BR9810657A - "processo de preparação de um per-hidroisoindol substituìdo" - Google Patents

"processo de preparação de um per-hidroisoindol substituìdo"

Info

Publication number
BR9810657A
BR9810657A BR9810657-0A BR9810657A BR9810657A BR 9810657 A BR9810657 A BR 9810657A BR 9810657 A BR9810657 A BR 9810657A BR 9810657 A BR9810657 A BR 9810657A
Authority
BR
Brazil
Prior art keywords
preparing
perhydroisoindole
substituted
substituted perhydroisoindole
perhydroisoindol
Prior art date
Application number
BR9810657-0A
Other languages
English (en)
Inventor
Jean-Pierre Lecouve
Claude Fugier
Jean-Claude Souvie
Original Assignee
Adir
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adir filed Critical Adir
Publication of BR9810657A publication Critical patent/BR9810657A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44Iso-indoles; Hydrogenated iso-indoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Indole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Patente de Invenção: <B>"PROCESSO DE PREPARAçãO DE UM PER-HIDROISOINDOL SUBSTITUìDO"<D>. A presente invenção refere-se a um processo de síntese industrial de um per-hidroisoindol substituído de fórmula (I) e de seus sais farmaceuticamente aceitáveis.
BR9810657-0A 1997-07-03 1998-07-01 "processo de preparação de um per-hidroisoindol substituìdo" BR9810657A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9708431A FR2765578B1 (fr) 1997-07-03 1997-07-03 Procede de preparation d'un perhydroisoindole substitue
PCT/FR1998/001405 WO1999001430A1 (fr) 1997-07-03 1998-07-01 Procede de preparation d'un perhydroisoindole substitue

Publications (1)

Publication Number Publication Date
BR9810657A true BR9810657A (pt) 2000-10-03

Family

ID=9508815

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9810657-0A BR9810657A (pt) 1997-07-03 1998-07-01 "processo de preparação de um per-hidroisoindol substituìdo"

Country Status (22)

Country Link
US (1) US6133454A (pt)
EP (1) EP0994854B1 (pt)
JP (1) JP4056093B2 (pt)
KR (1) KR100421073B1 (pt)
CN (1) CN1108291C (pt)
AT (1) ATE224368T1 (pt)
AU (1) AU734398B2 (pt)
BR (1) BR9810657A (pt)
CA (1) CA2295992C (pt)
DE (1) DE69808092T2 (pt)
DK (1) DK0994854T3 (pt)
EA (1) EA002151B1 (pt)
ES (1) ES2184304T3 (pt)
FR (1) FR2765578B1 (pt)
HK (1) HK1028610A1 (pt)
HU (1) HUP0002778A3 (pt)
NO (1) NO313095B1 (pt)
NZ (1) NZ501835A (pt)
PL (1) PL190861B1 (pt)
PT (1) PT994854E (pt)
WO (1) WO1999001430A1 (pt)
ZA (1) ZA985882B (pt)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2793411B1 (fr) * 1999-05-11 2001-06-29 Synthelabo Utilisation de derives de l'acide succinique pour obtenir un medicament destine au traitement de l'inflammation
FR2834892B1 (fr) * 2002-01-23 2004-02-27 Servier Lab Composition pharmaceutique orodispersible de mitiglinide
US6684422B2 (en) * 2002-02-27 2004-02-03 Ginger Magnolia Toy retention blanket and system
WO2004002473A1 (ja) * 2002-06-28 2004-01-08 Kissei Pharmaceutical Co., Ltd. 血糖コントロール用医薬組成物
JPWO2004002474A1 (ja) * 2002-06-28 2005-10-27 キッセイ薬品工業株式会社 糖尿病性合併症の予防又は進展阻止用医薬組成物
CA2496479A1 (en) * 2002-08-23 2004-03-04 Banyu Pharmaceutical Co., Ltd. Process for producing indolopyrrolocarbazole derivative
FR2860231B1 (fr) * 2003-09-25 2005-11-18 Servier Lab Nouveau procede de preparation du cis-octahydro-isoindole
US7230022B2 (en) * 2004-02-19 2007-06-12 Bristol-Myers Squibb Company Substituted fused bicyclic amines as modulators of chemokine receptor activity
CN1634885B (zh) * 2004-11-09 2011-05-04 北京乐力健生物科技有限公司 米格列奈晶型及其制备方法
CN1324010C (zh) * 2005-01-12 2007-07-04 江苏省药物研究所 一种米格列奈的制备方法
JP4918257B2 (ja) * 2005-12-27 2012-04-18 キッセイ薬品工業株式会社 不斉還元方法
WO2009047797A2 (en) * 2007-10-08 2009-04-16 Ind-Swift Laboratories Limited Process for the preparation of perhydroisoindole derivative
CN102382033B (zh) * 2010-08-31 2013-04-03 凯瑞斯德生化(苏州)有限公司 一种光学活性米格列奈酯及米格列奈盐的制备方法
ES2710452T3 (es) 2011-06-10 2019-04-25 Bluebird Bio Inc Vectores de terapia génica para la adrenoleucodistrofia y la adrenomieloneuropatía
KR101327866B1 (ko) * 2011-10-27 2013-11-11 주식회사 메디켐코리아 미티글리나이드 칼슘염의 개선된 제조방법
WO2013189829A1 (en) 2012-06-22 2013-12-27 Laboratorios Lesvi, S. L. Process for obtaining (s)-2-benzyl-4-((3ar,7as)-hexahydro-1 h-isoindol- 2(3h)-yl)-4-oxobutanoic acid and salts thereof
CN103450069B (zh) * 2013-06-24 2015-04-15 山西大同大学 一种米格列奈钙的制备方法
CN103709092B (zh) * 2013-11-04 2016-07-06 河北科技大学 米格列奈钙的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU654331B2 (en) * 1991-03-30 1994-11-03 Kissei Pharmaceutical Co. Ltd. Succinic acid compounds

Also Published As

Publication number Publication date
JP2002507222A (ja) 2002-03-05
NO313095B1 (no) 2002-08-12
HU0002778D0 (en) 1998-07-01
NO996577D0 (no) 1999-12-30
CA2295992A1 (fr) 1999-01-14
NO996577L (no) 2000-03-02
FR2765578B1 (fr) 1999-09-10
DE69808092T2 (de) 2003-04-30
HUP0002778A2 (hu) 2001-01-29
ZA985882B (en) 1999-01-26
US6133454A (en) 2000-10-17
NZ501835A (en) 2000-11-24
EA200000094A1 (ru) 2000-06-26
JP4056093B2 (ja) 2008-03-05
HUP0002778A3 (en) 2001-12-28
AU8445098A (en) 1999-01-25
DE69808092D1 (de) 2002-10-24
ES2184304T3 (es) 2003-04-01
EP0994854B1 (fr) 2002-09-18
PT994854E (pt) 2002-12-31
DK0994854T3 (da) 2002-12-30
ATE224368T1 (de) 2002-10-15
FR2765578A1 (fr) 1999-01-08
CA2295992C (fr) 2003-09-23
EA002151B1 (ru) 2001-12-24
HK1028610A1 (en) 2001-02-23
WO1999001430A1 (fr) 1999-01-14
CN1108291C (zh) 2003-05-14
KR100421073B1 (ko) 2004-06-11
KR19990013522A (ko) 1999-02-25
CN1261879A (zh) 2000-08-02
PL337728A1 (en) 2000-08-28
EP0994854A1 (fr) 2000-04-26
PL190861B1 (pl) 2006-02-28
AU734398B2 (en) 2001-06-14

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DE INT.CL: C07D 209/44, A61K 31/4035, A61P 3/10

Ipc: C07D 209/44 (2007.10), A61K 31/4035 (2007.10), A61

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO, UMA VEZ QUE O MESMO NAO ATENDE AO DISPOSTO NOS ARTIGOS 8O E 13 DA LPI