CA2123684A1 - Method for making steroidal peracyl glycosides - Google Patents

Method for making steroidal peracyl glycosides

Info

Publication number
CA2123684A1
CA2123684A1 CA002123684A CA2123684A CA2123684A1 CA 2123684 A1 CA2123684 A1 CA 2123684A1 CA 002123684 A CA002123684 A CA 002123684A CA 2123684 A CA2123684 A CA 2123684A CA 2123684 A1 CA2123684 A1 CA 2123684A1
Authority
CA
Canada
Prior art keywords
beta
zinc
recited
tigogenin
cellobioside
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002123684A
Other languages
English (en)
French (fr)
Inventor
Douglas J. M. Allen
Frank R. Busch
John F. Lambert
Russell J. Shine
Stanley W. Walinsky
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2123684A1 publication Critical patent/CA2123684A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
CA002123684A 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides Abandoned CA2123684A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79757491A 1991-11-25 1991-11-25
US07/797,574 1991-11-25

Publications (1)

Publication Number Publication Date
CA2123684A1 true CA2123684A1 (en) 1993-06-10

Family

ID=25171219

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002123684A Abandoned CA2123684A1 (en) 1991-11-25 1992-10-15 Method for making steroidal peracyl glycosides

Country Status (13)

Country Link
EP (1) EP0619822A1 (fi)
JP (1) JPH0826064B2 (fi)
AU (1) AU659506B2 (fi)
CA (1) CA2123684A1 (fi)
FI (1) FI942394A0 (fi)
HU (1) HUT67035A (fi)
IL (1) IL103797A0 (fi)
MX (1) MX9206761A (fi)
NZ (1) NZ245244A (fi)
PT (1) PT101088A (fi)
TW (1) TW232699B (fi)
WO (1) WO1993011150A1 (fi)
ZA (1) ZA929081B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5563259A (en) * 1992-06-26 1996-10-08 Pfizer Inc. Process for making β-O-cellobiosyl steroid derivatives and trimethyl silyl steroid intermediates used therein
US5606041A (en) * 1992-06-26 1997-02-25 Pfizer Inc. Process for steroidal peracyl glycosides
SK158394A3 (en) * 1992-06-26 1995-05-10 Pfizer Steroidal glycosides
PL311278A1 (en) * 1993-04-28 1996-02-05 Pfizer Crystalline glycosidal spirostantil monohydrate
US5502038A (en) * 1993-06-21 1996-03-26 Medical Research Foundation Of Oregon Cholesterol sequestrant glycosides that inhibit intestinal cholesterol absorption
AU7948394A (en) * 1993-12-28 1995-07-17 Pfizer Inc. Hypocholesterolemic agents
WO1996038466A1 (en) * 1995-05-29 1996-12-05 Pfizer Inc. Steroidal glycosides
US5756470A (en) * 1996-10-29 1998-05-26 Schering Corporation Sugar-substituted 2-azetidinones useful as hypocholesterolemic agents

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4602003A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Synthetic compounds to inhibit intestinal absorption of cholesterol in the treatment of hypercholesterolemia
US4602005A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Tigogenin cellobioside for treating hypercholesterolemia and atherosclerosis

Also Published As

Publication number Publication date
IL103797A0 (en) 1993-04-04
FI942394A (fi) 1994-05-24
PT101088A (pt) 1994-02-28
JPH06510794A (ja) 1994-12-01
JPH0826064B2 (ja) 1996-03-13
MX9206761A (es) 1995-01-31
AU2775892A (en) 1993-06-28
WO1993011150A1 (en) 1993-06-10
ZA929081B (en) 1994-05-24
AU659506B2 (en) 1995-05-18
NZ245244A (en) 1995-04-27
HUT67035A (en) 1995-01-30
HU9401374D0 (en) 1994-08-29
EP0619822A1 (en) 1994-10-19
FI942394A0 (fi) 1994-05-24
TW232699B (fi) 1994-10-21

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued