BRPI0517643A - derivados de ácido piridono-carboxìlico ou seus sais - Google Patents

derivados de ácido piridono-carboxìlico ou seus sais

Info

Publication number
BRPI0517643A
BRPI0517643A BRPI0517643-3A BRPI0517643A BRPI0517643A BR PI0517643 A BRPI0517643 A BR PI0517643A BR PI0517643 A BRPI0517643 A BR PI0517643A BR PI0517643 A BRPI0517643 A BR PI0517643A
Authority
BR
Brazil
Prior art keywords
atom
present
pyridono
salts
group
Prior art date
Application number
BRPI0517643-3A
Other languages
English (en)
Inventor
Akira Yazaki
Yasuhiro Kuramoto
Kenji Itoh
Kazusa Yoshikai
Yuzo Hirao
Yoshihiro Ohshita
Norihiro Hayashi
Hirotaka Amano
Takayuki Amago
Hitomi Takenaka
Original Assignee
Wakunaga Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wakunaga Pharma Co Ltd filed Critical Wakunaga Pharma Co Ltd
Publication of BRPI0517643A publication Critical patent/BRPI0517643A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

DERIVADOS DE ACIDO PIRIDONO-CARBOXILICO OU SEUS SAIS. A invenção propõe medicamentos que apresentam uma atividade antibacteriana excelente, baixa toxicidade, uma melhor biodisponibilidade e baixos graus de ligação àsproteínas do plasma. Os derivados de ácidos piridono-carbo-xílicos representados pela fórmula geral (1) ou seus sais; e agentes antibacterianos ou medicamentos, contendo os mesmos. A fórmula geral (1) em que R˜ e metila, flúor ou cloro; R e hidrogênio ou alquila inferior; R é isopropila ou tercbutila; R~ 4~ é metila ou halogênio; e R~ 5~ é flúor ou cloro.
BRPI0517643-3A 2004-11-17 2005-11-17 derivados de ácido piridono-carboxìlico ou seus sais BRPI0517643A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2004333244 2004-11-17
PCT/JP2005/021093 WO2006054623A1 (ja) 2004-11-17 2005-11-17 新規ピリドンカルボン酸誘導体又はその塩

Publications (1)

Publication Number Publication Date
BRPI0517643A true BRPI0517643A (pt) 2008-10-14

Family

ID=36407161

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0517643-3A BRPI0517643A (pt) 2004-11-17 2005-11-17 derivados de ácido piridono-carboxìlico ou seus sais

Country Status (21)

Country Link
US (1) US7713997B2 (pt)
EP (1) EP1813610B1 (pt)
JP (1) JP3995705B2 (pt)
KR (1) KR20070084159A (pt)
CN (1) CN101061109B (pt)
AT (1) ATE480535T1 (pt)
AU (1) AU2005307447B2 (pt)
BR (1) BRPI0517643A (pt)
CA (1) CA2588034A1 (pt)
CY (1) CY1110898T1 (pt)
DE (1) DE602005023513D1 (pt)
DK (1) DK1813610T3 (pt)
ES (1) ES2349278T3 (pt)
HK (1) HK1109616A1 (pt)
MX (1) MX2007005892A (pt)
PL (1) PL1813610T3 (pt)
PT (1) PT1813610E (pt)
RU (1) RU2379304C2 (pt)
SI (1) SI1813610T1 (pt)
WO (1) WO2006054623A1 (pt)
ZA (1) ZA200704862B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112018076175A2 (pt) * 2016-06-15 2019-03-26 Wakunaga Pharmaceutical Co., Ltd. novo derivado de ácido piridonacarboxílico ou sal deste
RU2634122C1 (ru) * 2016-12-14 2017-10-24 федеральное государственное автономное образовательное учреждение высшего образования "Казанский (Приволжский) федеральный университет" (ФГАОУ ВО КФУ) Фторхинолоны на основе 4-дезоксипиридоксина
CN114539213A (zh) * 2021-08-18 2022-05-27 广东工业大学 一种氟喹诺酮类化合物及其制备方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2171252C2 (ru) * 1995-09-22 2001-07-27 Вакунага Фармасьютикал КО., Лтд. Аминосоединение для получения новых производных пиридонкарбоновой кислоты или их солей
CZ302033B6 (cs) * 1999-07-01 2010-09-08 Wakunaga Pharmaceutical Co., Ltd. Derivát chinolinkarboxylové kyseliny a jeho soli, farmaceutický prostredek je obsahující, jejich použití
EP1345603A4 (en) * 2000-12-20 2004-09-08 Merck & Co Inc P38 KINASE INHIBITORS (HALO-BENZO CARBONYL) HETEROCYCLO- FUSIONNES PHENYL

Also Published As

Publication number Publication date
AU2005307447B2 (en) 2011-03-10
US7713997B2 (en) 2010-05-11
ES2349278T3 (es) 2010-12-29
ATE480535T1 (de) 2010-09-15
AU2005307447A1 (en) 2006-05-26
DE602005023513D1 (de) 2010-10-21
DK1813610T3 (da) 2010-12-06
RU2379304C2 (ru) 2010-01-20
WO2006054623A1 (ja) 2006-05-26
KR20070084159A (ko) 2007-08-24
EP1813610B1 (en) 2010-09-08
JP3995705B2 (ja) 2007-10-24
MX2007005892A (es) 2007-06-19
CY1110898T1 (el) 2015-06-10
SI1813610T1 (sl) 2010-12-31
CN101061109A (zh) 2007-10-24
CA2588034A1 (en) 2006-05-26
JPWO2006054623A1 (ja) 2008-05-29
PT1813610E (pt) 2010-10-11
HK1109616A1 (en) 2008-06-13
US20090149440A1 (en) 2009-06-11
EP1813610A1 (en) 2007-08-01
RU2007122499A (ru) 2008-12-27
CN101061109B (zh) 2011-05-25
PL1813610T3 (pl) 2011-02-28
ZA200704862B (en) 2008-12-31
EP1813610A4 (en) 2009-05-20

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2260 DE 29/04/2014.