CA1050028A - N-substituted 1,2,4-triazoles - Google Patents

N-substituted 1,2,4-triazoles

Info

Publication number
CA1050028A
CA1050028A CA222,366A CA222366A CA1050028A CA 1050028 A CA1050028 A CA 1050028A CA 222366 A CA222366 A CA 222366A CA 1050028 A CA1050028 A CA 1050028A
Authority
CA
Canada
Prior art keywords
triazole
compound
whenever prepared
obvious chemical
carboxamido
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA222,366A
Other languages
English (en)
French (fr)
Inventor
Joseph T. Witkowski
Roland K. Robins
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Valeant Pharmaceuticals International Inc USA
Original Assignee
ICN Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/452,213 external-priority patent/US3991078A/en
Application filed by ICN Pharmaceuticals Inc filed Critical ICN Pharmaceuticals Inc
Application granted granted Critical
Publication of CA1050028A publication Critical patent/CA1050028A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
    • C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/056—Triazole or tetrazole radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
CA222,366A 1974-03-18 1975-03-18 N-substituted 1,2,4-triazoles Expired CA1050028A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/452,213 US3991078A (en) 1971-06-01 1974-03-18 N-substituted 1,2,4-triazoles

Publications (1)

Publication Number Publication Date
CA1050028A true CA1050028A (en) 1979-03-06

Family

ID=23795554

Family Applications (1)

Application Number Title Priority Date Filing Date
CA222,366A Expired CA1050028A (en) 1974-03-18 1975-03-18 N-substituted 1,2,4-triazoles

Country Status (13)

Country Link
JP (2) JPS50154252A (de)
AR (1) AR207138A1 (de)
BE (2) BE826777R (de)
CA (1) CA1050028A (de)
DE (1) DE2511829A1 (de)
DK (1) DK154343C (de)
ES (1) ES435690A2 (de)
FR (1) FR2264533B2 (de)
GB (1) GB1490272A (de)
NL (1) NL7503209A (de)
SE (1) SE7502994L (de)
YU (1) YU42138B (de)
ZA (1) ZA751663B (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02106421U (de) * 1989-02-07 1990-08-23
RU2624018C2 (ru) * 2016-09-26 2017-06-30 Федеральное государственное бюджетное учреждение науки Институт биоорганической химии им. академиков М.М. Шемякина и Ю.А. Овчинникова РАН (ИБХ РАН) Амид 5-(тетрагидрофуран-2-ил)-1,2,4-триазол-3-карбоновой кислоты, обладающий противовирусной активностью, и способ его получения

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3798209A (en) * 1971-06-01 1974-03-19 Icn Pharmaceuticals 1,2,4-triazole nucleosides

Also Published As

Publication number Publication date
SE7502994L (de) 1975-09-19
YU42138B (en) 1988-06-30
AR207138A1 (es) 1976-09-15
ES435690A2 (es) 1977-02-01
GB1490272A (en) 1977-10-26
JPS50154252A (de) 1975-12-12
DK154343C (da) 1989-05-22
DE2511829C2 (de) 1989-06-22
DE2511829A1 (de) 1975-09-25
YU65875A (en) 1983-01-21
BE826777R (fr) 1975-07-16
FR2264533B2 (de) 1978-09-01
DK106475A (de) 1975-09-19
DK154343B (da) 1988-11-07
FR2264533A2 (de) 1975-10-17
ZA751663B (en) 1976-02-25
BE904149Q (fr) 1986-05-15
AU7914475A (en) 1976-09-23
NL7503209A (nl) 1975-09-22
JPS6133822B2 (de) 1986-08-04
JPS59144773A (ja) 1984-08-18

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