AU2003286300A1 - Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders - Google Patents
Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders Download PDFInfo
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- AU2003286300A1 AU2003286300A1 AU2003286300A AU2003286300A AU2003286300A1 AU 2003286300 A1 AU2003286300 A1 AU 2003286300A1 AU 2003286300 A AU2003286300 A AU 2003286300A AU 2003286300 A AU2003286300 A AU 2003286300A AU 2003286300 A1 AU2003286300 A1 AU 2003286300A1
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- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Anesthesiology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43349102P | 2002-12-13 | 2002-12-13 | |
| US60/433,491 | 2002-12-13 | ||
| US48348203P | 2003-06-27 | 2003-06-27 | |
| US60/483,482 | 2003-06-27 | ||
| PCT/IB2003/005684 WO2004054565A1 (en) | 2002-12-13 | 2003-12-03 | Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2003286300A1 true AU2003286300A1 (en) | 2004-07-09 |
Family
ID=32600152
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2003286300A Abandoned AU2003286300A1 (en) | 2002-12-13 | 2003-12-03 | Pregabalin and derivates thereof for the treatment of fibromyalgia and other related disorders |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20040138305A1 (https=) |
| EP (1) | EP1572187A1 (https=) |
| JP (1) | JP2006511604A (https=) |
| KR (1) | KR100845932B1 (https=) |
| AU (1) | AU2003286300A1 (https=) |
| BR (1) | BR0317263A (https=) |
| CA (1) | CA2508297A1 (https=) |
| MX (1) | MXPA05006209A (https=) |
| PL (1) | PL377662A1 (https=) |
| TW (1) | TW200412939A (https=) |
| WO (1) | WO2004054565A1 (https=) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL126999A (en) | 1996-07-24 | 2002-03-10 | Warner Lambert Co | Pharmaceutical preparations containing isobutylgaba and its history for use in the treatment of pain |
| AU2004271796A1 (en) * | 2003-09-12 | 2005-03-24 | Warner-Lambert Company Llc | Combination comprising an alpha-2-delta ligand and an SSRI and/or SNRI for treatment of depression and anxiety disorders |
| CN101420947A (zh) * | 2006-03-06 | 2009-04-29 | 辉瑞产品公司 | 用于非恢复性睡眠的α-2-δ配体 |
| EP1857836B1 (en) * | 2006-05-15 | 2009-10-21 | Eldim Sa | Device and method for discriminating cerenkov and scintillation radiation |
| WO2008073257A1 (en) * | 2006-12-08 | 2008-06-19 | Xenoport, Inc. | Use of prodrugs of gaba analogs for treating diseases |
| US7868043B2 (en) | 2008-01-25 | 2011-01-11 | Xenoport, Inc. | Mesophasic forms of (3S)-aminomethyl-5-methyl-hexanoic acid prodrugs and methods of use |
| CA2706575C (en) * | 2008-01-25 | 2015-07-14 | Xenoport, Inc. | Enantiomerically resolving acyloxyalkyl thiocarbonates used in synthesizing acyloxyalkyl carbamate prodrugs |
| EP2250148B1 (en) * | 2008-01-25 | 2016-08-17 | XenoPort, Inc. | Crystalline form of calcium-salts of (3s)-aminomethyl-5-methyl-hexanoic acids and methods of use |
| EP2509596B1 (en) | 2009-12-08 | 2019-08-28 | Case Western Reserve University | Gamma aminoacids for treating ocular disorders |
| US8580850B2 (en) | 2011-08-11 | 2013-11-12 | Xenoport, Inc. | Anhydrous and hemihydrate crystalline forms of an (R)-baclofen prodrug, methods of synthesis and methods of use |
| WO2014112152A1 (ja) * | 2013-01-18 | 2014-07-24 | 有限会社ケムフィズ | 神経因性疾病の治療のための医薬 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4087544A (en) * | 1974-12-21 | 1978-05-02 | Warner-Lambert Company | Treatment of cranial dysfunctions using novel cyclic amino acids |
| DE2460891C2 (de) * | 1974-12-21 | 1982-09-23 | Gödecke AG, 1000 Berlin | 1-Aminomethyl-1-cycloalkanessigsäuren und deren Ester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
| US6197819B1 (en) * | 1990-11-27 | 2001-03-06 | Northwestern University | Gamma amino butyric acid analogs and optical isomers |
| US6372792B1 (en) * | 1996-04-26 | 2002-04-16 | Guy Chouinard | Method for treating anxiety, anxiety disorders and insomnia |
| IL126999A (en) * | 1996-07-24 | 2002-03-10 | Warner Lambert Co | Pharmaceutical preparations containing isobutylgaba and its history for use in the treatment of pain |
| ATE361909T1 (de) * | 1996-10-23 | 2007-06-15 | Warner Lambert Co | Substituierte gamma-aminobuttersäurederivate als arzneimittel |
| WO1999008670A1 (en) * | 1997-08-20 | 1999-02-25 | Guglietta, Antonio | Gaba analogs to prevent and treat gastrointestinal damage |
| EP0974351A3 (en) * | 1998-04-24 | 2000-12-13 | Jouveinal | Medicament for preventing and treating gastrointestinal damage |
| WO1999061424A1 (en) * | 1998-05-26 | 1999-12-02 | Warner-Lambert Company | Conformationally constrained amino acid compounds having affinity for the alpha2delta subunit of a calcium channel |
| WO2000002546A2 (en) * | 1998-07-09 | 2000-01-20 | Warner-Lambert Company | Use of caba-analogues for treating insomnia |
| CA2344407C (en) * | 1998-10-16 | 2007-01-09 | Warner-Lambert Company | Method for the treatment of mania and bipolar disorder |
| US6627771B1 (en) * | 1998-11-25 | 2003-09-30 | Pfizer Inc | Gamma amino butyric and acid analogs |
| WO2000067742A2 (en) * | 1999-05-05 | 2000-11-16 | Warner-Lambert Company | Use of gaba analogues for the modulation of substance p |
| ES2317839T3 (es) * | 1999-06-10 | 2009-05-01 | Warner-Lambert Company Llc | Acidos 3-propil gamma-aminobutiricos monosustituidos. |
| ATE540678T1 (de) * | 2001-06-11 | 2012-01-15 | Xenoport Inc | Prodrugs aus gaba-analoga, zusammensetzungen und ihre verwendungen |
| US6635675B2 (en) * | 2001-11-05 | 2003-10-21 | Cypress Bioscience, Inc. | Method of treating chronic fatigue syndrome |
| EP1471909A4 (en) * | 2002-01-16 | 2007-07-25 | Endo Pharmaceuticals Inc | PHARMACEUTICAL COMPOSITION AND METHOD FOR THE TREATMENT OF DISEASES OF THE CENTRAL NERVOUS SYSTEM |
-
2003
- 2003-12-03 MX MXPA05006209A patent/MXPA05006209A/es unknown
- 2003-12-03 EP EP03777043A patent/EP1572187A1/en not_active Withdrawn
- 2003-12-03 AU AU2003286300A patent/AU2003286300A1/en not_active Abandoned
- 2003-12-03 CA CA002508297A patent/CA2508297A1/en not_active Abandoned
- 2003-12-03 WO PCT/IB2003/005684 patent/WO2004054565A1/en not_active Ceased
- 2003-12-03 BR BR0317263-5A patent/BR0317263A/pt not_active IP Right Cessation
- 2003-12-03 KR KR1020057010503A patent/KR100845932B1/ko not_active Expired - Fee Related
- 2003-12-03 JP JP2005502468A patent/JP2006511604A/ja not_active Withdrawn
- 2003-12-03 PL PL377662A patent/PL377662A1/pl not_active Application Discontinuation
- 2003-12-09 US US10/731,225 patent/US20040138305A1/en not_active Abandoned
- 2003-12-12 TW TW092135200A patent/TW200412939A/zh unknown
-
2007
- 2007-05-18 US US11/804,789 patent/US20070238749A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA05006209A (es) | 2005-08-19 |
| JP2006511604A (ja) | 2006-04-06 |
| CA2508297A1 (en) | 2004-07-01 |
| TW200412939A (en) | 2004-08-01 |
| WO2004054565A1 (en) | 2004-07-01 |
| EP1572187A1 (en) | 2005-09-14 |
| BR0317263A (pt) | 2005-11-08 |
| PL377662A1 (pl) | 2006-02-06 |
| KR20050084236A (ko) | 2005-08-26 |
| US20070238749A1 (en) | 2007-10-11 |
| WO2004054565A8 (en) | 2004-09-10 |
| US20040138305A1 (en) | 2004-07-15 |
| KR100845932B1 (ko) | 2008-07-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |