BRPI0817445A2 - composto, composição farmacêutica, método de tratamento, e, processo para preparar um composto - Google Patents
composto, composição farmacêutica, método de tratamento, e, processo para preparar um compostoInfo
- Publication number
- BRPI0817445A2 BRPI0817445A2 BRPI0817445A BRPI0817445A BRPI0817445A2 BR PI0817445 A2 BRPI0817445 A2 BR PI0817445A2 BR PI0817445 A BRPI0817445 A BR PI0817445A BR PI0817445 A BRPI0817445 A BR PI0817445A BR PI0817445 A2 BRPI0817445 A2 BR PI0817445A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- preparing
- treatment
- pharmaceutical composition
- pharmaceutical
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Psychiatry (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US97586507P | 2007-09-28 | 2007-09-28 | |
PCT/US2008/077626 WO2009045831A1 (en) | 2007-09-28 | 2008-09-25 | Glycogen phosphorylase inhibitor compound and pharmaceutical composition thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0817445A2 true BRPI0817445A2 (pt) | 2015-10-27 |
Family
ID=40120238
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0817445A BRPI0817445A2 (pt) | 2007-09-28 | 2008-09-25 | composto, composição farmacêutica, método de tratamento, e, processo para preparar um composto |
Country Status (16)
Country | Link |
---|---|
US (1) | US20100234433A1 (pt) |
EP (1) | EP2197845A1 (pt) |
JP (1) | JP2010540553A (pt) |
KR (1) | KR20100075568A (pt) |
CN (1) | CN101861303A (pt) |
AU (1) | AU2008309004A1 (pt) |
BR (1) | BRPI0817445A2 (pt) |
CA (1) | CA2701020A1 (pt) |
CO (1) | CO6321157A2 (pt) |
CR (1) | CR11397A (pt) |
DO (1) | DOP2010000088A (pt) |
EA (1) | EA201000392A1 (pt) |
MA (1) | MA31775B1 (pt) |
MX (1) | MX2010003442A (pt) |
WO (1) | WO2009045831A1 (pt) |
ZA (1) | ZA201002182B (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011107494A1 (de) | 2010-03-03 | 2011-09-09 | Sanofi | Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
WO2013037390A1 (en) | 2011-09-12 | 2013-03-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
EP2760862B1 (en) | 2011-09-27 | 2015-10-21 | Sanofi | 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2236757T3 (es) * | 1995-11-24 | 2005-07-16 | Glaxosmithkline S.P.A. | Derivados de quinolina. |
US20070249670A1 (en) * | 2004-11-09 | 2007-10-25 | Smithkline Beecham Corporation | Glycogen Phosphorylase Inhibitor Compounds and Pharmaceutical Compositions Thereof |
-
2008
- 2008-09-25 BR BRPI0817445A patent/BRPI0817445A2/pt not_active IP Right Cessation
- 2008-09-25 CN CN200880116662A patent/CN101861303A/zh active Pending
- 2008-09-25 EA EA201000392A patent/EA201000392A1/ru unknown
- 2008-09-25 KR KR1020107009325A patent/KR20100075568A/ko not_active Application Discontinuation
- 2008-09-25 AU AU2008309004A patent/AU2008309004A1/en not_active Abandoned
- 2008-09-25 WO PCT/US2008/077626 patent/WO2009045831A1/en active Application Filing
- 2008-09-25 MX MX2010003442A patent/MX2010003442A/es not_active Application Discontinuation
- 2008-09-25 JP JP2010527131A patent/JP2010540553A/ja not_active Withdrawn
- 2008-09-25 CA CA2701020A patent/CA2701020A1/en not_active Abandoned
- 2008-09-25 EP EP08836469A patent/EP2197845A1/en not_active Withdrawn
- 2008-09-25 US US12/677,855 patent/US20100234433A1/en not_active Abandoned
-
2010
- 2010-03-19 DO DO2010000088A patent/DOP2010000088A/es unknown
- 2010-03-26 CO CO10036282A patent/CO6321157A2/es unknown
- 2010-03-26 ZA ZA2010/02182A patent/ZA201002182B/en unknown
- 2010-04-14 MA MA32770A patent/MA31775B1/fr unknown
- 2010-04-28 CR CR11397A patent/CR11397A/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP2197845A1 (en) | 2010-06-23 |
CN101861303A (zh) | 2010-10-13 |
ZA201002182B (en) | 2011-05-25 |
CO6321157A2 (es) | 2011-09-20 |
EA201000392A1 (ru) | 2010-10-29 |
US20100234433A1 (en) | 2010-09-16 |
AU2008309004A1 (en) | 2009-04-09 |
DOP2010000088A (es) | 2010-07-15 |
CA2701020A1 (en) | 2009-04-09 |
MA31775B1 (fr) | 2010-10-01 |
MX2010003442A (es) | 2010-04-21 |
WO2009045831A1 (en) | 2009-04-09 |
JP2010540553A (ja) | 2010-12-24 |
CR11397A (es) | 2010-05-24 |
KR20100075568A (ko) | 2010-07-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 4A, 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |