BRPI0512049A - usos antivirais de complexos de ácido borìnico - Google Patents
usos antivirais de complexos de ácido borìnicoInfo
- Publication number
- BRPI0512049A BRPI0512049A BRPI0512049-7A BRPI0512049A BRPI0512049A BR PI0512049 A BRPI0512049 A BR PI0512049A BR PI0512049 A BRPI0512049 A BR PI0512049A BR PI0512049 A BRPI0512049 A BR PI0512049A
- Authority
- BR
- Brazil
- Prior art keywords
- acid complexes
- boronic acid
- antiviral
- antiviral uses
- complexes
- Prior art date
Links
- 150000001642 boronic acid derivatives Chemical class 0.000 title abstract 2
- 230000000840 anti-viral effect Effects 0.000 title 1
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 3
- 241000700605 Viruses Species 0.000 abstract 1
- 239000003443 antiviral agent Substances 0.000 abstract 1
- UYANAUSDHIFLFQ-UHFFFAOYSA-N borinic acid Chemical class OB UYANAUSDHIFLFQ-UHFFFAOYSA-N 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- SIOXPEMLGUPBBT-UHFFFAOYSA-N picolinic acid Chemical class OC(=O)C1=CC=CC=N1 SIOXPEMLGUPBBT-UHFFFAOYSA-N 0.000 abstract 1
- MCJGNVYPOGVAJF-UHFFFAOYSA-N quinolin-8-ol Chemical compound C1=CN=C2C(O)=CC=CC2=C1 MCJGNVYPOGVAJF-UHFFFAOYSA-N 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/20—Antivirals for DNA viruses
- A61P31/22—Antivirals for DNA viruses for herpes viruses
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Molecular Biology (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57941904P | 2004-06-14 | 2004-06-14 | |
| PCT/US2005/020978 WO2006085932A2 (en) | 2004-06-14 | 2005-06-14 | Anti-viral uses of borinic acid complexes |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0512049A true BRPI0512049A (pt) | 2008-02-06 |
Family
ID=36623539
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0512049-7A BRPI0512049A (pt) | 2004-06-14 | 2005-06-14 | usos antivirais de complexos de ácido borìnico |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7393856B2 (enExample) |
| EP (1) | EP1765360B1 (enExample) |
| JP (1) | JP2008502694A (enExample) |
| AT (1) | ATE447960T1 (enExample) |
| BR (1) | BRPI0512049A (enExample) |
| CA (1) | CA2570577A1 (enExample) |
| DE (1) | DE602005017626D1 (enExample) |
| ES (1) | ES2333244T3 (enExample) |
| MX (1) | MXPA06014417A (enExample) |
| PT (1) | PT1765360E (enExample) |
| TW (1) | TW200612967A (enExample) |
| WO (1) | WO2006085932A2 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2008130902A (ru) * | 2005-12-28 | 2010-02-10 | Анакор Фармасьютикалз, Инк. (Us) | Способ получения пиколинатбориновых сложных эфиров |
| RS54108B1 (sr) | 2006-02-16 | 2015-12-31 | Anacor Pharmaceuticals Inc. | Mali molekuli koji sadrže boron kao agensi protiv zapaljenja |
| US8853424B2 (en) | 2008-08-11 | 2014-10-07 | Japan Science And Technology Agency | Protein cross-linking inhibitor |
| US8980544B2 (en) | 2012-11-27 | 2015-03-17 | The Penn State Research Foundation | Boronic and borinic acid compounds as inhibitors of sulfenic acid-containing proteins |
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| MX356059B (es) | 2013-01-30 | 2018-05-11 | Dow Agrosciences Llc | Uso de benzoxaboroles como agentes antimicrobianos volatiles en carnes, plantas, o partes de plantas. |
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| US9585396B2 (en) | 2013-01-30 | 2017-03-07 | Agrofresh Inc. | Volatile applications against pathogens |
| US8669207B1 (en) | 2013-01-30 | 2014-03-11 | Dow Agrosciences, Llc. | Compounds and compositions |
| KR101756785B1 (ko) | 2015-03-10 | 2017-07-12 | 한국화학연구원 | 4배위 유기 붕소 화합물의 제조방법 |
| EP3426029B1 (en) | 2016-03-07 | 2023-08-30 | AgroFresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
| EP3609504A4 (en) | 2017-03-01 | 2021-03-03 | Anacor Pharmaceuticals, Inc. | NEW OXABOROLE ANALOGUES AND USES OF THE LATEST |
| TWI883391B (zh) * | 2020-02-18 | 2025-05-11 | 美商基利科學股份有限公司 | 抗病毒化合物 |
| US20230340530A1 (en) | 2020-08-31 | 2023-10-26 | Pfizer Inc. | Methods of Protecting RNA |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU5788800A (en) | 1999-07-07 | 2001-01-22 | Du Pont Pharmaceuticals Company | Peptide boronic acid inhibitors of hepatitis c virus protease |
| JP2006511613A (ja) * | 2002-12-18 | 2006-04-06 | アナコア ファーマシューティカルズ インコーポレイテッド | ボロン酸複合体を含む抗生物質および使用法 |
-
2005
- 2005-06-14 ES ES05856817T patent/ES2333244T3/es not_active Expired - Lifetime
- 2005-06-14 MX MXPA06014417A patent/MXPA06014417A/es active IP Right Grant
- 2005-06-14 PT PT05856817T patent/PT1765360E/pt unknown
- 2005-06-14 WO PCT/US2005/020978 patent/WO2006085932A2/en not_active Ceased
- 2005-06-14 AT AT05856817T patent/ATE447960T1/de not_active IP Right Cessation
- 2005-06-14 JP JP2007516648A patent/JP2008502694A/ja not_active Withdrawn
- 2005-06-14 DE DE602005017626T patent/DE602005017626D1/de not_active Expired - Lifetime
- 2005-06-14 US US11/152,959 patent/US7393856B2/en not_active Expired - Fee Related
- 2005-06-14 BR BRPI0512049-7A patent/BRPI0512049A/pt not_active IP Right Cessation
- 2005-06-14 EP EP05856817A patent/EP1765360B1/en not_active Expired - Lifetime
- 2005-06-14 TW TW094119708A patent/TW200612967A/zh unknown
- 2005-06-14 CA CA002570577A patent/CA2570577A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP2008502694A (ja) | 2008-01-31 |
| ATE447960T1 (de) | 2009-11-15 |
| WO2006085932A3 (en) | 2006-10-05 |
| US7393856B2 (en) | 2008-07-01 |
| TW200612967A (en) | 2006-05-01 |
| PT1765360E (pt) | 2009-12-24 |
| WO2006085932A2 (en) | 2006-08-17 |
| CA2570577A1 (en) | 2006-08-17 |
| EP1765360B1 (en) | 2009-11-11 |
| HK1102702A1 (en) | 2007-11-30 |
| US20060019927A1 (en) | 2006-01-26 |
| DE602005017626D1 (de) | 2009-12-24 |
| MXPA06014417A (es) | 2007-03-08 |
| EP1765360A2 (en) | 2007-03-28 |
| ES2333244T3 (es) | 2010-02-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012. |