CA2444145C - Preparation of formulations of angiotensin ii at1 receptors antagonists for the treatment of arterial hypertension, other cardiovascular illness and its complications - Google Patents
Preparation of formulations of angiotensin ii at1 receptors antagonists for the treatment of arterial hypertension, other cardiovascular illness and its complications Download PDFInfo
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- CA2444145C CA2444145C CA002444145A CA2444145A CA2444145C CA 2444145 C CA2444145 C CA 2444145C CA 002444145 A CA002444145 A CA 002444145A CA 2444145 A CA2444145 A CA 2444145A CA 2444145 C CA2444145 C CA 2444145C
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BRPI0102252-0 | 2001-04-10 | ||
| BRPI0102252-0B1A BR0102252B1 (pt) | 2001-04-10 | 2001-04-10 | Sistema de liberação controlada para antagonista do receptor AT1 da angiotensina II, composição farmacêutica e seu uso |
| PCT/BR2002/000051 WO2002080910A1 (en) | 2001-04-10 | 2002-04-09 | Preparation of formulations of angiotensin ii at1 receptors antagonists for the treatment of arterial hypertension, other cardiovascular illnesses and its complications |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2444145A1 CA2444145A1 (en) | 2002-10-17 |
| CA2444145C true CA2444145C (en) | 2009-11-10 |
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| CA002444145A Expired - Fee Related CA2444145C (en) | 2001-04-10 | 2002-04-09 | Preparation of formulations of angiotensin ii at1 receptors antagonists for the treatment of arterial hypertension, other cardiovascular illness and its complications |
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| US (4) | US7858597B2 (https=) |
| EP (1) | EP1389106A1 (https=) |
| JP (2) | JP4439814B2 (https=) |
| CN (1) | CN1523985B (https=) |
| BR (1) | BR0102252B1 (https=) |
| CA (1) | CA2444145C (https=) |
| WO (1) | WO2002080910A1 (https=) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR0102252B1 (pt) * | 2001-04-10 | 2013-10-22 | Sistema de liberação controlada para antagonista do receptor AT1 da angiotensina II, composição farmacêutica e seu uso | |
| US8101209B2 (en) | 2001-10-09 | 2012-01-24 | Flamel Technologies | Microparticulate oral galenical form for the delayed and controlled release of pharmaceutical active principles |
| BRPI0105509B8 (pt) * | 2001-11-05 | 2021-05-25 | Univ Minas Gerais | formulações do peptídeo angiotensina-(1-7) usando as ciclodextrinas, lipossomas e o polímero plga |
| CA2480826C (fr) | 2002-04-09 | 2012-02-07 | Flamel Technologies | Formulation pharmaceutique orale sous forme de suspension aqueuse de microcapsules permettant la liberation modifiee de principe(s) actif(s) |
| KR20050005437A (ko) | 2002-04-09 | 2005-01-13 | 플라멜 테크놀로지스 | 아목시실린의 변형 방출을 위한 마이크로캡슐 수성 현탁액형태의 경구 제약학적 제제 |
| US7041832B2 (en) | 2002-04-29 | 2006-05-09 | Tava Pharmaceutical Industries, Ltd. | Processes for preparing losartan and losartan potassium |
| KR100554156B1 (ko) | 2003-07-26 | 2006-02-22 | 학교법인 포항공과대학교 | 쿠커비투릴 유도체가 응집되어 형성된 나노 입자, 그 나노입자에 약물이 담지된 약제학적 조성물, 및 이들의 제조방법 |
| HRP20031029A2 (en) * | 2003-12-12 | 2005-08-31 | Belupo - Lijekovi I Kozmetika D.D. | Process for production of inclusion complexes of valsartan with?-cylodextrin |
| JP2008530185A (ja) * | 2005-02-21 | 2008-08-07 | フラメル・テクノロジー | ロサルタンの経口医薬剤形態 |
| FR2882260A1 (fr) * | 2005-02-21 | 2006-08-25 | Flamel Technologies Sa | Forme pharmaceutique orale multimicroparticulaire a liberation modifiee d'antagonistes des recepteurs de l'angiotensine ii |
| FR2884145A1 (fr) * | 2005-04-06 | 2006-10-13 | Flamel Technologies Sa | Forme pharmaceutique orale de losartan |
| WO2008052295A1 (en) * | 2006-10-30 | 2008-05-08 | Universidade Federal De Minas Gerais | Process for the preparation of compounds of at1 receptor antagonists with angiotensin-(1-7), analogues thereof and/or mixtures of these systems, pharmaceutical compositions thereof and use of their derivative products |
| WO2008089532A1 (en) * | 2007-01-26 | 2008-07-31 | Universidade Federal De Minas Gerais - Ufmg | Pharmaceutical compositions and methods for treating erectile dysfunction |
| EP2197416A1 (en) * | 2007-10-09 | 2010-06-23 | Novartis Ag | Pharmaceutical formulation of valsartan |
| BRPI0800585B8 (pt) | 2008-02-13 | 2021-05-25 | Univ Minas Gerais | composições farmacêuticas do peptídeo des-[asp1]-[ala1]-angiotensina-(1-7) e uso do peptídeo des-[asp1]-[ala1]-angiotensina-(1-7) |
| BR102012009317B1 (pt) * | 2012-04-20 | 2022-05-31 | Universidade Federal De Minas Gerais - Ufmg | Processo de preparação de compostos de inclusão envolvendo ciclodextrinas e fármacos, usando um sistema de fluxo contínuo |
| CN108367079B (zh) * | 2015-11-12 | 2022-11-22 | 灰色视觉公司 | 用于治疗的聚集性微粒 |
| CA3056923A1 (en) | 2017-03-23 | 2018-09-27 | Graybug Vision, Inc. | Drugs and compositions for the treatment of ocular disorders |
| US11160870B2 (en) | 2017-05-10 | 2021-11-02 | Graybug Vision, Inc. | Extended release microparticles and suspensions thereof for medical therapy |
| CN115175664A (zh) * | 2020-03-25 | 2022-10-11 | 耶路撒冷希伯来大学伊森姆研究发展有限公司 | 包含ati受体阻滞剂的脂质体制剂及其用途 |
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-
2001
- 2001-04-10 BR BRPI0102252-0B1A patent/BR0102252B1/pt not_active IP Right Cessation
-
2002
- 2002-04-09 JP JP2002578949A patent/JP4439814B2/ja not_active Expired - Fee Related
- 2002-04-09 CA CA002444145A patent/CA2444145C/en not_active Expired - Fee Related
- 2002-04-09 WO PCT/BR2002/000051 patent/WO2002080910A1/en not_active Ceased
- 2002-04-09 EP EP02713951A patent/EP1389106A1/en not_active Withdrawn
- 2002-04-09 US US10/474,640 patent/US7858597B2/en not_active Expired - Fee Related
- 2002-04-09 CN CN028106814A patent/CN1523985B/zh not_active Expired - Fee Related
-
2007
- 2007-10-31 US US11/980,345 patent/US20080108575A1/en not_active Abandoned
-
2009
- 2009-11-30 JP JP2009272002A patent/JP2010047611A/ja active Pending
-
2010
- 2010-12-23 US US12/977,402 patent/US8293723B2/en not_active Expired - Fee Related
-
2012
- 2012-10-22 US US13/656,941 patent/US20130164341A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1523985B (zh) | 2010-05-12 |
| CN1523985A (zh) | 2004-08-25 |
| US20110091541A1 (en) | 2011-04-21 |
| CA2444145A1 (en) | 2002-10-17 |
| JP2004525167A (ja) | 2004-08-19 |
| US8293723B2 (en) | 2012-10-23 |
| JP4439814B2 (ja) | 2010-03-24 |
| US20080108575A1 (en) | 2008-05-08 |
| US20040171584A1 (en) | 2004-09-02 |
| BR0102252B1 (pt) | 2013-10-22 |
| EP1389106A1 (en) | 2004-02-18 |
| BR0102252A (pt) | 2003-01-21 |
| JP2010047611A (ja) | 2010-03-04 |
| WO2002080910A1 (en) | 2002-10-17 |
| US20130164341A1 (en) | 2013-06-27 |
| US7858597B2 (en) | 2010-12-28 |
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