BRPI0415023A - derivados de triterpenos inusitados, sua preparação e seu uso - Google Patents
derivados de triterpenos inusitados, sua preparação e seu usoInfo
- Publication number
- BRPI0415023A BRPI0415023A BRPI0415023-6A BRPI0415023A BRPI0415023A BR PI0415023 A BRPI0415023 A BR PI0415023A BR PI0415023 A BRPI0415023 A BR PI0415023A BR PI0415023 A BRPI0415023 A BR PI0415023A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- unusual
- derivatives
- triterpene derivatives
- triterpene
- Prior art date
Links
- 150000003648 triterpenes Chemical class 0.000 title abstract 4
- 206010038997 Retroviral infections Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
- C07C69/67—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of saturated acids
- C07C69/708—Ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/34—Esters of acyclic saturated polycarboxylic acids having an esterified carboxyl group bound to an acyclic carbon atom
- C07C69/40—Succinic acid esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/34—Esters of acyclic saturated polycarboxylic acids having an esterified carboxyl group bound to an acyclic carbon atom
- C07C69/42—Glutaric acid esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/608—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a ring other than a six-membered aromatic ring in the acid moiety
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
- C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/52—Ortho- or ortho- and peri-condensed systems containing five condensed rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US50589903P | 2003-09-26 | 2003-09-26 | |
| US55935804P | 2004-04-05 | 2004-04-05 | |
| PCT/US2004/031370 WO2005030790A1 (en) | 2003-09-26 | 2004-09-27 | Novel triterpene derivatives, preparation thereof and use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0415023A true BRPI0415023A (pt) | 2006-11-07 |
Family
ID=34396277
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0415023-6A BRPI0415023A (pt) | 2003-09-26 | 2004-09-27 | derivados de triterpenos inusitados, sua preparação e seu uso |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20050148561A1 (enExample) |
| EP (1) | EP1675866A1 (enExample) |
| JP (1) | JP2007506761A (enExample) |
| KR (1) | KR20060096147A (enExample) |
| AU (1) | AU2004276307A1 (enExample) |
| BR (1) | BRPI0415023A (enExample) |
| CA (1) | CA2540160A1 (enExample) |
| IL (1) | IL174317A0 (enExample) |
| NO (1) | NO20061792L (enExample) |
| WO (1) | WO2005030790A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1730163A4 (en) * | 2004-03-17 | 2009-12-30 | Panacos Pharmaceuticals Inc | Pharmaceutical salts of 3-O- (3,3-dimethylsuccinyl) betulinic acid |
| BRPI0610668A2 (pt) * | 2005-04-12 | 2010-07-13 | Panacos Pharmaceuticals Inc | polimorfas de di-n-metil-d-glucamina do ácido 3-o-(3',3'-dimetilsuccinil) betulìnico |
| EP1893629A4 (en) * | 2005-06-22 | 2008-12-17 | Myriad Genetics Inc | ANTIVIRAL CONNECTIONS |
| GB0604899D0 (en) * | 2006-03-10 | 2006-04-19 | York Pharma Plc | Derivatives of 18-glycyrrhetinic acid |
| US20080039428A1 (en) * | 2006-06-29 | 2008-02-14 | Panacos Pharmaceuticals, Inc. | Antiretroviral combination therapy |
| WO2008115281A2 (en) * | 2006-10-16 | 2008-09-25 | Myriad Genetics, Inc. | Compounds for treating viral infections |
| WO2008057420A2 (en) | 2006-11-03 | 2008-05-15 | Panacos Pharmaceuticals, Inc. | Extended triterpene derivatives |
| WO2008146305A2 (en) * | 2007-06-01 | 2008-12-04 | Council Of Scientific & Industrial Research | A pharmaceutical composition having virucidal and spermicidal activity |
| KR100941595B1 (ko) * | 2008-06-05 | 2010-02-11 | 주식회사 알앤엘바이오 | 바이러스 억제제로서 유용한 트리테르페노이드계 화합물 |
| CN102532245B (zh) * | 2011-12-31 | 2013-05-15 | 中国人民解放军第三军医大学 | 一种熊果酸衍生物及其制备方法 |
| WO2018128956A1 (en) | 2017-01-05 | 2018-07-12 | Regents Of The University Of California | Contraceptive use of triterpenoids |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1415601A (en) * | 1973-03-14 | 1975-11-26 | Biorex Laboratories Ltd | Dihydrobetulinic acid derivatives |
| JP2004509972A (ja) * | 2000-09-29 | 2004-04-02 | リージェンツ オブ ザ ユニバーシティ オブ ミネソタ | 酵母に対する殺真菌活性を有するトリテルペン |
-
2004
- 2004-09-27 EP EP04784972A patent/EP1675866A1/en active Pending
- 2004-09-27 WO PCT/US2004/031370 patent/WO2005030790A1/en not_active Ceased
- 2004-09-27 US US10/949,875 patent/US20050148561A1/en not_active Abandoned
- 2004-09-27 JP JP2006528207A patent/JP2007506761A/ja not_active Withdrawn
- 2004-09-27 AU AU2004276307A patent/AU2004276307A1/en not_active Abandoned
- 2004-09-27 BR BRPI0415023-6A patent/BRPI0415023A/pt not_active IP Right Cessation
- 2004-09-27 KR KR1020067008088A patent/KR20060096147A/ko not_active Withdrawn
- 2004-09-27 CA CA002540160A patent/CA2540160A1/en not_active Abandoned
-
2006
- 2006-03-14 IL IL174317A patent/IL174317A0/en unknown
- 2006-04-24 NO NO20061792A patent/NO20061792L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2007506761A (ja) | 2007-03-22 |
| IL174317A0 (en) | 2006-08-01 |
| EP1675866A1 (en) | 2006-07-05 |
| WO2005030790A1 (en) | 2005-04-07 |
| AU2004276307A1 (en) | 2005-04-07 |
| US20050148561A1 (en) | 2005-07-07 |
| NO20061792L (no) | 2006-06-14 |
| KR20060096147A (ko) | 2006-09-07 |
| CA2540160A1 (en) | 2005-04-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A E 7A ANUIDADE(S) |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011. |