CA1133495A - Cis et trans-3-aryloxy-4-hydroxypyrrolidines et derives - Google Patents
Cis et trans-3-aryloxy-4-hydroxypyrrolidines et derivesInfo
- Publication number
- CA1133495A CA1133495A CA343,328A CA343328A CA1133495A CA 1133495 A CA1133495 A CA 1133495A CA 343328 A CA343328 A CA 343328A CA 1133495 A CA1133495 A CA 1133495A
- Authority
- CA
- Canada
- Prior art keywords
- trans
- process according
- pyrrolidinol
- formula
- hydrogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/12—Oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/20—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Psychiatry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US215179A | 1979-01-09 | 1979-01-09 | |
US002,151 | 1979-01-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
CA1133495A true CA1133495A (fr) | 1982-10-12 |
Family
ID=21699450
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA343,328A Expired CA1133495A (fr) | 1979-01-09 | 1980-01-09 | Cis et trans-3-aryloxy-4-hydroxypyrrolidines et derives |
Country Status (9)
Country | Link |
---|---|
JP (1) | JPS5598160A (fr) |
CA (1) | CA1133495A (fr) |
CH (1) | CH643243A5 (fr) |
DE (1) | DE3000625A1 (fr) |
FR (1) | FR2446279B1 (fr) |
GB (1) | GB2040933B (fr) |
IT (1) | IT1127967B (fr) |
MX (1) | MX6634E (fr) |
SE (1) | SE435927B (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE45511B1 (en) | 1976-09-01 | 1982-09-08 | Ciba Geigy Ag | New derivatives of perhydro-aza-heterocycles and processesfor the production thereof |
US4547514A (en) * | 1983-12-05 | 1985-10-15 | A. H. Robins Company, Incorporated | Aryloxy-N-(aminoalkyl)-1-pyrrolidine and piperidine carboxamides and carbothioamides having antiarrhythmic activity |
JPS60178860A (ja) * | 1984-02-24 | 1985-09-12 | Sankyo Co Ltd | 3−メルカプトピロリジンまたはその塩の製法 |
JPS6157552A (ja) * | 1984-08-29 | 1986-03-24 | Toyama Chem Co Ltd | 3−アミノピロリジンまたはその塩の製法 |
DE3813416A1 (de) * | 1988-04-21 | 1989-11-02 | Hoechst Ag | 3,4-dihydroxypyrrolidin-2-on-derivate, verfahren zu ihrer herstellung, diese enthaltende mittel und ihre verwendung sowie die bei der herstellung anfallenden neuen zwischenprodukte |
EP0407701A3 (en) * | 1989-05-15 | 1992-04-22 | Fujisawa Pharmaceutical Co., Ltd. | Antiretroviral pyrroline and pyrrolidine sulfonic acid derivatives |
JP5323063B2 (ja) | 2007-05-31 | 2013-10-23 | 塩野義製薬株式会社 | オキシイミノ化合物およびその使用 |
EP2346820B1 (fr) | 2008-06-11 | 2013-02-13 | Shionogi & Co., Ltd. | Composés oxycarbamoyle et leur utilisation |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR1000308A (fr) * | 1949-05-28 | 1952-02-11 | Basf Ag | Procédé pour la production de 3. 4-dioxypyrrolidines |
FR1000310A (fr) * | 1949-06-18 | 1952-02-11 | Basf Ag | Procédé pour la production de dérivés de pyrrolidine |
FR1532221A (fr) * | 1963-10-22 | 1968-07-12 | Robins Co Inc A H | Procédé de production de n, n-di (aryl monocarbocyclique)-carbamates de 1-(alkylinférieur)-3-pyrrolidyle |
CH521338A (de) * | 1967-03-13 | 1972-04-15 | Robins Co Inc A H | Verfahren zur Herstellung von neuen Pyrrolidinderivaten |
US3577415A (en) * | 1968-12-23 | 1971-05-04 | Robins Co Inc A H | 1-substituted-3-substituted phenoxypyrrolidines |
IE45511B1 (en) * | 1976-09-01 | 1982-09-08 | Ciba Geigy Ag | New derivatives of perhydro-aza-heterocycles and processesfor the production thereof |
-
1980
- 1980-01-03 MX MX808576U patent/MX6634E/es unknown
- 1980-01-07 SE SE8000085A patent/SE435927B/sv not_active IP Right Cessation
- 1980-01-08 CH CH10280A patent/CH643243A5/fr not_active IP Right Cessation
- 1980-01-08 IT IT67020/80A patent/IT1127967B/it active
- 1980-01-08 FR FR8000272A patent/FR2446279B1/fr not_active Expired
- 1980-01-09 DE DE19803000625 patent/DE3000625A1/de active Granted
- 1980-01-09 CA CA343,328A patent/CA1133495A/fr not_active Expired
- 1980-01-09 JP JP123280A patent/JPS5598160A/ja active Granted
- 1980-01-09 GB GB8000709A patent/GB2040933B/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
FR2446279B1 (fr) | 1985-10-31 |
CH643243A5 (fr) | 1984-05-30 |
MX6634E (es) | 1985-09-12 |
IT8067020A0 (it) | 1980-01-08 |
DE3000625C2 (fr) | 1989-04-20 |
JPS5598160A (en) | 1980-07-25 |
GB2040933B (en) | 1983-07-20 |
SE435927B (sv) | 1984-10-29 |
DE3000625A1 (de) | 1980-07-17 |
IT1127967B (it) | 1986-05-28 |
SE8000085L (sv) | 1980-08-26 |
JPS648621B2 (fr) | 1989-02-14 |
FR2446279A1 (fr) | 1980-08-08 |
GB2040933A (en) | 1980-09-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MKEX | Expiry |