CA2076431A1 - Condensed pyrimidine derivative - Google Patents

Condensed pyrimidine derivative

Info

Publication number
CA2076431A1
CA2076431A1 CA002076431A CA2076431A CA2076431A1 CA 2076431 A1 CA2076431 A1 CA 2076431A1 CA 002076431 A CA002076431 A CA 002076431A CA 2076431 A CA2076431 A CA 2076431A CA 2076431 A1 CA2076431 A1 CA 2076431A1
Authority
CA
Canada
Prior art keywords
group
set forth
acceptable salt
pharmacologically acceptable
pyrimidine derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002076431A
Other languages
English (en)
French (fr)
Inventor
Hiroaki Nomura
Toru Haneda
Yoshihiko Kotake
Norihiro Ueda
Kyosuke Kitoh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eisai Co Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2076431A1 publication Critical patent/CA2076431A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA002076431A 1991-08-21 1992-08-19 Condensed pyrimidine derivative Abandoned CA2076431A1 (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP20925291 1991-08-21
JP209252/91 1991-08-21
JP251548/91 1991-09-30
JP25154891 1991-09-30
JP21767092A JP3144903B2 (ja) 1991-08-21 1992-08-17 縮合ピリミジン誘導体
JP217670/92 1992-08-17

Publications (1)

Publication Number Publication Date
CA2076431A1 true CA2076431A1 (en) 1993-02-22

Family

ID=27328976

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002076431A Abandoned CA2076431A1 (en) 1991-08-21 1992-08-19 Condensed pyrimidine derivative

Country Status (9)

Country Link
JP (1) JP3144903B2 (enrdf_load_stackoverflow)
KR (1) KR950011740B1 (enrdf_load_stackoverflow)
CN (1) CN1070402A (enrdf_load_stackoverflow)
AU (1) AU655051B2 (enrdf_load_stackoverflow)
CA (1) CA2076431A1 (enrdf_load_stackoverflow)
FI (1) FI923697A7 (enrdf_load_stackoverflow)
HU (1) HUT70180A (enrdf_load_stackoverflow)
NO (1) NO923249L (enrdf_load_stackoverflow)
TW (1) TW202451B (enrdf_load_stackoverflow)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT70208A (en) * 1992-09-25 1995-09-28 Lilly Co Eli Process for preparing 5-substituted pyrrolo[2,3-d]-pyrimidines
US8252804B2 (en) 2008-10-01 2012-08-28 Duquesne University Of The Holy Spirit Selective proton coupled folate transporter and folate receptor, and GARFTase inhibitor compounds and methods of using the same
US20110082158A1 (en) * 2008-10-01 2011-04-07 Aleem Gangjee Selective proton coupled folate transporter and folate receptor, and garftase and/or other folate metabolizing enzymes inhibitor compounds and methods of using the same
CN106188060A (zh) * 2015-04-29 2016-12-07 厦门大学 嘧啶并吡咯类化合物、其制备方法、药用组合物及其应用
CN113788834B (zh) * 2021-09-18 2022-11-29 河南奥思恩医药科技有限公司 2,4-二氯-6,7-二氢-5H-吡咯并[3,4-d]嘧啶盐酸盐的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0438261A3 (en) * 1990-01-16 1992-02-26 Takeda Chemical Industries, Ltd. Condensed heterocyclic glutamic acid derivatives, their production and use

Also Published As

Publication number Publication date
TW202451B (enrdf_load_stackoverflow) 1993-03-21
FI923697A0 (fi) 1992-08-18
KR930004307A (ko) 1993-03-22
AU2115792A (en) 1993-02-25
JP3144903B2 (ja) 2001-03-12
FI923697A7 (fi) 1993-02-22
NO923249D0 (no) 1992-08-19
JPH05186437A (ja) 1993-07-27
NO923249L (no) 1993-02-22
KR950011740B1 (ko) 1995-10-09
CN1070402A (zh) 1993-03-31
AU655051B2 (en) 1994-12-01
HUT70180A (en) 1995-09-28

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Legal Events

Date Code Title Description
FZDE Discontinued