BR9912907A - Pirazóis nematicidas - Google Patents

Pirazóis nematicidas

Info

Publication number
BR9912907A
BR9912907A BR9912907-8A BR9912907A BR9912907A BR 9912907 A BR9912907 A BR 9912907A BR 9912907 A BR9912907 A BR 9912907A BR 9912907 A BR9912907 A BR 9912907A
Authority
BR
Brazil
Prior art keywords
total number
carbons
alkyl
haloalkyl
optionally substituted
Prior art date
Application number
BR9912907-8A
Other languages
English (en)
Inventor
Katsuaki Wada
Takuya Gomibuchi
Yuichi Otsu
Katsuhiko Shibuya
Takahisa Abe
Wolfram Andersch
Achim Harder
Peter Loesel
Original Assignee
Bayer Agrochem Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Agrochem Kk filed Critical Bayer Agrochem Kk
Publication of BR9912907A publication Critical patent/BR9912907A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Patente de Invenção: <B>"PIRAZóIS NEMATICIDAS"<D>. Esta invenção refere-se a novos pirazóis de fórmula (I), em que R¹ representa halogênio, C~ 1-6~ alquila, C~ 1-5~ haloalquila, C~ 2-6~ alcóxi, C~ 1-4~ alquiltio, C~ 2-5~ alquenilóxi, C~ 3-5~ alquinilóxi, C~ 2-6~ (número total de carbonos) alcoxialquila, C~ 2-6~ (número total de carbonos) alquiltioalquila, C~1-5~ haloalcóxi, C~ 2-6~ (número total de carbonos) alcoxialcóxi, hidróxi ou fenila opcionalmente substituída, R² representa hidrogênio, halogênio, C~ 1-5~ alquila, C~ 2-6~ (número total de carbonos) alcoxialquila, C~ 2-6~ (número total de carbonos) alquiltioalquila, C~ 2-6~ (número total de carbonos) alquilsulfinialquila, C~ 2-6~ (número total de carbonos) alquilsulfonilalquila ou C~ 1-5~ haloalquila, R^ 3^ representa hidrogênio, C~ 1-5~ alquila, -COR^ 4^, COOR^ 5^, CH(OR^ 6^)~ 2~ ou CH~ 2~Si(R^ 7^)~ 3~, R^ 4^ representa C~ 1-10~ alquila, C~ 1-6~ haloalquila, C~ 2-6~ alquenila, C~ 3-6~ cicloalquila opcionalmente substituída, C~ 2-6~ (número total de carbonos) alcoxialquila, C~ 2-6~ (número total de carbonos) alquiltioalquila, fenila opcionalmente substituída, C~ 1-6~ haloalquila, alquilamino, di-(C~ 1-4~ alquil)amino ou fenilamino opcionalmente substituído, R^ 5^ representa C~ 1-5~ alquila, R^ 6^ e R^ 7^ representam C~ 1-4~ alquila, e n é 1, 2, ou 3, e quando n é 2 ou 3, o número (n) correspondente de radicais R¹ poderá ser o mesmo ou diferente, a processos para preparação desses compostos e a seu uso como nematicidas e anti-helmínticos.
BR9912907-8A 1998-08-11 1999-08-03 Pirazóis nematicidas BR9912907A (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP23795898 1998-08-11
JP3859699 1999-02-17
JP16811799 1999-06-15
PCT/EP1999/005684 WO2000009500A2 (en) 1998-08-11 1999-08-03 Nematicidal pyrazoles

Publications (1)

Publication Number Publication Date
BR9912907A true BR9912907A (pt) 2001-05-08

Family

ID=27289881

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9912907-8A BR9912907A (pt) 1998-08-11 1999-08-03 Pirazóis nematicidas

Country Status (9)

Country Link
US (2) US6310049B1 (pt)
EP (1) EP1104418A2 (pt)
JP (1) JP2003519081A (pt)
KR (1) KR20010071975A (pt)
AU (1) AU5510799A (pt)
BR (1) BR9912907A (pt)
CA (1) CA2339970A1 (pt)
TR (1) TR200100426T2 (pt)
WO (1) WO2000009500A2 (pt)

Families Citing this family (24)

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Publication number Priority date Publication date Assignee Title
DE19955634A1 (de) * 1999-11-21 2001-06-13 Morphochem Ag Kupplungs-Kondensations-Synthese von Heterocyclen
EP1398029A1 (en) * 2002-09-10 2004-03-17 LION Bioscience AG NR3B1 nuclear receptor binding 3-substituted pyrazole derivatives
WO2005030848A1 (en) * 2003-09-19 2005-04-07 Dow Global Technologies Inc. Multifunctional monomers and polyarylene compositions therefrom
HUE036519T2 (hu) 2007-08-13 2018-07-30 Monsanto Technology Llc Készítmények és eljárások nematódák irtására
WO2010093650A2 (en) * 2009-02-10 2010-08-19 Divergence, Inc. Compositions and methods for controlling nematodes
CN102647984B (zh) 2009-10-02 2015-03-25 埃维克辛公司 抗炎症的2-羰基噻唑和2-羰基恶唑
CA2829790C (en) * 2010-03-30 2018-06-05 Verseon Corporation Multisubstituted aromatic compounds as inhibitors of thrombin
BR112012033341B1 (pt) 2010-06-30 2022-08-23 Cyclerion Therapeutics, Inc Estimulantes de sgc
PL2605652T3 (pl) * 2010-08-18 2018-04-30 Samumed, Llc Diketony i hydroksyketony jako aktywatory szlaku sygnalizacji kateninowej
BR112013005136B1 (pt) 2010-09-02 2018-03-20 Monsanto Technology Llc Compostos e composições nematicidas, bem como métodos para controlar pragas de nematódeo
US9061030B2 (en) 2010-11-09 2015-06-23 Ironwood Pharmaceuticals, Inc. sGC stimulators
AR086992A1 (es) 2011-06-20 2014-02-05 Bayer Ip Gmbh Tienilpiri(mi)dinilpirazoles
EP2797915B1 (en) 2011-12-27 2016-07-13 Ironwood Pharmaceuticals, Inc. 2-benzyl-3-(oxazole/thiazole)-5-(pyrimidin-2-yl)-1(H)-pyrazole derivatives as stimulators of the soluble guanylate cyclase (sGC) for the treatment of e.g. hypertension or heart failure
CN105102438B (zh) 2013-01-29 2019-04-30 埃维克辛公司 抗炎症和抗肿瘤的2-氧代噻唑类和2-氧代噻吩类化合物
CA2901671C (en) 2013-02-22 2021-07-13 Samumed, Llc .gamma.-diketones as wnt/.beta. -catenin signaling pathway activators
AU2014238478B2 (en) 2013-03-15 2018-07-19 Verseon Corporation Halogenopyrazoles as inhibitors of thrombin
MX2015012867A (es) 2013-03-15 2016-06-10 Verseon Corp Compuestos aromaticos multisustituidos como inhibidores de serina proteasa.
UY35428A (es) 2013-03-15 2014-10-31 Monsanto Technology Llc ?azoles n-,c-disustituidos y composiciones y métodos para controlar plagas de nematodos?.
GB201413695D0 (en) 2014-08-01 2014-09-17 Avexxin As Compound
RU2727039C2 (ru) 2014-08-20 2020-07-17 СЭМЬЮМЕД, ЭлЭлСи Гамма-дикетоны для лечения и профилактики старения кожи и морщин
WO2016044662A1 (en) 2014-09-17 2016-03-24 Verseon Corporation Pyrazolyl-substituted pyridone compounds as serine protease inhibitors
SG10201907699YA (en) 2015-02-27 2019-09-27 Verseon Corp Substituted pyrazole compounds as serine protease inhibitors
GB201604318D0 (en) 2016-03-14 2016-04-27 Avexxin As Combination therapy
WO2020219871A1 (en) * 2019-04-26 2020-10-29 Celgene Corporation Heterocyclic compounds and their use for treatment of helminthic infections and diseases

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Publication number Priority date Publication date Assignee Title
US3991073A (en) * 1972-02-09 1976-11-09 U.S. Philips Corporation Pyrazoline compounds having insecticidal activity
US4122200A (en) 1974-11-20 1978-10-24 Lipha, Lyonnaise Industrielle Pharmaceutique 6',2-(2'Arylchromonyl) propionic acids, and analgesic and anti-inflammatory derivatives thereof
JPS6011882B2 (ja) 1980-03-04 1985-03-28 兼商株式会社 殺線虫剤
US4645796A (en) 1985-03-15 1987-02-24 The Dow Chemical Company Polyblends of styrene/α-methylstyrene copolymers with reinforcing interpolymerized styrene-grafted rubber concentrates
AU7301587A (en) 1986-04-30 1987-11-24 Fmc Corporation Photoactive azole pesticides

Also Published As

Publication number Publication date
JP2003519081A (ja) 2003-06-17
US6605730B2 (en) 2003-08-12
TR200100426T2 (tr) 2001-06-21
CA2339970A1 (en) 2000-02-24
WO2000009500A2 (en) 2000-02-24
US20030028034A1 (en) 2003-02-06
US6310049B1 (en) 2001-10-30
KR20010071975A (ko) 2001-07-31
EP1104418A2 (en) 2001-06-06
AU5510799A (en) 2000-03-06
WO2000009500A3 (en) 2000-06-15

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5O, 6O, 7O E 8O ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1913 DE 04/09/2007.