CA2074075A1 - Process for preparing homochiral amines and process for preparing intermediates for the preparation thereof, and the intermediates/in accordance with this process prepared - Google Patents

Process for preparing homochiral amines and process for preparing intermediates for the preparation thereof, and the intermediates/in accordance with this process prepared

Info

Publication number
CA2074075A1
CA2074075A1 CA 2074075 CA2074075A CA2074075A1 CA 2074075 A1 CA2074075 A1 CA 2074075A1 CA 2074075 CA2074075 CA 2074075 CA 2074075 A CA2074075 A CA 2074075A CA 2074075 A1 CA2074075 A1 CA 2074075A1
Authority
CA
Canada
Prior art keywords
phenyl
ethyl
preparing
accordance
glycidyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA 2074075
Other languages
English (en)
French (fr)
Inventor
Lars Westfelt
Aina Westfelt
Bo Birgersson
Lena Andersson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nobel Chemicals AB
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2074075A1 publication Critical patent/CA2074075A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C217/28—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines
    • C07C217/30—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines having the oxygen atom of at least one of the etherified hydroxy groups further bound to a carbon atom of a six-membered aromatic ring
    • C07C217/32—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines having the oxygen atom of at least one of the etherified hydroxy groups further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/02—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions involving the formation of amino groups from compounds containing hydroxy groups or etherified or esterified hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/04—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C235/34—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/16—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals
CA 2074075 1990-01-22 1991-01-15 Process for preparing homochiral amines and process for preparing intermediates for the preparation thereof, and the intermediates/in accordance with this process prepared Abandoned CA2074075A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9000206A SE468211B (sv) 1990-01-22 1990-01-22 Flerstegsfoerfarande foer framstaellning av homokirala aminer
SE9000206-4 1990-01-22

Publications (1)

Publication Number Publication Date
CA2074075A1 true CA2074075A1 (en) 1991-07-23

Family

ID=20378305

Family Applications (1)

Application Number Title Priority Date Filing Date
CA 2074075 Abandoned CA2074075A1 (en) 1990-01-22 1991-01-15 Process for preparing homochiral amines and process for preparing intermediates for the preparation thereof, and the intermediates/in accordance with this process prepared

Country Status (7)

Country Link
EP (1) EP0512020A1 (fi)
JP (1) JPH05506008A (fi)
AU (1) AU638801B2 (fi)
CA (1) CA2074075A1 (fi)
FI (1) FI923305A (fi)
SE (1) SE468211B (fi)
WO (1) WO1991010642A1 (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE222231T1 (de) * 1996-09-18 2002-08-15 Daiso Co Ltd Verfahren zur herstellung von 3-amino-2-hydroxy-1-propylethern
AU3345599A (en) * 1998-04-14 1999-11-01 Samsung Fine Chemicals Co., Ltd. A process for preparing chiral (s)-2,3-disubstituted-1-propylamine derivatives
CN103739512A (zh) * 2014-01-24 2014-04-23 南京工业大学 一种制备(s)-阿替洛尔的方法
JP7108436B2 (ja) * 2018-03-22 2022-07-28 三井化学株式会社 ビフェニル骨格含有エポキシ化合物の製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1269776A (en) * 1968-08-29 1972-04-06 Ici Ltd Epoxides and halohydrins and conversion thereof to alkanolamine derivatives
GB1458392A (en) * 1973-11-09 1976-12-15 Ici Ltd Optically-active 1-aryloxy-2,3-epoxypropane derivatives
US4408063A (en) * 1978-06-27 1983-10-04 Merck & Co., Inc. Preparation of epihalohydrin enantiomers
WO1988000190A1 (en) * 1986-06-25 1988-01-14 Massachusetts Institute Of Technology Optically active derivatives of glycidol

Also Published As

Publication number Publication date
JPH05506008A (ja) 1993-09-02
SE9000206D0 (sv) 1990-01-22
WO1991010642A1 (en) 1991-07-25
AU638801B2 (en) 1993-07-08
AU7224991A (en) 1991-08-05
SE468211B (sv) 1992-11-23
SE9000206L (sv) 1991-07-23
FI923305A0 (fi) 1992-07-20
FI923305A (fi) 1992-07-20
EP0512020A1 (en) 1992-11-11

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Dead