BRPI0611555A2 - composição de metformina transmucosa oral, processo para produzir uma composição transmucosa oral de metformina, uso da composição e método de tratamento de diabetes - Google Patents
composição de metformina transmucosa oral, processo para produzir uma composição transmucosa oral de metformina, uso da composição e método de tratamento de diabetes Download PDFInfo
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- BRPI0611555A2 BRPI0611555A2 BRPI0611555-1A BRPI0611555A BRPI0611555A2 BR PI0611555 A2 BRPI0611555 A2 BR PI0611555A2 BR PI0611555 A BRPI0611555 A BR PI0611555A BR PI0611555 A2 BRPI0611555 A2 BR PI0611555A2
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- metformin
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Zoology (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Reproductive Health (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66647505P | 2005-03-30 | 2005-03-30 | |
| US60/666,475 | 2005-03-30 | ||
| PCT/CA2006/000472 WO2006102752A1 (en) | 2005-03-30 | 2006-03-30 | Compositions for oral transmucosal delivery of metformin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0611555A2 true BRPI0611555A2 (pt) | 2010-09-21 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0611555-1A BRPI0611555A2 (pt) | 2005-03-30 | 2006-03-30 | composição de metformina transmucosa oral, processo para produzir uma composição transmucosa oral de metformina, uso da composição e método de tratamento de diabetes |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20090069437A1 (enExample) |
| EP (1) | EP1863465A4 (enExample) |
| JP (1) | JP2008534523A (enExample) |
| AR (1) | AR052960A1 (enExample) |
| AU (1) | AU2006228949A1 (enExample) |
| BR (1) | BRPI0611555A2 (enExample) |
| CA (1) | CA2603450A1 (enExample) |
| CR (1) | CR9363A (enExample) |
| IL (1) | IL185931A0 (enExample) |
| MX (1) | MX2007012047A (enExample) |
| NZ (1) | NZ560990A (enExample) |
| PE (1) | PE20061245A1 (enExample) |
| RU (2) | RU2409357C2 (enExample) |
| UY (1) | UY29445A1 (enExample) |
| WO (1) | WO2006102752A1 (enExample) |
| ZA (1) | ZA200708834B (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009080025A1 (en) * | 2007-12-20 | 2009-07-02 | Fertin Pharma A/S | Compressed chewing gum comprising metformin |
| WO2009090210A2 (en) * | 2008-01-16 | 2009-07-23 | Janssen Pharmaceutica Nv | Combination of metformin and an mtp inhibitor |
| CA2638240C (en) * | 2008-08-29 | 2010-02-02 | Alexander Macgregor | Method of treating dysglycemia and glucose excursions |
| CN102316872B (zh) * | 2008-11-26 | 2016-12-21 | 萨蒂奥根制药公司 | 治疗肥胖症和糖尿病的胆汁酸再循环抑制剂 |
| EP2445494A4 (en) * | 2009-06-24 | 2012-12-12 | Univ Koebenhavn | TREATMENT OF INSULIN RESISTANCE AND OBESITY BY STIMULATING GLP-1 RELEASE |
| WO2011051974A1 (en) * | 2009-10-29 | 2011-05-05 | Nutracryst Therapeutics Private Limited | Metformin and a-amino acids |
| EP3593802A3 (en) | 2010-05-26 | 2020-03-25 | Satiogen Pharmaceuticals, Inc. | Bile acid recycling inhibitors and satiogens for treatment of diabetes, obesity, and inflammatory gastrointestinal conditions |
| EA030839B1 (ru) | 2011-10-28 | 2018-10-31 | ЛУМЕНА ФАРМАСЬЮТИКАЛС ЭлЭлСи | Ингибиторы рециклинга желчных кислот при лечении холестатических заболеваний печени у детей |
| WO2013063526A1 (en) | 2011-10-28 | 2013-05-02 | Lumena Pharmaceuticals, Inc. | Bile acid recycling inhibitors for treatment of hypercholemia and cholestatic liver disease |
| EP3696281A1 (en) * | 2019-02-13 | 2020-08-19 | Johann Wolfgang Goethe-Universität Frankfurt am Main | Arginase as biomarker and drug target for pcos |
| WO2020227344A1 (en) * | 2019-05-06 | 2020-11-12 | The Regents Of The University Of California | Chloride intracellular channel 1 for regulation of food intake |
Family Cites Families (17)
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|---|---|---|---|---|
| DK161428C (da) * | 1985-05-10 | 1991-12-16 | Fertin Lab As | Fast, oralt cariesmodvirkende middel |
| DK365389D0 (da) * | 1989-07-24 | 1989-07-24 | Fertin Lab As | Antifungalt tyggegummipraeparat |
| US20030095925A1 (en) * | 1997-10-01 | 2003-05-22 | Dugger Harry A. | Buccal, polar and non-polar spray or capsule containing drugs for treating metabolic disorders |
| FR2775188B1 (fr) * | 1998-02-23 | 2001-03-09 | Lipha | Forme galenique a liberation immediate ou liberation prolongee administrable par voie orale comprenant un agent promoteur d'absorption et utilisation de cet agent promoteur d'absorption |
| US6099859A (en) * | 1998-03-20 | 2000-08-08 | Andrx Pharmaceuticals, Inc. | Controlled release oral tablet having a unitary core |
| WO1999055320A1 (en) * | 1998-04-29 | 1999-11-04 | Sumitomo Pharmaceuticals Co., Ltd. | Oral formulation comprising biguanide and an organic acid |
| DK0974356T3 (da) * | 1998-07-15 | 2003-10-27 | Merck Sante Sas | Tabletter omfattende en kombination af metformin og glibenclamid |
| US6099862A (en) * | 1998-08-31 | 2000-08-08 | Andrx Corporation | Oral dosage form for the controlled release of a biguanide and sulfonylurea |
| US6344222B1 (en) * | 1998-09-03 | 2002-02-05 | Jsr Llc | Medicated chewing gum delivery system for nicotine |
| US6312665B1 (en) * | 1998-12-21 | 2001-11-06 | Generex Pharmaceuticals Incorporated | Aerosol formulations for buccal and pulmonary application |
| US6432383B1 (en) * | 2000-03-30 | 2002-08-13 | Generex Pharmaceuticals Incorporated | Method for administering insulin |
| BR0115390A (pt) * | 2000-11-03 | 2004-02-25 | Andrx Corp | Formulações para liberação controlada de metformina, liberação controlada da forma farmacêutica oral, método de diminuição dos nìveis de glicose sanguìnea, uso da forma farmacêutica |
| ITMI20011337A1 (it) * | 2001-06-26 | 2002-12-26 | Farmatron Ltd | Composizioni farmaceutiche orali a rilascio modificato del principio attivo |
| ITFI20010230A1 (it) * | 2001-11-29 | 2003-05-29 | Menarini Int Operations Lu Sa | Composizioni farmaceutiche per il trattamento del diabete mellito di tipo ii |
| KR20100137023A (ko) * | 2002-09-20 | 2010-12-29 | 안드렉스 랩스 엘엘씨 | 약제학적 정제 |
| US20040253307A1 (en) * | 2003-02-04 | 2004-12-16 | Brian Hague | Sugar-free oral transmucosal solid dosage forms and uses thereof |
| WO2005041926A1 (en) * | 2003-10-31 | 2005-05-12 | Alza Corporation | Compositions and dosage forms for enhanced absorption of 3-amino-n-butyl-phosphinic acid |
-
2006
- 2006-03-29 UY UY29445A patent/UY29445A1/es not_active Application Discontinuation
- 2006-03-29 PE PE2006000346A patent/PE20061245A1/es not_active Application Discontinuation
- 2006-03-30 BR BRPI0611555-1A patent/BRPI0611555A2/pt not_active IP Right Cessation
- 2006-03-30 AU AU2006228949A patent/AU2006228949A1/en not_active Abandoned
- 2006-03-30 EP EP06721733A patent/EP1863465A4/en not_active Withdrawn
- 2006-03-30 MX MX2007012047A patent/MX2007012047A/es not_active Application Discontinuation
- 2006-03-30 AR ARP060101262A patent/AR052960A1/es not_active Application Discontinuation
- 2006-03-30 US US11/887,284 patent/US20090069437A1/en not_active Abandoned
- 2006-03-30 RU RU2007139886/15A patent/RU2409357C2/ru not_active IP Right Cessation
- 2006-03-30 JP JP2008503334A patent/JP2008534523A/ja not_active Withdrawn
- 2006-03-30 WO PCT/CA2006/000472 patent/WO2006102752A1/en not_active Ceased
- 2006-03-30 CA CA002603450A patent/CA2603450A1/en not_active Abandoned
- 2006-03-30 NZ NZ560990A patent/NZ560990A/en not_active IP Right Cessation
-
2007
- 2007-09-04 CR CR9363A patent/CR9363A/es not_active Application Discontinuation
- 2007-09-11 IL IL185931A patent/IL185931A0/en unknown
- 2007-10-16 ZA ZA200708834A patent/ZA200708834B/xx unknown
-
2010
- 2010-09-20 RU RU2010139163/15A patent/RU2010139163A/ru unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2007139886A (ru) | 2009-05-10 |
| JP2008534523A (ja) | 2008-08-28 |
| RU2010139163A (ru) | 2012-03-27 |
| US20090069437A1 (en) | 2009-03-12 |
| AU2006228949A1 (en) | 2006-10-05 |
| EP1863465A1 (en) | 2007-12-12 |
| ZA200708834B (en) | 2008-11-26 |
| WO2006102752A1 (en) | 2006-10-05 |
| NZ560990A (en) | 2009-02-28 |
| RU2409357C2 (ru) | 2011-01-20 |
| UY29445A1 (es) | 2006-10-02 |
| MX2007012047A (es) | 2007-12-12 |
| CR9363A (es) | 2008-02-12 |
| IL185931A0 (en) | 2008-02-09 |
| EP1863465A4 (en) | 2010-12-15 |
| AR052960A1 (es) | 2007-04-11 |
| PE20061245A1 (es) | 2007-01-06 |
| CA2603450A1 (en) | 2006-10-05 |
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Legal Events
| Date | Code | Title | Description |
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| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE 7A, ANUIDADE(S). |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2212 DE 28/05/2013. |