CA2431545A1 - Excitatory amino acid receptor antagonists - Google Patents

Excitatory amino acid receptor antagonists Download PDF

Info

Publication number
CA2431545A1
CA2431545A1 CA002431545A CA2431545A CA2431545A1 CA 2431545 A1 CA2431545 A1 CA 2431545A1 CA 002431545 A CA002431545 A CA 002431545A CA 2431545 A CA2431545 A CA 2431545A CA 2431545 A1 CA2431545 A1 CA 2431545A1
Authority
CA
Canada
Prior art keywords
compound
pharmaceutically acceptable
alkyl
acceptable salt
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002431545A
Other languages
English (en)
French (fr)
Inventor
Michael John Martinelli
Vien Van Khau
Michael Edward Letourneau
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2431545A1 publication Critical patent/CA2431545A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
CA002431545A 2001-01-05 2001-12-20 Excitatory amino acid receptor antagonists Abandoned CA2431545A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US26001401P 2001-01-05 2001-01-05
US60/260,014 2001-01-05
PCT/US2001/044715 WO2002053561A1 (en) 2001-01-05 2001-12-20 Excitatory amino acid receptor antagonists

Publications (1)

Publication Number Publication Date
CA2431545A1 true CA2431545A1 (en) 2002-07-11

Family

ID=22987455

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002431545A Abandoned CA2431545A1 (en) 2001-01-05 2001-12-20 Excitatory amino acid receptor antagonists

Country Status (23)

Country Link
EP (1) EP1351955A1 (ru)
JP (1) JP2004520335A (ru)
KR (1) KR20030066797A (ru)
CN (1) CN1484642A (ru)
AR (1) AR035679A1 (ru)
BR (1) BR0116672A (ru)
CA (1) CA2431545A1 (ru)
CZ (1) CZ20031856A3 (ru)
DZ (1) DZ3460A1 (ru)
EA (1) EA200300770A1 (ru)
EC (1) ECSP034682A (ru)
HR (1) HRP20030544A2 (ru)
HU (1) HUP0302528A2 (ru)
IL (1) IL156138A0 (ru)
MX (1) MXPA03005981A (ru)
NO (1) NO20032973L (ru)
NZ (1) NZ525821A (ru)
PE (1) PE20020792A1 (ru)
PL (1) PL361934A1 (ru)
SK (1) SK8242003A3 (ru)
TW (1) TW591023B (ru)
WO (1) WO2002053561A1 (ru)
ZA (1) ZA200304311B (ru)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5284957A (en) * 1992-09-03 1994-02-08 Eli Lilly And Company Excitatory amino acid receptor antagonists
CA2319652A1 (en) * 1998-02-06 1999-08-12 Michael Urquhart Salts of paroxetine
GB9908175D0 (en) * 1999-04-09 1999-06-02 Lilly Co Eli Method of treating neurological disorders
WO2001001972A2 (en) * 1999-07-06 2001-01-11 Eli Lilly And Company SELECTIVE iGluR5 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF MIGRAINE

Also Published As

Publication number Publication date
EA200300770A1 (ru) 2003-10-30
HRP20030544A2 (en) 2004-08-31
NZ525821A (en) 2004-07-30
TW591023B (en) 2004-06-11
AR035679A1 (es) 2004-06-23
IL156138A0 (en) 2003-12-23
SK8242003A3 (en) 2004-01-08
PE20020792A1 (es) 2002-09-06
NO20032973D0 (no) 2003-06-27
ZA200304311B (en) 2004-09-02
PL361934A1 (en) 2004-10-18
KR20030066797A (ko) 2003-08-09
HUP0302528A2 (hu) 2003-11-28
CZ20031856A3 (cs) 2003-09-17
WO2002053561A1 (en) 2002-07-11
ECSP034682A (es) 2003-08-29
JP2004520335A (ja) 2004-07-08
BR0116672A (pt) 2003-09-23
MXPA03005981A (es) 2003-09-10
CN1484642A (zh) 2004-03-24
DZ3460A1 (fr) 2002-07-11
NO20032973L (no) 2003-06-27
EP1351955A1 (en) 2003-10-15

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Legal Events

Date Code Title Description
FZDE Discontinued