BR9810554A - Aroil piperazinas para regular a atividade sexual - Google Patents

Aroil piperazinas para regular a atividade sexual

Info

Publication number
BR9810554A
BR9810554A BR9810554-0A BR9810554A BR9810554A BR 9810554 A BR9810554 A BR 9810554A BR 9810554 A BR9810554 A BR 9810554A BR 9810554 A BR9810554 A BR 9810554A
Authority
BR
Brazil
Prior art keywords
aroil
piperazines
sexual activity
regulate
sexual
Prior art date
Application number
BR9810554-0A
Other languages
English (en)
Inventor
Alexander B Zolotoy
Eric S Hayes
Original Assignee
Nortran Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nortran Pharmaceuticals Inc filed Critical Nortran Pharmaceuticals Inc
Publication of BR9810554A publication Critical patent/BR9810554A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence

Abstract

"AROIL PIPERAZINAS PARA REGULAR A ATIVIDADE SEXUAL" A presente invenção revela que derivados do ácido acético substituído contendo frações de N-alquil piperazina são úteis como agentes pró-libido para machos e fêmeas, e podem ser usados no tratamento de disfunção sexual incluindo a impotência e para estimular o desempenho sexual.
BR9810554-0A 1997-07-09 1998-07-09 Aroil piperazinas para regular a atividade sexual BR9810554A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5205197P 1997-07-09 1997-07-09
PCT/CA1998/000662 WO1999002159A1 (en) 1997-07-09 1998-07-09 Aroylpiperazines for modulating sexual activity

Publications (1)

Publication Number Publication Date
BR9810554A true BR9810554A (pt) 2000-08-15

Family

ID=21975120

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9810554-0A BR9810554A (pt) 1997-07-09 1998-07-09 Aroil piperazinas para regular a atividade sexual

Country Status (10)

Country Link
US (1) US6399618B1 (pt)
EP (1) EP1001776A1 (pt)
JP (1) JP2001509482A (pt)
CN (1) CN1269719A (pt)
AU (1) AU8203398A (pt)
BR (1) BR9810554A (pt)
CA (1) CA2295640A1 (pt)
IL (1) IL133822A0 (pt)
TW (1) TWI227139B (pt)
WO (1) WO1999002159A1 (pt)

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US6399618B1 (en) 1997-07-09 2002-06-04 Cardiome Pharma Corp Compositions and methods for modulating sexual activity
BRPI9909282B8 (pt) 1998-04-01 2021-07-06 Cardiome Pharma Corp compostos de Éter aminociclohexÍlicos e usos dos mesmos.
WO2000002550A2 (en) * 1998-07-08 2000-01-20 Nortran Pharmaceuticals, Inc. Acetylpiperazines for modulating sexual activity
WO2000028993A1 (en) * 1998-11-19 2000-05-25 Nortran Pharmaceuticals, Inc. Serotonin ligands as pro-erectile compounds
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US7057053B2 (en) 2000-10-06 2006-06-06 Cardiome Pharma Corp. Ion channel modulating compounds and uses thereof
US7524879B2 (en) 2000-10-06 2009-04-28 Cardiome Pharma Corp. Ion channel modulating compounds and uses thereof
US20020091129A1 (en) * 2000-11-20 2002-07-11 Mitradev Boolell Treatment of premature ejaculation
CA2440920C (en) * 2001-03-16 2012-01-24 David Bar-Or Use of tramadol to delay ejaculation
EP1421071B1 (en) * 2001-07-02 2009-11-18 High Point Pharmaceuticals, LLC Substituted piperazine and diazepane derivaives as histamine h3 receptor modulators
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US8058304B2 (en) 2004-04-01 2011-11-15 Cardiome Pharma Corp. Merged ion channel modulating compounds and uses thereof
JP5173190B2 (ja) 2004-08-25 2013-03-27 武田薬品工業株式会社 腹圧性尿失禁の予防・治療剤及びそのスクリーニング方法
JP5583325B2 (ja) 2004-11-08 2014-09-03 カーディオム ファーマ コーポレイション イオンチャネル調節化合物の投与レジメ
US7618972B2 (en) 2005-03-21 2009-11-17 Pfizer Inc Substituted triazole derivatives as oxytocin antagonists
EP2018863B9 (en) 2006-05-16 2015-02-18 Takeda Pharmaceutical Company Limited Fused heterocyclic compound and use thereof
WO2009063992A1 (ja) 2007-11-15 2009-05-22 Takeda Pharmaceutical Company Limited 縮合ピリジン誘導体およびその用途
US20120253036A1 (en) 2009-12-11 2012-10-04 Yukinori Nagakura Agent for treating fibromyalgia
US20210052600A1 (en) 2017-12-27 2021-02-25 Takeda Pharmaceutical Company Limited Therapeutic agents for stress urinary incontinence and incotinence of feces

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WO2000002550A2 (en) 1998-07-08 2000-01-20 Nortran Pharmaceuticals, Inc. Acetylpiperazines for modulating sexual activity

Also Published As

Publication number Publication date
CN1269719A (zh) 2000-10-11
WO1999002159A1 (en) 1999-01-21
JP2001509482A (ja) 2001-07-24
US6399618B1 (en) 2002-06-04
IL133822A0 (en) 2001-04-30
TWI227139B (en) 2005-02-01
CA2295640A1 (en) 1999-01-21
EP1001776A1 (en) 2000-05-24
AU8203398A (en) 1999-02-08

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]