BRPI0914531B1 - Método para preparação de polimorfo a de 3-bromo-1-(3-cloro-2-piridinil)-n-[4-ciano-2-metil- 6-[(metilamino)-carbonil]fenil]-1h-pirazol-5-carboxamida - Google Patents

Método para preparação de polimorfo a de 3-bromo-1-(3-cloro-2-piridinil)-n-[4-ciano-2-metil- 6-[(metilamino)-carbonil]fenil]-1h-pirazol-5-carboxamida Download PDF

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Publication number
BRPI0914531B1
BRPI0914531B1 BRPI0914531-1A BRPI0914531A BRPI0914531B1 BR PI0914531 B1 BRPI0914531 B1 BR PI0914531B1 BR PI0914531 A BRPI0914531 A BR PI0914531A BR PI0914531 B1 BRPI0914531 B1 BR PI0914531B1
Authority
BR
Brazil
Prior art keywords
polymorph
compound
water
mixture
solvent
Prior art date
Application number
BRPI0914531-1A
Other languages
English (en)
Portuguese (pt)
Inventor
Mathew Richard Oberholzer
Original Assignee
Fmc Corporation
Fmc Agro Singapore Pte. Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fmc Corporation, Fmc Agro Singapore Pte. Ltd. filed Critical Fmc Corporation
Publication of BRPI0914531A2 publication Critical patent/BRPI0914531A2/pt
Publication of BRPI0914531B1 publication Critical patent/BRPI0914531B1/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BRPI0914531-1A 2008-11-14 2009-11-11 Método para preparação de polimorfo a de 3-bromo-1-(3-cloro-2-piridinil)-n-[4-ciano-2-metil- 6-[(metilamino)-carbonil]fenil]-1h-pirazol-5-carboxamida BRPI0914531B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11462908P 2008-11-14 2008-11-14
US61/114,629 2008-11-14
PCT/US2009/063991 WO2010056720A1 (en) 2008-11-14 2009-11-11 Method for preparing a non-hydratable crystal form

Publications (2)

Publication Number Publication Date
BRPI0914531A2 BRPI0914531A2 (pt) 2015-08-04
BRPI0914531B1 true BRPI0914531B1 (pt) 2021-01-05

Family

ID=42044745

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0914531-1A BRPI0914531B1 (pt) 2008-11-14 2009-11-11 Método para preparação de polimorfo a de 3-bromo-1-(3-cloro-2-piridinil)-n-[4-ciano-2-metil- 6-[(metilamino)-carbonil]fenil]-1h-pirazol-5-carboxamida

Country Status (19)

Country Link
US (1) US8410278B2 (enExample)
EP (1) EP2350046B8 (enExample)
JP (1) JP5570520B2 (enExample)
KR (1) KR101693901B1 (enExample)
CN (1) CN102216284B (enExample)
AU (1) AU2009314203B2 (enExample)
BR (1) BRPI0914531B1 (enExample)
CA (1) CA2737932C (enExample)
DK (1) DK2350046T3 (enExample)
ES (1) ES2445699T3 (enExample)
IL (1) IL211727A (enExample)
MX (1) MX2011004950A (enExample)
MY (1) MY150568A (enExample)
PL (1) PL2350046T3 (enExample)
RS (1) RS53150B (enExample)
RU (1) RU2500676C2 (enExample)
UA (1) UA101395C2 (enExample)
WO (1) WO2010056720A1 (enExample)
ZA (1) ZA201101855B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI325302B (en) 2001-08-13 2010-06-01 Du Pont Benzoxazinone compounds
TWI283164B (en) 2001-09-21 2007-07-01 Du Pont Anthranilamide arthropodicide treatment
BR112022025066A2 (pt) * 2020-06-08 2023-03-07 Adama Makhteshim Ltd Processo de preparação de antranilamidas
WO2023095161A1 (en) * 2021-11-24 2023-06-01 Natco Pharma Limited An improved process for the preparation of crystalline form-a of cyantraniliprole
AR131889A1 (es) * 2023-02-21 2025-05-14 Upl Ltd Un proceso para la preparación de un compuesto de antranilamida e intermedios del mismo
PY2419787A (es) 2023-03-15 2024-11-28 Adama Makhteshim Ltd Composición en suspensión acuosa de cianraniliprol y acetamiprid
WO2025104727A1 (en) * 2023-11-16 2025-05-22 Adama Makhteshim Ltd. Solid state forms of cyantraniliprole and uses thereof
CN118146190A (zh) * 2024-02-01 2024-06-07 南开大学 溴氰虫酰胺的新晶型及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0003154D0 (en) * 2000-02-12 2000-04-05 Astrazeneca Uk Ltd Novel compounds
CA2461080A1 (en) * 2001-09-25 2003-04-03 Pharmacia Corporation Solid-state forms of n-(2-hydroxyacetyl)-5-(4-piperidyl)-4-(4-pyrimidinyl)-3-(4-chlorophenyl)pyrazole
VN23181A1 (en) * 2003-01-28 2010-07-26 Du Pont Cyano anthranilamide insecticides
TWI363756B (en) * 2004-12-07 2012-05-11 Du Pont Method for preparing n-phenylpyrazole-1-carboxamides
JP5449669B2 (ja) * 2006-12-14 2014-03-19 石原産業株式会社 有害生物防除組成物
JP5551371B2 (ja) * 2008-03-24 2014-07-16 石原産業株式会社 有害生物防除用固形組成物

Also Published As

Publication number Publication date
KR101693901B1 (ko) 2017-01-06
MX2011004950A (es) 2011-05-30
DK2350046T3 (en) 2014-03-24
RS53150B (sr) 2014-06-30
JP2012508747A (ja) 2012-04-12
RU2500676C2 (ru) 2013-12-10
UA101395C2 (ru) 2013-03-25
IL211727A0 (en) 2011-06-30
RU2011123800A (ru) 2012-12-20
EP2350046A1 (en) 2011-08-03
PL2350046T3 (pl) 2014-05-30
WO2010056720A1 (en) 2010-05-20
CA2737932A1 (en) 2010-05-20
CN102216284B (zh) 2014-02-19
EP2350046B1 (en) 2014-01-01
AU2009314203B2 (en) 2015-01-22
EP2350046B8 (en) 2014-04-02
CA2737932C (en) 2016-05-17
AU2009314203A1 (en) 2010-05-20
IL211727A (en) 2014-02-27
CN102216284A (zh) 2011-10-12
US20110184183A1 (en) 2011-07-28
MY150568A (en) 2014-01-30
US8410278B2 (en) 2013-04-02
ZA201101855B (en) 2012-05-30
KR20110082632A (ko) 2011-07-19
JP5570520B2 (ja) 2014-08-13
ES2445699T3 (es) 2014-03-04
BRPI0914531A2 (pt) 2015-08-04

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B25A Requested transfer of rights approved

Owner name: FMC CORPORATION (US)

B06T Formal requirements before examination [chapter 6.20 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07G Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette]
B25K Entry of change of name and/or headquarter and transfer of application, patent and certificate of addition of invention: republication

Owner name: FMC CORPORATION (US) ; FMC AGRO SINGAPORE PTE. LTD. (SG)

Free format text: RETIFICACAO DO DESPACHO 25.1 ? TRANSFERENCIA DE TITULAR PUBLICADO NA RPI NO 2486, DE 28/08/2018, QUANTO AO ITEM 71 - DEPOSITANTE.ONDE SE LE: FMC CORPORATIONLEIA-SE: FMC CORPORATION E FMC AGRO SINGAPORE PTE. LTD.

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 05/01/2021, OBSERVADAS AS CONDICOES LEGAIS.

B25G Requested change of headquarter approved

Owner name: FMC CORPORATION (US) ; FMC AGRO SINGAPORE PTE. LTD. (SG)

B25A Requested transfer of rights approved

Owner name: FMC CORPORATION (US) ; FMC IP TECHNOLOGY GMBH (CH)