BRPI0512108A - antibióticos contendo complexos de ácido borìnico e métodos de uso - Google Patents
antibióticos contendo complexos de ácido borìnico e métodos de usoInfo
- Publication number
- BRPI0512108A BRPI0512108A BRPI0512108-6A BRPI0512108A BRPI0512108A BR PI0512108 A BRPI0512108 A BR PI0512108A BR PI0512108 A BRPI0512108 A BR PI0512108A BR PI0512108 A BRPI0512108 A BR PI0512108A
- Authority
- BR
- Brazil
- Prior art keywords
- methods
- antibiotics
- acid complexes
- boronic acid
- containing boronic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/04—Esters of boric acids
Abstract
ANTIBIóTICOS CONTENDO COMPLEXOS DE áCIDO BORìNICO E MéTODOS E USO A estrutura e preparação de antibióticos que incorporam complexos de ácido borínico são reveladas, especialmente derivados de hidroxiquinolina, imidazol e ácido picolínico, juntamente com composições desses antibióticos e métodos de utilização dos antibióticos e composições como agentes bactericidas e fungicidas, bem como agentes terapêuticos para o tratamento de doenças causadas por bactérias e fungos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/867,465 US7390806B2 (en) | 2002-12-18 | 2004-06-14 | Antibiotics containing borinic acid complexes and methods of use |
PCT/US2005/021214 WO2006007384A2 (en) | 2004-06-14 | 2005-06-14 | Antibiotics containing borinic acid complexes and methods of use |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0512108A true BRPI0512108A (pt) | 2008-02-06 |
Family
ID=35415124
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0512108-6A BRPI0512108A (pt) | 2004-06-14 | 2005-06-14 | antibióticos contendo complexos de ácido borìnico e métodos de uso |
Country Status (13)
Country | Link |
---|---|
US (2) | US7390806B2 (pt) |
EP (1) | EP1765359A2 (pt) |
JP (1) | JP2008502701A (pt) |
KR (1) | KR20070026783A (pt) |
CN (1) | CN1972694A (pt) |
AU (1) | AU2005262536A1 (pt) |
BR (1) | BRPI0512108A (pt) |
CA (1) | CA2570591A1 (pt) |
IL (1) | IL179748A0 (pt) |
MX (1) | MXPA06014418A (pt) |
RU (1) | RU2007101284A (pt) |
TW (2) | TW200612939A (pt) |
WO (1) | WO2006007384A2 (pt) |
Families Citing this family (43)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20040224923A1 (en) * | 2002-12-18 | 2004-11-11 | Ving Lee | Antibiotics containing borinic acid complexes and methods of use |
US7390806B2 (en) | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
FR2864083B1 (fr) * | 2003-12-18 | 2007-04-13 | Galderma Res & Dev | Nouveaux derives d'acides phenyl-boroniques et leurs procedes de preparation. |
AR049916A1 (es) * | 2004-06-14 | 2006-09-13 | Anacor Pharmaceuticals Inc | Usos anti-parasitarios de complejos de acido borinico |
HUE040060T2 (hu) | 2005-02-16 | 2019-02-28 | Anacor Pharmaceuticals Inc | Halogén-szubsztituált boronftalidok fertõzések kezelésére |
AU2006332797A1 (en) * | 2005-12-28 | 2007-07-12 | Anacor Pharmaceuticals, Inc. | Process for manufacturing picolinate borinic esters |
CN106008583A (zh) | 2005-12-30 | 2016-10-12 | 安纳考尔医药公司 | 含硼的小分子 |
US8168614B2 (en) | 2006-02-16 | 2012-05-01 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-inflammatory agents |
US20070286822A1 (en) * | 2006-06-12 | 2007-12-13 | Anacor Pharmaceuticals Inc. | Compounds for the Treatment of Periodontal Disease |
MX2008015918A (es) * | 2006-06-12 | 2009-01-14 | Anacor Pharmaceuticals Inc | Compuestos para el tratamiento de enfermedad periodontal. |
JO3598B1 (ar) | 2006-10-10 | 2020-07-05 | Infinity Discovery Inc | الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني |
RU2547441C2 (ru) | 2008-03-06 | 2015-04-10 | Анакор Фармасьютикалз, Инк. | Борсодержащие малые молекулы в качестве противовоспалительных агентов |
PE20091838A1 (es) | 2008-04-09 | 2009-12-18 | Infinity Pharmaceuticals Inc | Inhibidores de amida hidrolasa de acido graso |
EP2285384A4 (en) * | 2008-05-12 | 2012-04-25 | Anacor Pharmaceuticals Inc | BORN SMALL MOLECULES |
EP2348863A4 (en) * | 2008-09-04 | 2012-03-07 | Anacor Pharmaceuticals Inc | BORN SMALL MOLECULES |
WO2010028005A1 (en) | 2008-09-04 | 2010-03-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
US9493489B2 (en) * | 2008-10-15 | 2016-11-15 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agents |
US8461364B2 (en) * | 2008-12-17 | 2013-06-11 | Glaxosmithkline Llc | Polymorphs of (S)-3-aminomethyl-7-(3-hydroxy-propoxy)-3H-benzo[C][1,2]oxaborol-1-OL |
EP2416660B1 (en) | 2009-04-07 | 2014-07-02 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
CA2757622A1 (en) | 2009-04-07 | 2010-10-14 | Infinity Pharmaceuticals, Inc. | Inhibitors of fatty acid amide hydrolase |
TW201109022A (en) | 2009-06-03 | 2011-03-16 | Colgate Palmolive Co | Borinic compositions |
WO2011017125A1 (en) * | 2009-07-28 | 2011-02-10 | Anacor Pharmaceuticals, Inc. | Trisubstituted boron-containing molecules |
WO2011019618A1 (en) * | 2009-08-14 | 2011-02-17 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
WO2011022337A1 (en) * | 2009-08-19 | 2011-02-24 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
WO2011037731A1 (en) * | 2009-09-25 | 2011-03-31 | Anacor Pharmaceuticals, Inc. | Boron containing small molecules |
WO2011049971A1 (en) | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
US20110212918A1 (en) * | 2009-11-11 | 2011-09-01 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
US8716478B2 (en) | 2010-01-27 | 2014-05-06 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
RU2569061C2 (ru) | 2010-02-03 | 2015-11-20 | Инфинити Фармасьютикалз, Инк. | Ингибиторы амид-гидролазы жирных кислот |
AP2012006482A0 (en) | 2010-03-19 | 2012-10-31 | Anacor Pharmacueticals Inc | Boron-containing small molecules as anti-protozoalagent |
ES2635333T3 (es) | 2010-09-07 | 2017-10-03 | Anacor Pharmaceuticals, Inc. | Derivados de benzoxaborol para tratar infecciones bacterianas |
US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
US8669207B1 (en) | 2013-01-30 | 2014-03-11 | Dow Agrosciences, Llc. | Compounds and compositions |
CA2899317A1 (en) | 2013-01-30 | 2014-08-07 | Dow Agrosciences Llc | Use of benzoxaboroles as volatile antimicrobial agents on meats, plants, or plant parts |
US9585396B2 (en) | 2013-01-30 | 2017-03-07 | Agrofresh Inc. | Volatile applications against pathogens |
KR101636431B1 (ko) | 2013-07-30 | 2016-07-05 | 동아에스티 주식회사 | 트리사이클릭 벤즈옥사보롤 화합물, 이의 제조방법 및 용도 |
KR101756785B1 (ko) * | 2015-03-10 | 2017-07-12 | 한국화학연구원 | 4배위 유기 붕소 화합물의 제조방법 |
CA3015662A1 (en) | 2016-03-07 | 2017-09-14 | Agrofresh Inc. | Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops |
EP3576747A4 (en) * | 2017-03-09 | 2020-12-16 | The Penn State Research Foundation | SMALL MOLECULES CONTAINING BORON TO INHIBIT THE ACTIVITY OF A RECEPTOR-TYPE PROTEIN TYROSINE PHOSPHATASE |
US10526343B2 (en) | 2018-03-26 | 2020-01-07 | University Of Sharjah | Heterocyclic systems and pharmaceutical applications thereof |
CN111995634B (zh) * | 2020-08-28 | 2022-08-05 | 深圳大学 | 一种四配位有机硼化合物、荧光探针及其制备方法与应用 |
WO2022043936A1 (en) | 2020-08-31 | 2022-03-03 | Pfizer Inc. | Methods of protecting rna |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5348948A (en) | 1993-05-07 | 1994-09-20 | American Cyanamid Company | 2,2-diaryl-1-(oxa and thia)-2a-azonia-2-borataacenaphthene fungicidal |
US5348947A (en) * | 1993-05-07 | 1994-09-20 | American Cyanamid Company | Diarylboron ester and thioester fungicidal agents |
WO2000044387A1 (fr) * | 1999-01-29 | 2000-08-03 | Nitto Kasei Co., Ltd. | Composes organobores presentant une activite de coccidiostats |
CN1370170A (zh) | 1999-05-25 | 2002-09-18 | 宾夕法尼亚州研究基金会 | Dna甲基转移酶抑制剂 |
JP4138662B2 (ja) | 2002-01-10 | 2008-08-27 | ザ・ペンシルバニア・ステイト・リサーチ・フアウンデイシヨン | アルキルジアリールボリネートおよび錯化ジアリールボロン酸を調製するための方法。 |
US20040007657A1 (en) | 2002-07-08 | 2004-01-15 | Mcenroe John D. | Casting form for a cast-in-place structural element and fencing system including cast-in-place structural elements |
US7390806B2 (en) | 2002-12-18 | 2008-06-24 | Anacor Pharmaceuticals, Inc. | Antibiotics containing borinic acid complexes and methods of use |
US20040224923A1 (en) | 2002-12-18 | 2004-11-11 | Ving Lee | Antibiotics containing borinic acid complexes and methods of use |
-
2004
- 2004-06-14 US US10/867,465 patent/US7390806B2/en not_active Expired - Fee Related
-
2005
- 2005-06-13 TW TW094119534A patent/TW200612939A/zh unknown
- 2005-06-13 TW TW098110801A patent/TW200938195A/zh unknown
- 2005-06-14 KR KR1020077000300A patent/KR20070026783A/ko not_active Application Discontinuation
- 2005-06-14 EP EP05792513A patent/EP1765359A2/en not_active Withdrawn
- 2005-06-14 MX MXPA06014418A patent/MXPA06014418A/es not_active Application Discontinuation
- 2005-06-14 BR BRPI0512108-6A patent/BRPI0512108A/pt not_active IP Right Cessation
- 2005-06-14 CA CA002570591A patent/CA2570591A1/en not_active Abandoned
- 2005-06-14 CN CNA2005800194769A patent/CN1972694A/zh active Pending
- 2005-06-14 JP JP2007516705A patent/JP2008502701A/ja active Pending
- 2005-06-14 AU AU2005262536A patent/AU2005262536A1/en not_active Abandoned
- 2005-06-14 RU RU2007101284/04A patent/RU2007101284A/ru not_active Application Discontinuation
- 2005-06-14 WO PCT/US2005/021214 patent/WO2006007384A2/en active Application Filing
-
2006
- 2006-11-30 IL IL179748A patent/IL179748A0/en unknown
-
2008
- 2008-01-09 US US11/971,693 patent/US7888356B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US7390806B2 (en) | 2008-06-24 |
WO2006007384B1 (en) | 2006-08-17 |
KR20070026783A (ko) | 2007-03-08 |
EP1765359A2 (en) | 2007-03-28 |
RU2007101284A (ru) | 2008-07-20 |
AU2005262536A1 (en) | 2006-01-19 |
US7888356B2 (en) | 2011-02-15 |
JP2008502701A (ja) | 2008-01-31 |
US20080293675A1 (en) | 2008-11-27 |
CA2570591A1 (en) | 2006-01-19 |
WO2006007384A2 (en) | 2006-01-19 |
TW200612939A (en) | 2006-05-01 |
WO2006007384A3 (en) | 2006-04-06 |
TW200938195A (en) | 2009-09-16 |
MXPA06014418A (es) | 2007-03-08 |
US20050070503A1 (en) | 2005-03-31 |
IL179748A0 (en) | 2007-05-15 |
CN1972694A (zh) | 2007-05-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012. |