BR9815220A - Uso de tiazolidinedionas para o tratamento da hiperglicemia - Google Patents

Uso de tiazolidinedionas para o tratamento da hiperglicemia

Info

Publication number
BR9815220A
BR9815220A BR9815220-3A BR9815220A BR9815220A BR 9815220 A BR9815220 A BR 9815220A BR 9815220 A BR9815220 A BR 9815220A BR 9815220 A BR9815220 A BR 9815220A
Authority
BR
Brazil
Prior art keywords
treatment
hyperglycemia
thiazolidinediones
thiazolidinedions
mammal
Prior art date
Application number
BR9815220-3A
Other languages
English (en)
Inventor
Robin Edwing Buckingham
Stephen Alistair Smith
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of BR9815220A publication Critical patent/BR9815220A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"USO DE TIAZOLIDINEDIONAS PARA O TRATAMENTO DA HIPERGLICEMIA" A presente invenção refere-se um método para o tratamento da hiperglicemia onde os níveis plasmáticos de glicose na faixa de >126 mg/dl a 140 mg/dl, cujo método compreende a administração de uma quantidade eficaz, não-tóxica e farmaceuticamente aceitável de um sensibilizador da insulina, para um mamífero que necessite do tratamento.
BR9815220-3A 1997-10-13 1998-10-12 Uso de tiazolidinedionas para o tratamento da hiperglicemia BR9815220A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9721692.3A GB9721692D0 (en) 1997-10-13 1997-10-13 Novel treatment
PCT/GB1998/003067 WO1999018944A1 (en) 1997-10-13 1998-10-12 Use of thiazolidinediones for the treatment of hyperglycaemia

Publications (1)

Publication Number Publication Date
BR9815220A true BR9815220A (pt) 2000-11-14

Family

ID=10820481

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9815220-3A BR9815220A (pt) 1997-10-13 1998-10-12 Uso de tiazolidinedionas para o tratamento da hiperglicemia

Country Status (24)

Country Link
EP (1) EP1023057A1 (pt)
JP (1) JP2001519383A (pt)
KR (1) KR20010024482A (pt)
CN (1) CN1281358A (pt)
AP (1) AP1223A (pt)
AU (1) AU9547198A (pt)
BG (1) BG104405A (pt)
BR (1) BR9815220A (pt)
CA (1) CA2305289A1 (pt)
CZ (1) CZ20001298A3 (pt)
EA (1) EA200000418A1 (pt)
GB (1) GB9721692D0 (pt)
HR (1) HRP20000256A2 (pt)
HU (1) HUP0003673A3 (pt)
ID (1) ID24439A (pt)
IL (1) IL135515A0 (pt)
NO (1) NO20001897L (pt)
OA (1) OA11519A (pt)
PL (1) PL339804A1 (pt)
SK (1) SK5322000A3 (pt)
TR (1) TR200000957T2 (pt)
UA (1) UA66809C2 (pt)
WO (1) WO1999018944A1 (pt)
YU (1) YU28700A (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200100207T2 (tr) * 1998-07-21 2001-05-21 Smithkline Beecham P.L.C. Apoptozun redüksiyonu için glükoz alımını kuvvetlendirici maddenin kullanıması

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0842925A1 (en) * 1987-09-04 1998-05-20 Beecham Group Plc Substituted thiazolidinedione derivatives
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
US5478852C1 (en) * 1993-09-15 2001-03-13 Sankyo Co Use of thiazolidinedione derivatives and related antihyperglycemic agents in the treatment of impaired glucose tolerance in order to prevent or delay the onset of noninsulin-dependent diabetes mellitus

Also Published As

Publication number Publication date
OA11519A (en) 2004-02-09
NO20001897L (no) 2000-06-09
WO1999018944A1 (en) 1999-04-22
PL339804A1 (en) 2001-01-02
HRP20000256A2 (en) 2000-12-31
EA200000418A1 (ru) 2000-10-30
EP1023057A1 (en) 2000-08-02
YU28700A (sh) 2003-10-31
AP1223A (en) 2003-11-13
CA2305289A1 (en) 1999-04-22
UA66809C2 (uk) 2004-06-15
JP2001519383A (ja) 2001-10-23
GB9721692D0 (en) 1997-12-10
TR200000957T2 (tr) 2000-08-21
KR20010024482A (ko) 2001-03-26
IL135515A0 (en) 2001-05-20
CN1281358A (zh) 2001-01-24
AU9547198A (en) 1999-05-03
HUP0003673A3 (en) 2001-12-28
AP2000001788A0 (en) 2000-06-30
CZ20001298A3 (cs) 2001-08-15
ID24439A (id) 2000-07-20
BG104405A (en) 2000-12-29
SK5322000A3 (en) 2000-09-12
NO20001897D0 (no) 2000-04-12
HUP0003673A2 (hu) 2001-10-28

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO DE PATENTE DE ACORDO COM ART. 8O DA LPI.