CA2352461A1 - Pharmaceutical composition for periodic administration - Google Patents

Pharmaceutical composition for periodic administration Download PDF

Info

Publication number
CA2352461A1
CA2352461A1 CA002352461A CA2352461A CA2352461A1 CA 2352461 A1 CA2352461 A1 CA 2352461A1 CA 002352461 A CA002352461 A CA 002352461A CA 2352461 A CA2352461 A CA 2352461A CA 2352461 A1 CA2352461 A1 CA 2352461A1
Authority
CA
Canada
Prior art keywords
period
menstrual
estrogen antagonist
pharmaceutical composition
menstruation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002352461A
Other languages
English (en)
French (fr)
Inventor
Tomohito Fujii
Kodo Sato
Yasushi Shimizu
Hiroo Takahashi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aska Pharmaceutical Co Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP10335435A external-priority patent/JP2000159688A/ja
Priority claimed from JP10336019A external-priority patent/JP2000159689A/ja
Application filed by Individual filed Critical Individual
Publication of CA2352461A1 publication Critical patent/CA2352461A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/56Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4535Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CA002352461A 1998-11-26 1999-11-16 Pharmaceutical composition for periodic administration Abandoned CA2352461A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP10335435A JP2000159688A (ja) 1998-11-26 1998-11-26 子宮内膜症の処置又は予防剤
JP10/335435 1998-11-26
JP10/336019 1998-11-26
JP10336019A JP2000159689A (ja) 1998-11-26 1998-11-26 月経異常の処置又は予防剤
PCT/JP1999/006383 WO2000030684A1 (fr) 1998-11-26 1999-11-16 Compositions medicamenteuses a administration periodique

Publications (1)

Publication Number Publication Date
CA2352461A1 true CA2352461A1 (en) 2000-06-02

Family

ID=26575168

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002352461A Abandoned CA2352461A1 (en) 1998-11-26 1999-11-16 Pharmaceutical composition for periodic administration

Country Status (5)

Country Link
EP (1) EP1133996A4 (ko)
KR (1) KR20010080254A (ko)
AU (1) AU1180900A (ko)
CA (1) CA2352461A1 (ko)
WO (1) WO2000030684A1 (ko)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4990538A (en) * 1989-08-23 1991-02-05 Harris Adrian L Use of toremifene and its metabolites for the reversal of multidrug resistance of cancer cells against cytotoxic drugs
GB8926171D0 (en) * 1989-11-20 1990-01-10 Applied Research Systems Treatment of infertility
JP3157882B2 (ja) * 1991-11-15 2001-04-16 帝国臓器製薬株式会社 新規なベンゾチオフエン誘導体
US5461065A (en) * 1993-10-15 1995-10-24 Eli Lilly And Company Methods for inhibiting endometriosis
US5446053A (en) * 1993-12-21 1995-08-29 Eli Lilly And Company Methods of inhibiting dysfunctional uterine bleeding
US5455275A (en) * 1994-05-11 1995-10-03 Eli Lilly And Company Methods for inhibiting endometriosis and uterine fibroid disease with 1,1,2-triphenylbut-1-ene derivatives

Also Published As

Publication number Publication date
EP1133996A1 (en) 2001-09-19
AU1180900A (en) 2000-06-13
WO2000030684A1 (fr) 2000-06-02
EP1133996A4 (en) 2003-04-02
KR20010080254A (ko) 2001-08-22

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Legal Events

Date Code Title Description
FZDE Discontinued