002-07-09 | ワーナー−ランバート・カンパニー | 不眠症を治療する方法 |
| EP1121114B1 (en) * | 1998-10-16 | 2007-01-10 | Warner-Lambert Company Llc | Use of gaba analogs for the manufacture of a medicament for the treatment of mania and bipolar disorders |
| AU1602100A (en) * | 1998-11-25 | 2000-06-13 | Warner-Lambert Company | Improved gamma amino butyric acid analogs |
| AU3735000A (en) * | 1999-05-05 | 2000-11-21 | Warner-Lambert Company | Modulation of substance p by gaba analogs and methods relating thereto |
| RS50352B (sr) * | 1999-06-10 | 2009-11-10 | Warner-Lambert Company Llc., | Monosupstituisane 3-propil gama-aminobuterne kiseline |
| CA2449729C (en) * | 2001-06-11 | 2009-11-03 | Xenoport, Inc. | Prodrugs of gaba analogs, compositions and uses thereof |
| US6635675B2 (en) * | 2001-11-05 | 2003-10-21 | Cypress Bioscience, Inc. | Method of treating chronic fatigue syndrome |
| EP1471909A4 (en) * | 2002-01-16 | 2007-07-25 | Endo Pharmaceuticals Inc | PHARMACEUTICAL COMPOSITION AND METHOD FOR THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM |
-
2003
- 2003-12-03 EP EP03777043A patent/EP1572187A1/en not_active Withdrawn
- 2003-12-03 AU AU2003286300A patent/AU2003286300A1/en not_active Abandoned
- 2003-12-03 JP JP2005502468A patent/JP2006511604A/ja not_active Withdrawn
- 2003-12-03 MX MXPA05006209A patent/MXPA05006209A/es unknown
- 2003-12-03 BR BR0317263-5A patent/BR0317263A/pt not_active IP Right Cessation
- 2003-12-03 KR KR1020057010503A patent/KR100845932B1/ko not_active Expired - Fee Related
- 2003-12-03 PL PL377662A patent/PL377662A1/pl not_active Application Discontinuation
- 2003-12-03 WO PCT/IB2003/005684 patent/WO2004054565A1/en not_active Ceased
- 2003-12-03 CA CA002508297A patent/CA2508297A1/en not_active Abandoned
- 2003-12-09 US US10/731,225 patent/US20040138305A1/en not_active Abandoned
- 2003-12-12 TW TW092135200A patent/TW200412939A/zh unknown
-
2007
- 2007-05-18 US US11/804,789 patent/US20070238749A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004054565A8 (en) | 2004-09-10 |
| EP1572187A1 (en) | 2005-09-14 |
| US20070238749A1 (en) | 2007-10-11 |
| JP2006511604A (ja) | 2006-04-06 |
| KR100845932B1 (ko) | 2008-07-11 |
| US20040138305A1 (en) | 2004-07-15 |
| TW200412939A (en) | 2004-08-01 |
| BR0317263A (pt) | 2005-11-08 |
| MXPA05006209A (es) | 2005-08-19 |
| KR20050084236A (ko) | 2005-08-26 |
| PL377662A1 (pl) | 2006-02-06 |
| WO2004054565A1 (en) | 2004-07-01 |
| AU2003286300A1 (en) | 2004-07-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |