CA2264527A1 - Process to prepare pharmaceutical compounds - Google Patents

Process to prepare pharmaceutical compounds Download PDF

Info

Publication number
CA2264527A1
CA2264527A1 CA002264527A CA2264527A CA2264527A1 CA 2264527 A1 CA2264527 A1 CA 2264527A1 CA 002264527 A CA002264527 A CA 002264527A CA 2264527 A CA2264527 A CA 2264527A CA 2264527 A1 CA2264527 A1 CA 2264527A1
Authority
CA
Canada
Prior art keywords
group
alkyl
hydrogen
phenyl
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002264527A
Other languages
English (en)
French (fr)
Inventor
Eric David Moher
Michael John Martinelli
Andrew Hendley Fray
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
University of Hawaii
Wayne State University
Eli Lilly and Co
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2264527A1 publication Critical patent/CA2264527A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C235/34—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CA002264527A 1996-09-06 1997-09-05 Process to prepare pharmaceutical compounds Abandoned CA2264527A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2543796P 1996-09-06 1996-09-06
US60/025,437 1996-09-06
PCT/US1997/015668 WO1998009601A2 (en) 1996-09-06 1997-09-05 Process to prepare pharmaceutical compounds

Publications (1)

Publication Number Publication Date
CA2264527A1 true CA2264527A1 (en) 1998-03-12

Family

ID=21826065

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002264527A Abandoned CA2264527A1 (en) 1996-09-06 1997-09-05 Process to prepare pharmaceutical compounds

Country Status (9)

Country Link
EP (1) EP0934250A4 (de)
JP (1) JP2001500128A (de)
KR (1) KR20010029475A (de)
AU (1) AU4334397A (de)
BR (1) BR9711695A (de)
CA (1) CA2264527A1 (de)
HU (1) HUP0000212A3 (de)
IL (2) IL128643A0 (de)
WO (1) WO1998009601A2 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19911088A1 (de) * 1999-03-12 2000-09-28 Fraunhofer Ges Forschung Manuell geführtes Montagesystem
AU775373B2 (en) 1999-10-01 2004-07-29 Immunogen, Inc. Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1995017093A1 (en) * 1993-12-21 1995-06-29 University Of Hawaii New cryptophycins
US5952298A (en) * 1993-12-21 1999-09-14 The University Of Hawaii Cryptophycins
MD2196B2 (ro) * 1995-03-07 2003-06-30 Юнивэсити Эв Хауайи Criptoficine, procedeu de obţinere, compoziţii farmaceutice pe baza acestora, metodă de inhibare a proliferării celulelor mamiferelor şi metodă de atenuare a stării patologice cauzate de hiperproliferarea celulelor mamiferelor
JP2000501067A (ja) * 1995-08-30 2000-02-02 イーライ・リリー・アンド・カンパニー 医薬化合物
CA2241086A1 (en) * 1995-12-22 1997-07-03 University Of Hawai'i Pharmaceutical compounds
DE69704731D1 (de) * 1996-02-27 2001-06-13 Lilly Co Eli Cryptophycinderivate und ihre Verwendung als antimikrotubuli Mittel

Also Published As

Publication number Publication date
HUP0000212A2 (en) 2000-07-28
EP0934250A2 (de) 1999-08-11
IL128643A (en) 2006-04-10
JP2001500128A (ja) 2001-01-09
KR20010029475A (ko) 2001-04-06
EP0934250A4 (de) 2004-08-11
BR9711695A (pt) 2000-03-08
WO1998009601A2 (en) 1998-03-12
IL128643A0 (en) 2000-01-31
HUP0000212A3 (en) 2001-12-28
WO1998009601A3 (en) 1998-04-23
AU4334397A (en) 1998-03-26

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued