BR9911046A - Uso de antidepressivos tricìclicos para analgesia local - Google Patents

Uso de antidepressivos tricìclicos para analgesia local

Info

Publication number
BR9911046A
BR9911046A BR9911046-6A BR9911046A BR9911046A BR 9911046 A BR9911046 A BR 9911046A BR 9911046 A BR9911046 A BR 9911046A BR 9911046 A BR9911046 A BR 9911046A
Authority
BR
Brazil
Prior art keywords
generation
local
antidepressants
tricyclic antidepressants
tricyclic
Prior art date
Application number
BR9911046-6A
Other languages
English (en)
Inventor
Jana Sawynok
Mike Esser
Allison Reid
Original Assignee
Univ Dalhousie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Dalhousie filed Critical Univ Dalhousie
Publication of BR9911046A publication Critical patent/BR9911046A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A61P23/02—Local anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Anesthesiology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Patente de Invenção: <B>"USO DE ANTIDEPRESSIVOS TRICìCLICOS PARA ANALGESIA LOCAL"<D>. Quando administrados localmente, os antidepressivos tricíclicos, de segunda geração e terceira geração, tal como amitriptilina e desipramina, mostraram produzir analgesia em um indivíduo tendo um lugar de desconforto local. O efeito analgésico de tais antidepressivos, quando administrados localmente, é igual àquele conseguido através da administração sistêmica e dura mais. A invenção provê composições contendo antidepressivos tricíclicos, de segunda geração e de terceira geração para administração local, tal como aqueles formulados para aplicação tópica, ou para injeção em veículos de aplicação de liberação lenta, e método para o seu uso para produzir anestesia local.
BR9911046-6A 1998-05-19 1999-05-19 Uso de antidepressivos tricìclicos para analgesia local BR9911046A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/081,709 US6211171B1 (en) 1998-05-19 1998-05-19 Use of antidepressants for local analgesia
PCT/CA1999/000449 WO1999059598A1 (en) 1998-05-19 1999-05-19 Use of tricyclic antidepressants for local analgesia

Publications (1)

Publication Number Publication Date
BR9911046A true BR9911046A (pt) 2001-04-24

Family

ID=22165886

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9911046-6A BR9911046A (pt) 1998-05-19 1999-05-19 Uso de antidepressivos tricìclicos para analgesia local

Country Status (12)

Country Link
US (1) US6211171B1 (pt)
EP (1) EP1094818A1 (pt)
JP (1) JP2002515438A (pt)
KR (1) KR20010071301A (pt)
CN (1) CN1308530A (pt)
AU (1) AU3807799A (pt)
BR (1) BR9911046A (pt)
CA (1) CA2333310A1 (pt)
NO (1) NO20005835L (pt)
NZ (1) NZ508991A (pt)
TR (1) TR200003438T2 (pt)
WO (1) WO1999059598A1 (pt)

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Also Published As

Publication number Publication date
WO1999059598A1 (en) 1999-11-25
AU3807799A (en) 1999-12-06
EP1094818A1 (en) 2001-05-02
NO20005835L (no) 2001-01-18
JP2002515438A (ja) 2002-05-28
TR200003438T2 (tr) 2001-03-21
NO20005835D0 (no) 2000-11-17
KR20010071301A (ko) 2001-07-28
US6211171B1 (en) 2001-04-03
CN1308530A (zh) 2001-08-15
CA2333310A1 (en) 1999-11-25
NZ508991A (en) 2003-09-26

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5A, 6A, 7A E 8A ANUIDADES.

B08G Application fees: restoration [chapter 8.7 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DE INT.CL: A61K 31/645, A61K 31/55

Ipc: A61K 31/55 (2009.01)

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8,10(VIII) E 11 DA LPI

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.