BRPI0606644A2 - derivados de 4-carboxamida tiazola - Google Patents
derivados de 4-carboxamida tiazolaInfo
- Publication number
- BRPI0606644A2 BRPI0606644A2 BRPI0606644-5A BRPI0606644A BRPI0606644A2 BR PI0606644 A2 BRPI0606644 A2 BR PI0606644A2 BR PI0606644 A BRPI0606644 A BR PI0606644A BR PI0606644 A2 BRPI0606644 A2 BR PI0606644A2
- Authority
- BR
- Brazil
- Prior art keywords
- carboxamide
- thiazole derivatives
- derivatives
- carboxamide thiazole
- tiazola
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Ophthalmology & Optometry (AREA)
- Psychology (AREA)
- Urology & Nephrology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
DERIVADOS DE 4-CARBOXAMIDA TIAZOLA. A presente invenção refere-se a novos derivados de 4-carbo-xamida tiazola da fórmula geral (I) e métodos para o preparo dos mesmos, compostos os quais são usados como antagonistas do receptor de glutamato metabotrópico: em que R^ 1^ a R^ 4^ são conforme definido na especificação.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP05100203 | 2005-01-14 | ||
PCT/EP2006/000090 WO2006074884A1 (en) | 2005-01-14 | 2006-01-09 | Thiazole-4-carboxamide derivatives as mglur5 antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0606644A2 true BRPI0606644A2 (pt) | 2009-07-14 |
Family
ID=35985686
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0606644-5A BRPI0606644A2 (pt) | 2005-01-14 | 2006-01-09 | derivados de 4-carboxamida tiazola |
Country Status (19)
Country | Link |
---|---|
US (1) | US7678815B2 (pt) |
EP (1) | EP1844044B1 (pt) |
JP (1) | JP4966866B2 (pt) |
KR (1) | KR100905810B1 (pt) |
CN (1) | CN101137653B (pt) |
AR (1) | AR052558A1 (pt) |
AT (1) | ATE474839T1 (pt) |
AU (1) | AU2006205920B2 (pt) |
BR (1) | BRPI0606644A2 (pt) |
CA (1) | CA2593439C (pt) |
DE (1) | DE602006015607D1 (pt) |
ES (1) | ES2346685T3 (pt) |
IL (1) | IL184427A (pt) |
MX (1) | MX2007008410A (pt) |
NO (1) | NO20073663L (pt) |
RU (1) | RU2007125622A (pt) |
TW (1) | TW200637550A (pt) |
WO (1) | WO2006074884A1 (pt) |
ZA (1) | ZA200705670B (pt) |
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JP2009521426A (ja) * | 2005-12-23 | 2009-06-04 | アストラゼネカ・アクチエボラーグ | ヘテロ環gaba−bモジュレーター |
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WO2009078432A1 (ja) * | 2007-12-18 | 2009-06-25 | Taisho Pharmaceutical Co., Ltd. | 1-アルキル-4-アミノ-1h-ピラゾール-3-カルボキサミド化合物 |
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EP1581525A2 (en) * | 2002-08-09 | 2005-10-05 | AstraZeneca AB | Compounds having an activity at metabotropic glutamate receptors |
WO2004014881A2 (en) * | 2002-08-09 | 2004-02-19 | Astra Zeneca Ab | '1,2,4'oxadiazoles as modulators of metabotropic glutamate receptor-5 |
AU2004226450A1 (en) * | 2003-03-26 | 2004-10-14 | Merck & Co. Inc. | Benzamide modulators of metabotropic glutamate receptors |
WO2006008545A2 (en) * | 2004-07-22 | 2006-01-26 | Astex Therapeutics Limited | Thiazole and isothiazole derivatives as protein kinase inhibitors |
-
2006
- 2006-01-09 AU AU2006205920A patent/AU2006205920B2/en not_active Ceased
- 2006-01-09 EP EP06701375A patent/EP1844044B1/en not_active Not-in-force
- 2006-01-09 CN CN2006800079746A patent/CN101137653B/zh not_active Expired - Fee Related
- 2006-01-09 DE DE602006015607T patent/DE602006015607D1/de active Active
- 2006-01-09 CA CA2593439A patent/CA2593439C/en not_active Expired - Fee Related
- 2006-01-09 JP JP2007550737A patent/JP4966866B2/ja not_active Expired - Fee Related
- 2006-01-09 MX MX2007008410A patent/MX2007008410A/es active IP Right Grant
- 2006-01-09 WO PCT/EP2006/000090 patent/WO2006074884A1/en active Application Filing
- 2006-01-09 BR BRPI0606644-5A patent/BRPI0606644A2/pt not_active IP Right Cessation
- 2006-01-09 ES ES06701375T patent/ES2346685T3/es active Active
- 2006-01-09 KR KR1020077018398A patent/KR100905810B1/ko not_active IP Right Cessation
- 2006-01-09 RU RU2007125622/04A patent/RU2007125622A/ru not_active Application Discontinuation
- 2006-01-09 AT AT06701375T patent/ATE474839T1/de active
- 2006-01-10 US US11/328,879 patent/US7678815B2/en not_active Expired - Fee Related
- 2006-01-12 TW TW095101218A patent/TW200637550A/zh unknown
- 2006-01-13 AR ARP060100140A patent/AR052558A1/es unknown
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2007
- 2007-07-05 IL IL184427A patent/IL184427A/en not_active IP Right Cessation
- 2007-07-10 ZA ZA200705670A patent/ZA200705670B/xx unknown
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Also Published As
Publication number | Publication date |
---|---|
ZA200705670B (en) | 2008-12-31 |
EP1844044A1 (en) | 2007-10-17 |
CA2593439C (en) | 2014-02-25 |
ATE474839T1 (de) | 2010-08-15 |
AU2006205920B2 (en) | 2012-11-15 |
CA2593439A1 (en) | 2006-07-20 |
WO2006074884A1 (en) | 2006-07-20 |
DE602006015607D1 (de) | 2010-09-02 |
IL184427A (en) | 2013-11-28 |
AU2006205920A1 (en) | 2006-07-20 |
US7678815B2 (en) | 2010-03-16 |
CN101137653A (zh) | 2008-03-05 |
JP2008526909A (ja) | 2008-07-24 |
KR100905810B1 (ko) | 2009-07-02 |
US20060160857A1 (en) | 2006-07-20 |
RU2007125622A (ru) | 2009-02-20 |
AR052558A1 (es) | 2007-03-21 |
KR20070094659A (ko) | 2007-09-20 |
IL184427A0 (en) | 2007-10-31 |
MX2007008410A (es) | 2007-08-21 |
EP1844044B1 (en) | 2010-07-21 |
TW200637550A (en) | 2006-11-01 |
JP4966866B2 (ja) | 2012-07-04 |
NO20073663L (no) | 2007-09-03 |
CN101137653B (zh) | 2012-05-09 |
ES2346685T3 (es) | 2010-10-19 |
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