CA1156656A - Process for the preparation of pyrimidyl-chinazolines - Google Patents
Process for the preparation of pyrimidyl-chinazolinesInfo
- Publication number
- CA1156656A CA1156656A CA000373945A CA373945A CA1156656A CA 1156656 A CA1156656 A CA 1156656A CA 000373945 A CA000373945 A CA 000373945A CA 373945 A CA373945 A CA 373945A CA 1156656 A CA1156656 A CA 1156656A
- Authority
- CA
- Canada
- Prior art keywords
- atoms
- formula
- amino
- process according
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pretreatment Of Seeds And Plants (AREA)
- Catching Or Destruction (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DEP3011809,3 | 1980-03-27 | ||
| DE19803011809 DE3011809A1 (de) | 1980-03-27 | 1980-03-27 | Pyrimidyl-chinazoline, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und ihre verwendung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1156656A true CA1156656A (en) | 1983-11-08 |
Family
ID=6098481
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA000373945A Expired CA1156656A (en) | 1980-03-27 | 1981-03-26 | Process for the preparation of pyrimidyl-chinazolines |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP0037495A1 (show.php) |
| JP (1) | JPS56150088A (show.php) |
| AR (1) | AR227542A1 (show.php) |
| AU (1) | AU6877481A (show.php) |
| CA (1) | CA1156656A (show.php) |
| CS (1) | CS219898B2 (show.php) |
| DD (1) | DD157614A5 (show.php) |
| DE (1) | DE3011809A1 (show.php) |
| DK (1) | DK115581A (show.php) |
| ES (1) | ES500738A0 (show.php) |
| FI (1) | FI810778A7 (show.php) |
| GR (1) | GR71870B (show.php) |
| IL (1) | IL62495A0 (show.php) |
| NO (1) | NO810870L (show.php) |
| PL (2) | PL233882A1 (show.php) |
| PT (1) | PT72724B (show.php) |
| SU (1) | SU1052158A3 (show.php) |
| ZA (1) | ZA812034B (show.php) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6267077A (ja) * | 1985-09-18 | 1987-03-26 | Mitsui Petrochem Ind Ltd | キナゾリン誘導体及び医薬 |
| JPS61140568A (ja) * | 1984-12-14 | 1986-06-27 | Mitsui Petrochem Ind Ltd | キナゾリン誘導体及びそれを有効成分とする血圧降下剤 |
| CN102127057A (zh) * | 2004-03-15 | 2011-07-20 | 武田药品工业株式会社 | 二肽基肽酶抑制剂 |
| WO2006014394A1 (en) | 2004-07-02 | 2006-02-09 | Corcept Therapeutics, Inc. | Modified pyrimidine glucocorticoid receptor modulators |
| PE20141378A1 (es) | 2011-03-18 | 2014-10-12 | Corcept Therapeutics Inc | Moduladores de receptores de glucocorticoides de pirimidina ciclohexilo |
| SG11202011948SA (en) | 2018-06-04 | 2020-12-30 | Corcept Therapeutics Inc | Pyrimidine cyclohexenyl glucocorticoid receptor modulators |
| NZ786586A (en) | 2019-12-11 | 2025-12-19 | Corcept Therapeutics Incorporated | Methods of treating antipsychotic-induced weight gain with miricorilant |
| PH12022553008A1 (en) | 2020-05-06 | 2024-03-04 | Corcept Therapeutics Inc | Formulations of pyrimidine cyclohexyl glucocorticoid receptor modulators |
| CA3182272A1 (en) | 2020-05-06 | 2021-11-11 | Corcept Therapeutics Incorporated | Polymorphs of pyrimidine cyclohexyl glucocorticoid receptor modulators |
| CN116848092A (zh) | 2020-12-21 | 2023-10-03 | 科赛普特治疗公司 | 制备嘧啶环己基糖皮质激素受体调节剂的方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2007656B (en) * | 1977-11-05 | 1982-05-19 | Pfizer Ltd | Therapeutic agents |
-
1980
- 1980-03-27 DE DE19803011809 patent/DE3011809A1/de not_active Withdrawn
- 1980-12-15 GR GR64485A patent/GR71870B/el unknown
-
1981
- 1981-03-13 DK DK115581A patent/DK115581A/da not_active Application Discontinuation
- 1981-03-13 NO NO810870A patent/NO810870L/no unknown
- 1981-03-13 FI FI810778A patent/FI810778A7/fi not_active Application Discontinuation
- 1981-03-20 EP EP81102088A patent/EP0037495A1/de not_active Ceased
- 1981-03-24 PT PT72724A patent/PT72724B/pt unknown
- 1981-03-25 DD DD81228589A patent/DD157614A5/de unknown
- 1981-03-25 SU SU813261941A patent/SU1052158A3/ru active
- 1981-03-25 CS CS812182A patent/CS219898B2/cs unknown
- 1981-03-25 PL PL23388281A patent/PL233882A1/xx unknown
- 1981-03-25 PL PL23032081A patent/PL230320A1/xx unknown
- 1981-03-25 JP JP4257181A patent/JPS56150088A/ja active Pending
- 1981-03-26 AR AR284752A patent/AR227542A1/es active
- 1981-03-26 CA CA000373945A patent/CA1156656A/en not_active Expired
- 1981-03-26 IL IL62495A patent/IL62495A0/xx unknown
- 1981-03-26 ZA ZA00812034A patent/ZA812034B/xx unknown
- 1981-03-26 ES ES500738A patent/ES500738A0/es active Granted
- 1981-03-26 AU AU68774/81A patent/AU6877481A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| GR71870B (show.php) | 1983-07-08 |
| SU1052158A3 (ru) | 1983-10-30 |
| ES8202000A1 (es) | 1982-01-16 |
| AR227542A1 (es) | 1982-11-15 |
| EP0037495A1 (de) | 1981-10-14 |
| DK115581A (da) | 1981-09-28 |
| PL233882A1 (show.php) | 1982-05-10 |
| CS219898B2 (en) | 1983-03-25 |
| DD157614A5 (de) | 1982-11-24 |
| PT72724A (de) | 1981-04-01 |
| PL230320A1 (show.php) | 1982-03-29 |
| DE3011809A1 (de) | 1981-10-01 |
| NO810870L (no) | 1981-09-28 |
| AU6877481A (en) | 1981-10-01 |
| FI810778L (fi) | 1981-09-28 |
| FI810778A7 (fi) | 1981-09-28 |
| PT72724B (de) | 1982-03-24 |
| ZA812034B (en) | 1982-05-26 |
| ES500738A0 (es) | 1982-01-16 |
| JPS56150088A (en) | 1981-11-20 |
| IL62495A0 (en) | 1981-05-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MKEX | Expiry |