CA1244006A - Substituted peptide compounds - Google Patents
Substituted peptide compoundsInfo
- Publication number
- CA1244006A CA1244006A CA000432071A CA432071A CA1244006A CA 1244006 A CA1244006 A CA 1244006A CA 000432071 A CA000432071 A CA 000432071A CA 432071 A CA432071 A CA 432071A CA 1244006 A CA1244006 A CA 1244006A
- Authority
- CA
- Canada
- Prior art keywords
- lower alkyl
- hydrogen
- carbons
- formula
- oxo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06086—Dipeptides with the first amino acid being basic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06086—Dipeptides with the first amino acid being basic
- C07K5/06095—Arg-amino acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Furan Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39965082A | 1982-07-19 | 1982-07-19 | |
| US399,650 | 1989-08-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1244006A true CA1244006A (en) | 1988-11-01 |
Family
ID=23580391
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA000432071A Expired CA1244006A (en) | 1982-07-19 | 1983-07-08 | Substituted peptide compounds |
Country Status (21)
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS55159749A (en) * | 1979-05-31 | 1980-12-12 | Takeda Chem Ind Ltd | Preparation of dried fish flesh |
| US4500518A (en) * | 1984-04-19 | 1985-02-19 | E. R. Squibb & Sons, Inc. | Amino thiol dipeptides |
| EP0175266B1 (en) * | 1984-09-12 | 1996-03-20 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Antihypertensive derivatives |
| US4629724A (en) * | 1984-12-03 | 1986-12-16 | E. R. Squibb & Sons, Inc. | Amino acid ester and amide renin inhibitors |
| FR2578544A1 (en) * | 1985-03-11 | 1986-09-12 | Usv Pharma Corp | Antihypertension spirocyclic compounds |
| FI89058C (fi) * | 1987-02-27 | 1993-08-10 | Yamanouchi Pharma Co Ltd | Foerfarande foer framstaellning av som remin-inhibitorer anvaenda 2-(l-alanyl-l-histidylamino)-butanol-derivat |
| EP1264707A3 (en) | 2001-05-14 | 2004-05-19 | Oji Paper Co., Ltd. | Thermosensitive recording material and novel color developer compounds |
| WO2018130576A1 (en) | 2017-01-10 | 2018-07-19 | Mitsubishi Hitec Paper Europe Gmbh | Novel colour developer for a thermo-sensitive recording medium, and a heat-sensitive recording material based on pla |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3751239A (en) * | 1969-05-29 | 1973-08-07 | Rohm & Haas | Herbicidal compositions containing n-(1,1-dialkyl-3-chloroacetonyl) benzamides |
| JPS5430167A (en) * | 1977-08-11 | 1979-03-06 | Mitsubishi Chem Ind Ltd | 4-aminomethyl-2-phenyloxazoles and their pharmaceutically acceptable acid salts |
| IL58849A (en) * | 1978-12-11 | 1983-03-31 | Merck & Co Inc | Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them |
| FR2480747A1 (fr) * | 1980-04-17 | 1981-10-23 | Roques Bernard | Derives d'acides amines et leur application therapeutique |
| IE51409B1 (en) * | 1980-07-24 | 1986-12-24 | Ici Ltd | Amide derivatives |
| GR75019B (enrdf_load_stackoverflow) * | 1980-09-17 | 1984-07-12 | Univ Miami | |
| ATE20469T1 (de) * | 1980-10-23 | 1986-07-15 | Schering Corp | Carboxyalkyl-dipeptide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel. |
| US4462943A (en) * | 1980-11-24 | 1984-07-31 | E. R. Squibb & Sons, Inc. | Carboxyalkyl amino acid derivatives of various substituted prolines |
| CY1406A (en) * | 1980-12-18 | 1988-04-22 | Schering Corp | Substituted dipeptides, processes for their preparation and pharmaceutical compositions containing them and their use in the inhibition of enkephalinase |
| US4514391A (en) * | 1983-07-21 | 1985-04-30 | E. R. Squibb & Sons, Inc. | Hydroxy substituted peptide compounds |
-
1983
- 1983-06-30 AU AU16432/83A patent/AU1643283A/en not_active Abandoned
- 1983-06-30 IL IL69136A patent/IL69136A0/xx unknown
- 1983-07-07 ZA ZA834980A patent/ZA834980B/xx unknown
- 1983-07-08 GB GB08318492A patent/GB2123834B/en not_active Expired
- 1983-07-08 CA CA000432071A patent/CA1244006A/en not_active Expired
- 1983-07-13 FR FR838311764A patent/FR2530238B1/fr not_active Expired
- 1983-07-14 JP JP58129255A patent/JPS5951246A/ja active Granted
- 1983-07-15 IE IE1655/83A patent/IE55818B1/en not_active IP Right Cessation
- 1983-07-18 NL NL8302562A patent/NL8302562A/nl not_active Application Discontinuation
- 1983-07-18 ES ES524200A patent/ES524200A0/es active Granted
- 1983-07-18 KR KR1019830003289A patent/KR840005709A/ko not_active Withdrawn
- 1983-07-18 HU HU832537A patent/HU187090B/hu unknown
- 1983-07-18 IT IT22114/83A patent/IT1163800B/it active
- 1983-07-18 GR GR71963A patent/GR79602B/el unknown
- 1983-07-18 DE DE19833325850 patent/DE3325850A1/de not_active Ceased
- 1983-07-18 PT PT77045A patent/PT77045B/pt unknown
- 1983-07-18 SE SE8304031A patent/SE8304031L/ not_active Application Discontinuation
- 1983-07-18 DK DK330683A patent/DK330683A/da not_active Application Discontinuation
- 1983-07-19 BE BE0/211203A patent/BE897327A/fr not_active IP Right Cessation
- 1983-07-19 CH CH3950/83A patent/CH659475A5/fr not_active IP Right Cessation
- 1983-07-19 FI FI832620A patent/FI832620L/fi not_active Application Discontinuation
-
1984
- 1984-01-05 FR FR8400115A patent/FR2540867B1/fr not_active Expired
- 1984-01-05 FR FR8400114A patent/FR2540866A1/fr active Pending
- 1984-12-27 ES ES539084A patent/ES8707550A1/es not_active Expired
- 1984-12-27 ES ES539083A patent/ES8707549A1/es not_active Expired
- 1984-12-27 ES ES539082A patent/ES8707548A1/es not_active Expired
-
1991
- 1991-09-11 JP JP3231633A patent/JPH0653713B2/ja not_active Expired - Lifetime
- 1991-09-11 JP JP3231635A patent/JPH0645582B2/ja not_active Expired - Lifetime
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MKEX | Expiry | ||
| MKEX | Expiry |
Effective date: 20051101 |