BRPI0920145B8 - compostos de tioamida, método de produção e método de uso dos mesmos - Google Patents

compostos de tioamida, método de produção e método de uso dos mesmos

Info

Publication number
BRPI0920145B8
BRPI0920145B8 BRPI0920145A BRPI0920145A BRPI0920145B8 BR PI0920145 B8 BRPI0920145 B8 BR PI0920145B8 BR PI0920145 A BRPI0920145 A BR PI0920145A BR PI0920145 A BRPI0920145 A BR PI0920145A BR PI0920145 B8 BRPI0920145 B8 BR PI0920145B8
Authority
BR
Brazil
Prior art keywords
production
thioamide compounds
thioamide
formula
compounds
Prior art date
Application number
BRPI0920145A
Other languages
English (en)
Portuguese (pt)
Inventor
Ik Lee Hyoung
Patrick Le Hir De Fallois Loïc
Reid Timmons Philip
Original Assignee
Merial Ltd
Merial Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd, Merial Inc filed Critical Merial Ltd
Publication of BRPI0920145A2 publication Critical patent/BRPI0920145A2/pt
Publication of BRPI0920145B1 publication Critical patent/BRPI0920145B1/pt
Publication of BRPI0920145B8 publication Critical patent/BRPI0920145B8/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/16Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C07D249/18Benzotriazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41921,2,3-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
BRPI0920145A 2008-10-21 2009-10-20 compostos de tioamida, método de produção e método de uso dos mesmos BRPI0920145B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10711408P 2008-10-21 2008-10-21
US61/107,114 2008-10-21
PCT/US2009/061337 WO2010048191A1 (en) 2008-10-21 2009-10-20 Thioamide compounds, method of making and method of using thereof

Publications (3)

Publication Number Publication Date
BRPI0920145A2 BRPI0920145A2 (pt) 2017-06-06
BRPI0920145B1 BRPI0920145B1 (pt) 2021-03-30
BRPI0920145B8 true BRPI0920145B8 (pt) 2021-05-25

Family

ID=41404569

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0920145A BRPI0920145B8 (pt) 2008-10-21 2009-10-20 compostos de tioamida, método de produção e método de uso dos mesmos

Country Status (15)

Country Link
US (2) US7964621B2 (show.php)
EP (1) EP2358687B9 (show.php)
JP (1) JP5614853B2 (show.php)
KR (2) KR101782311B1 (show.php)
CN (1) CN102239151B (show.php)
AU (1) AU2009307736B2 (show.php)
BR (1) BRPI0920145B8 (show.php)
CA (1) CA2741186C (show.php)
CL (1) CL2011000917A1 (show.php)
EA (1) EA026649B1 (show.php)
ES (1) ES2393965T3 (show.php)
MX (1) MX2011004217A (show.php)
NZ (1) NZ592382A (show.php)
WO (1) WO2010048191A1 (show.php)
ZA (1) ZA201103033B (show.php)

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PT2922845T (pt) 2012-11-20 2018-10-23 Merial Inc Compostos e composições anti-helmínticos e métodos de utilização dos mesmos
CN103073487B (zh) * 2013-01-15 2014-11-19 西华大学 N-双取代硫代乙酰胺类化合物的合成方法
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BR112017024773A2 (pt) 2015-05-20 2018-11-06 Merial, Inc. compostos depsipeptídeos anti-helmínticos
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CN113260419A (zh) 2018-11-20 2021-08-13 勃林格殷格翰动物保健美国公司 吲唑基氰基乙基氨基化合物、其组合物、其制备方法和其使用方法
KR102281492B1 (ko) * 2018-12-24 2021-07-26 동인당제약 주식회사 세벨라머 함유 경구투여용 현탁제 조성물 및 그 제조방법
KR20220002890A (ko) 2019-03-19 2022-01-07 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 아자-벤조티오펜 및 아자-벤조푸란 화합물
KR20230028268A (ko) 2020-05-29 2023-02-28 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 구충성 헤테로시클릭 화합물
CN111781291A (zh) * 2020-06-23 2020-10-16 广西壮族自治区水产科学研究院 一种水中13种大环内酯类抗生素的高分辨质谱检测方法
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JP2025507585A (ja) 2022-02-17 2025-03-21 ベーリンガー インゲルハイム フェトメディカ ゲーエムベーハー 流体製品メーラーを提供する方法及びシステム
CN117837424A (zh) * 2024-02-04 2024-04-09 黄淮学院 一种控制农作物灰飞虱的方法
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Also Published As

Publication number Publication date
CN102239151A (zh) 2011-11-09
AU2009307736B2 (en) 2015-02-05
CN102239151B (zh) 2014-07-02
EP2358687B1 (en) 2012-09-19
KR101782311B1 (ko) 2017-09-27
US7964621B2 (en) 2011-06-21
EA201100666A1 (ru) 2011-12-30
US20100130565A1 (en) 2010-05-27
US20110190231A1 (en) 2011-08-04
KR101782308B1 (ko) 2017-09-27
ES2393965T9 (es) 2013-07-19
BRPI0920145B1 (pt) 2021-03-30
ZA201103033B (en) 2012-02-29
MX2011004217A (es) 2011-06-20
EA026649B1 (ru) 2017-05-31
US8314146B2 (en) 2012-11-20
WO2010048191A1 (en) 2010-04-29
CA2741186A1 (en) 2010-04-29
AU2009307736A1 (en) 2010-04-29
EP2358687A1 (en) 2011-08-24
BRPI0920145A2 (pt) 2017-06-06
KR20110071140A (ko) 2011-06-28
CA2741186C (en) 2016-07-19
EP2358687B9 (en) 2013-04-17
CL2011000917A1 (es) 2011-09-16
ES2393965T3 (es) 2013-01-03
JP2012506441A (ja) 2012-03-15
NZ592382A (en) 2013-03-28
JP5614853B2 (ja) 2014-10-29
KR20170003704A (ko) 2017-01-09

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B25A Requested transfer of rights approved

Owner name: MERIAL, INC. (US)

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

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B16C Correction of notification of the grant [chapter 16.3 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 20/10/2009 OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF

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Free format text: ANULADA A PUBLICACAO CODIGO 16.3 NA RPI NO 2629 DE 25/05/2021 POR TER SIDO INDEVIDA.

B25A Requested transfer of rights approved

Owner name: BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC. (US)