BRPI0916270A2 - processo assimétrico para a produção de 2-amino-tiazolonas substituídas - Google Patents

processo assimétrico para a produção de 2-amino-tiazolonas substituídas

Info

Publication number
BRPI0916270A2
BRPI0916270A2 BRPI0916270A BRPI0916270A BRPI0916270A2 BR PI0916270 A2 BRPI0916270 A2 BR PI0916270A2 BR PI0916270 A BRPI0916270 A BR PI0916270A BR PI0916270 A BRPI0916270 A BR PI0916270A BR PI0916270 A2 BRPI0916270 A2 BR PI0916270A2
Authority
BR
Brazil
Prior art keywords
thiazolones
amino
substituted
production
asymmetric process
Prior art date
Application number
BRPI0916270A
Other languages
English (en)
Inventor
Faul Margaret
Caille Seb
Cui Sheng
Wang Xiang
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of BRPI0916270A2 publication Critical patent/BRPI0916270A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/54Nitrogen and either oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Steroid Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BRPI0916270A 2008-07-29 2009-07-28 processo assimétrico para a produção de 2-amino-tiazolonas substituídas BRPI0916270A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8454908P 2008-07-29 2008-07-29
PCT/US2009/051929 WO2010014586A1 (en) 2008-07-29 2009-07-28 Asymmetric process for making substituted 2-amino-thiazolones

Publications (1)

Publication Number Publication Date
BRPI0916270A2 true BRPI0916270A2 (pt) 2018-10-16

Family

ID=41020998

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0916270A BRPI0916270A2 (pt) 2008-07-29 2009-07-28 processo assimétrico para a produção de 2-amino-tiazolonas substituídas

Country Status (21)

Country Link
US (2) US8501954B2 (pt)
EP (1) EP2321290B1 (pt)
JP (1) JP2011529896A (pt)
KR (1) KR20110048520A (pt)
CN (1) CN102112454B (pt)
AU (1) AU2009276757A1 (pt)
BR (1) BRPI0916270A2 (pt)
CA (1) CA2730711A1 (pt)
CL (1) CL2011000120A1 (pt)
CY (1) CY1113135T1 (pt)
DK (1) DK2321290T3 (pt)
EA (1) EA019573B1 (pt)
ES (1) ES2386613T3 (pt)
HK (1) HK1154000A1 (pt)
IL (1) IL210562A (pt)
MX (1) MX2011001009A (pt)
PL (1) PL2321290T3 (pt)
PT (1) PT2321290E (pt)
SI (1) SI2321290T1 (pt)
WO (1) WO2010014586A1 (pt)
ZA (1) ZA201100358B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8853420B2 (en) 2008-07-29 2014-10-07 Boehringer Ingelheim International Gmbh Compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005116002A2 (en) * 2004-05-24 2005-12-08 Amgen Inc. Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
JP5204662B2 (ja) 2005-11-22 2013-06-05 アムジエン・インコーポレーテツド 11−β−ヒドロキシステロイドデヒドロゲナーゼ1型の阻害剤
AU2006317070B2 (en) * 2005-11-22 2011-06-23 Amgen, Inc. Catalyzed process of making C-5-substituted heterocyclic inhibitors of 11beta-hydroxy steroid dehydrogenase type 1
US8541593B2 (en) * 2007-06-21 2013-09-24 Amgen Inc. Process for making substituted 2-amino-thiazolones

Also Published As

Publication number Publication date
WO2010014586A1 (en) 2010-02-04
EP2321290A1 (en) 2011-05-18
IL210562A (en) 2013-11-28
US20130345432A1 (en) 2013-12-26
US20110178307A1 (en) 2011-07-21
CL2011000120A1 (es) 2011-06-24
PT2321290E (pt) 2012-08-10
IL210562A0 (en) 2011-03-31
AU2009276757A1 (en) 2010-02-04
ZA201100358B (en) 2011-10-26
PL2321290T3 (pl) 2012-11-30
HK1154000A1 (en) 2012-04-13
EA019573B1 (ru) 2014-04-30
MX2011001009A (es) 2011-04-27
JP2011529896A (ja) 2011-12-15
US8501954B2 (en) 2013-08-06
CN102112454A (zh) 2011-06-29
CA2730711A1 (en) 2010-02-04
CY1113135T1 (el) 2016-04-13
SI2321290T1 (sl) 2012-09-28
CN102112454B (zh) 2013-09-04
EA201170072A1 (ru) 2011-08-30
EP2321290B1 (en) 2012-06-20
KR20110048520A (ko) 2011-05-11
ES2386613T3 (es) 2012-08-23
DK2321290T3 (da) 2012-07-16

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 6A, 7A, 8A E 9A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2495 DE 30-10-2018 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.