BR9910804A - Processo para a preparação de sais cristalinos de amoxilina - Google Patents

Processo para a preparação de sais cristalinos de amoxilina

Info

Publication number
BR9910804A
BR9910804A BR9910804-6A BR9910804A BR9910804A BR 9910804 A BR9910804 A BR 9910804A BR 9910804 A BR9910804 A BR 9910804A BR 9910804 A BR9910804 A BR 9910804A
Authority
BR
Brazil
Prior art keywords
preparation
crystalline
salts
amoxylin
amoxicillin
Prior art date
Application number
BR9910804-6A
Other languages
English (en)
Inventor
Paul G Butterly
Esin F Kosal
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of BR9910804A publication Critical patent/BR9910804A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04Preparation
    • C07D499/14Preparation of salts
    • C07D499/16Preparation of salts of alkali or alkaline earth metals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE SAIS CRISTALINOS DE AMOXICILINA" é revelado um novo processo para a preparação de um cristalino sal de metal alcalino de amoxicilina.
BR9910804-6A 1998-06-01 1999-06-01 Processo para a preparação de sais cristalinos de amoxilina BR9910804A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8755498P 1998-06-01 1998-06-01
PCT/US1999/011991 WO1999062910A1 (en) 1998-06-01 1999-06-01 Process for preparing crystalline salts of amoxycillin

Publications (1)

Publication Number Publication Date
BR9910804A true BR9910804A (pt) 2001-02-13

Family

ID=22205864

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9910804-6A BR9910804A (pt) 1998-06-01 1999-06-01 Processo para a preparação de sais cristalinos de amoxilina

Country Status (15)

Country Link
EP (1) EP1086109A4 (pt)
JP (1) JP2002517398A (pt)
KR (1) KR20010043942A (pt)
CN (1) CN1182138C (pt)
AU (1) AU760934B2 (pt)
BR (1) BR9910804A (pt)
CA (1) CA2333943A1 (pt)
HU (1) HUP0102008A3 (pt)
IL (1) IL139736A (pt)
NO (1) NO20006073D0 (pt)
NZ (1) NZ508179A (pt)
PL (1) PL344348A1 (pt)
TR (1) TR200003517T2 (pt)
WO (1) WO1999062910A1 (pt)
ZA (1) ZA200006946B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6878386B1 (en) 1999-04-13 2005-04-12 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising amoxycillin and potassium clavulanate
US6294199B1 (en) 1999-04-13 2001-09-25 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising administering amoxycillin
WO2006072577A1 (en) * 2005-01-07 2006-07-13 Sandoz Ag Process for preparing granulates comprising amoxicillin
CN101633663B (zh) * 2009-08-28 2011-12-21 沈阳顺旺动物药业有限公司 一种青霉素类钠、钾盐的合成方法
MX2012014758A (es) * 2010-06-16 2013-10-01 Vardhman Chemtech Ltd Proceso mejorado para preparar amoxicilina sodica.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES8606871A1 (es) * 1985-10-21 1986-06-01 Antibioticos Sa Un procedimiento de preparacion de amoxicilina sodica
IT1255716B (it) * 1992-10-05 1995-11-10 Procedimento per la preparazione di antibiotici beta-lattamici sterili
TW347383B (en) * 1995-10-26 1998-12-11 Biochemie Gmbh A process for the production of a crystalline sodium salt of amoxicillin in ethanol as solvent

Also Published As

Publication number Publication date
EP1086109A1 (en) 2001-03-28
HUP0102008A2 (hu) 2001-12-28
IL139736A0 (en) 2002-02-10
EP1086109A4 (en) 2001-12-19
IL139736A (en) 2004-02-19
CN1182138C (zh) 2004-12-29
PL344348A1 (en) 2001-11-05
NO20006073L (no) 2000-11-30
AU4321699A (en) 1999-12-20
JP2002517398A (ja) 2002-06-18
NZ508179A (en) 2002-10-25
CN1304412A (zh) 2001-07-18
WO1999062910A1 (en) 1999-12-09
CA2333943A1 (en) 1999-12-09
ZA200006946B (en) 2002-01-28
NO20006073D0 (no) 2000-11-30
KR20010043942A (ko) 2001-05-25
TR200003517T2 (tr) 2001-06-21
HUP0102008A3 (en) 2002-07-29
AU760934B2 (en) 2003-05-22

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 9A E 10A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 1999 DE 28/04/2009.