CA2438001A1 - Use of the disorazoles and their derivatives for the treatment of benign and malignant oncoses - Google Patents
Use of the disorazoles and their derivatives for the treatment of benign and malignant oncoses Download PDFInfo
- Publication number
- CA2438001A1 CA2438001A1 CA002438001A CA2438001A CA2438001A1 CA 2438001 A1 CA2438001 A1 CA 2438001A1 CA 002438001 A CA002438001 A CA 002438001A CA 2438001 A CA2438001 A CA 2438001A CA 2438001 A1 CA2438001 A1 CA 2438001A1
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- Prior art keywords
- alkyl
- disorazole
- treatment
- medicament
- general formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
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- A—HUMAN NECESSITIES
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Pulmonology (AREA)
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- Tropical Medicine & Parasitology (AREA)
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- Dermatology (AREA)
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- Diabetes (AREA)
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- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
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- Orthopedic Medicine & Surgery (AREA)
- Hematology (AREA)
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- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40559402P | 2002-08-24 | 2002-08-24 | |
| US60/405,594 | 2002-08-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2438001A1 true CA2438001A1 (en) | 2004-02-24 |
Family
ID=31993935
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002438001A Abandoned CA2438001A1 (en) | 2002-08-24 | 2003-08-22 | Use of the disorazoles and their derivatives for the treatment of benign and malignant oncoses |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US20040106662A1 (enExample) |
| EP (1) | EP1536789A1 (enExample) |
| JP (1) | JP2006500398A (enExample) |
| KR (1) | KR20050038632A (enExample) |
| CN (1) | CN1678310A (enExample) |
| AR (1) | AR042617A1 (enExample) |
| AU (1) | AU2003296872B2 (enExample) |
| BR (1) | BR0313789A (enExample) |
| CA (1) | CA2438001A1 (enExample) |
| HR (1) | HRP20050277A2 (enExample) |
| IL (1) | IL166588A0 (enExample) |
| MX (1) | MXPA05002157A (enExample) |
| NO (1) | NO20051444L (enExample) |
| NZ (1) | NZ538926A (enExample) |
| PL (1) | PL376407A1 (enExample) |
| RU (1) | RU2322236C2 (enExample) |
| TW (1) | TW200404537A (enExample) |
| UA (1) | UA79480C2 (enExample) |
| WO (1) | WO2004024149A1 (enExample) |
| ZA (1) | ZA200501196B (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HRP20160631T1 (hr) * | 2006-09-06 | 2016-07-15 | Æterna Zentaris Gmbh | Konjugati disorazola i njihovi derivati sa staničnovezajućim molekulama, novi derivati disorazola, postupci njihove pripreme i njihove uporabe |
| BRPI0716190A2 (pt) * | 2006-09-06 | 2013-11-12 | Aeterna Zentaris Gmbh | Conjugados de disorazóis e seus derivados com móleculas de ligação celular, derivados de disorazol, processos para fabricação e uso dos mesmos |
| EP1900742A1 (en) | 2006-09-07 | 2008-03-19 | AEterna Zentaris GmbH | Conjugates of disorazoles and their derivatives with cell-binding molecules, novel disorazole derivatives, processes of manufacturing and uses thereof |
| WO2018237178A1 (en) * | 2017-06-22 | 2018-12-27 | William Marsh Rice University | Synthesis of disorazoles and analogs thereof as potent anticancer agents |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19605024A1 (de) * | 1996-01-31 | 1997-08-07 | Schering Ag | Neue selektive Taxane, Verfahren zu ihrer Herstellung und ihre pharmazeutische Verwendung |
| EA007205B1 (ru) * | 2001-07-31 | 2006-08-25 | Вейне Стейт Юниверсити | Производные хинолина и их использование в качестве противоопухолевых средств |
| UA79293C2 (en) * | 2002-07-03 | 2007-06-11 | Univ Wayne State | 4-(7'-halo-2-quino (xa-) linyloxy)phenoxy propionic acid derivatives as antineoplastic agents |
| WO2004053065A2 (en) * | 2002-12-06 | 2004-06-24 | Kosan Biosciences, Inc. | Disorazole polyketide synthase encoding polynucleotides |
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2003
- 2003-08-22 CN CNA038200937A patent/CN1678310A/zh active Pending
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- 2003-08-22 UA UAA200501355A patent/UA79480C2/uk unknown
- 2003-08-22 HR HR20050277A patent/HRP20050277A2/hr not_active Application Discontinuation
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2005
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2009
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Also Published As
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|---|---|
| BR0313789A (pt) | 2005-07-05 |
| TW200404537A (en) | 2004-04-01 |
| JP2006500398A (ja) | 2006-01-05 |
| IL166588A0 (en) | 2006-01-15 |
| RU2005108570A (ru) | 2005-08-27 |
| RU2322236C2 (ru) | 2008-04-20 |
| NO20051444L (no) | 2005-05-19 |
| NZ538926A (en) | 2006-03-31 |
| KR20050038632A (ko) | 2005-04-27 |
| US20090311264A1 (en) | 2009-12-17 |
| AU2003296872A1 (en) | 2004-04-30 |
| ZA200501196B (en) | 2005-10-26 |
| CN1678310A (zh) | 2005-10-05 |
| WO2004024149A1 (de) | 2004-03-25 |
| AR042617A1 (es) | 2005-06-29 |
| UA79480C2 (en) | 2007-06-25 |
| EP1536789A1 (de) | 2005-06-08 |
| PL376407A1 (en) | 2005-12-27 |
| MXPA05002157A (es) | 2005-05-23 |
| US20040106662A1 (en) | 2004-06-03 |
| AU2003296872B2 (en) | 2008-02-14 |
| HRP20050277A2 (en) | 2005-04-30 |
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