CA2268330A1 - 8(9)-dehydroestradiol derivatives - Google Patents
8(9)-dehydroestradiol derivatives Download PDFInfo
- Publication number
- CA2268330A1 CA2268330A1 CA002268330A CA2268330A CA2268330A1 CA 2268330 A1 CA2268330 A1 CA 2268330A1 CA 002268330 A CA002268330 A CA 002268330A CA 2268330 A CA2268330 A CA 2268330A CA 2268330 A1 CA2268330 A1 CA 2268330A1
- Authority
- CA
- Canada
- Prior art keywords
- dehydroestradiol
- delta
- alpha
- pharmaceutically acceptable
- beta
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0062—Estrane derivatives substituted in position 17 alfa not substituted in position 17 beta
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0066—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa
- C07J1/007—Estrane derivatives substituted in position 17 beta not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2793696P | 1996-10-11 | 1996-10-11 | |
| US60/027,936 | 1996-10-11 | ||
| PCT/US1997/018306 WO1998016544A1 (en) | 1996-10-11 | 1997-10-09 | 8(9)-dehydroestradiol derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2268330A1 true CA2268330A1 (en) | 1998-04-23 |
Family
ID=21840614
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002268330A Abandoned CA2268330A1 (en) | 1996-10-11 | 1997-10-09 | 8(9)-dehydroestradiol derivatives |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0934334A1 (ko) |
| JP (1) | JP2001502328A (ko) |
| KR (1) | KR20000049055A (ko) |
| CN (1) | CN1239967A (ko) |
| AR (1) | AR014096A1 (ko) |
| AU (1) | AU743530B2 (ko) |
| BR (1) | BR9712628A (ko) |
| CA (1) | CA2268330A1 (ko) |
| HU (1) | HUP9903369A3 (ko) |
| IL (1) | IL129029A0 (ko) |
| NZ (1) | NZ335183A (ko) |
| WO (1) | WO1998016544A1 (ko) |
| ZA (1) | ZA979069B (ko) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG154323A1 (en) * | 2001-03-16 | 2009-08-28 | Wyeth Corp | Estrogen replacement therapy |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES341947A1 (es) * | 1966-06-21 | 1968-08-01 | American Home Prod | Un procedimiento para preparar compuestos esteroides. |
| SU286675A1 (ru) * | 1969-01-10 | 1973-08-10 | Институт химии природных соединений СССР | СПОСОБ ПОЛУЧЕНИЯ dl-ЭСТРАДИОЛАйСС-СОЮЗНАЯfi^iffiTau-:::X:.:f-lAfiБИБЛИОТЕКА |
| FR2136891A1 (en) * | 1971-05-07 | 1972-12-29 | Inst Khim Prirodny | Racemic estra-3,17 beta-diol prepn - steroid hormones |
| US5210081A (en) * | 1992-02-26 | 1993-05-11 | American Home Products Corporation | Alkali metal 8,9-dehydroestrone sulfate esters |
| DE4338314C1 (de) * | 1993-11-10 | 1995-03-30 | Jenapharm Gmbh | Pharmazeutische Präparate zur Prophylaxe und Therapie radikalvermittelter Zellschädigungen |
-
1997
- 1997-10-06 AR ARP970104601A patent/AR014096A1/es not_active Application Discontinuation
- 1997-10-09 NZ NZ335183A patent/NZ335183A/xx unknown
- 1997-10-09 KR KR1019990703126A patent/KR20000049055A/ko not_active Application Discontinuation
- 1997-10-09 EP EP97946247A patent/EP0934334A1/en not_active Withdrawn
- 1997-10-09 WO PCT/US1997/018306 patent/WO1998016544A1/en not_active Application Discontinuation
- 1997-10-09 HU HU9903369A patent/HUP9903369A3/hu unknown
- 1997-10-09 CA CA002268330A patent/CA2268330A1/en not_active Abandoned
- 1997-10-09 BR BR9712628-4A patent/BR9712628A/pt not_active IP Right Cessation
- 1997-10-09 JP JP10518462A patent/JP2001502328A/ja active Pending
- 1997-10-09 ZA ZA979069A patent/ZA979069B/xx unknown
- 1997-10-09 CN CN97180394A patent/CN1239967A/zh active Pending
- 1997-10-09 IL IL12902997A patent/IL129029A0/xx unknown
- 1997-10-09 AU AU51459/98A patent/AU743530B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| HUP9903369A3 (en) | 2002-02-28 |
| CN1239967A (zh) | 1999-12-29 |
| EP0934334A1 (en) | 1999-08-11 |
| WO1998016544A1 (en) | 1998-04-23 |
| KR20000049055A (ko) | 2000-07-25 |
| HUP9903369A2 (hu) | 2001-06-28 |
| AU5145998A (en) | 1998-05-11 |
| JP2001502328A (ja) | 2001-02-20 |
| NZ335183A (en) | 2000-09-29 |
| IL129029A0 (en) | 2000-02-17 |
| BR9712628A (pt) | 1999-10-26 |
| AR014096A1 (es) | 2001-02-07 |
| AU743530B2 (en) | 2002-01-31 |
| ZA979069B (en) | 1999-04-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |