BR9509875A - Oximas-42 de rapamicina e hidroxilaminas - Google Patents
Oximas-42 de rapamicina e hidroxilaminasInfo
- Publication number
- BR9509875A BR9509875A BR9509875A BR9509875A BR9509875A BR 9509875 A BR9509875 A BR 9509875A BR 9509875 A BR9509875 A BR 9509875A BR 9509875 A BR9509875 A BR 9509875A BR 9509875 A BR9509875 A BR 9509875A
- Authority
- BR
- Brazil
- Prior art keywords
- alkyl
- independently
- hydroxylamines
- oximes
- rapamycin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/350,557 US5563145A (en) | 1994-12-07 | 1994-12-07 | Rapamycin 42-oximes and hydroxylamines |
PCT/US1995/015901 WO1996017845A1 (en) | 1994-12-07 | 1995-12-06 | Rapamycin 42-oximes and hydroxylamines |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9509875A true BR9509875A (pt) | 1997-09-30 |
Family
ID=23377241
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9509875A BR9509875A (pt) | 1994-12-07 | 1995-12-06 | Oximas-42 de rapamicina e hidroxilaminas |
Country Status (22)
Country | Link |
---|---|
US (2) | US5563145A (pt) |
EP (1) | EP0796260B1 (pt) |
JP (1) | JPH10510270A (pt) |
KR (1) | KR100380870B1 (pt) |
CN (1) | CN1085212C (pt) |
AT (1) | ATE202357T1 (pt) |
AU (1) | AU714120B2 (pt) |
BR (1) | BR9509875A (pt) |
CA (1) | CA2206965A1 (pt) |
CZ (1) | CZ172097A3 (pt) |
DE (1) | DE69521438T2 (pt) |
DK (1) | DK0796260T3 (pt) |
ES (1) | ES2157353T3 (pt) |
GR (1) | GR3036209T3 (pt) |
HK (1) | HK1002361A1 (pt) |
HU (1) | HU223471B1 (pt) |
MX (1) | MX9704057A (pt) |
NZ (1) | NZ298639A (pt) |
PT (1) | PT796260E (pt) |
RU (1) | RU2172316C2 (pt) |
UA (1) | UA49815C2 (pt) |
WO (1) | WO1996017845A1 (pt) |
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US5260300A (en) * | 1992-11-19 | 1993-11-09 | American Home Products Corporation | Rapamycin carbonate esters as immuno-suppressant agents |
US5373014A (en) * | 1993-10-08 | 1994-12-13 | American Home Products Corporation | Rapamycin oximes |
US5378836A (en) * | 1993-10-08 | 1995-01-03 | American Home Products Corporation | Rapamycin oximes and hydrazones |
US5385910A (en) * | 1993-11-22 | 1995-01-31 | American Home Products Corporation | Gem-distributed esters of rapamycin |
US5385908A (en) * | 1993-11-22 | 1995-01-31 | American Home Products Corporation | Hindered esters of rapamycin |
US5385909A (en) * | 1993-11-22 | 1995-01-31 | American Home Products Corporation | Heterocyclic esters of rapamycin |
-
1994
- 1994-12-07 US US08/350,557 patent/US5563145A/en not_active Expired - Lifetime
-
1995
- 1995-12-06 BR BR9509875A patent/BR9509875A/pt not_active IP Right Cessation
- 1995-12-06 AU AU44176/96A patent/AU714120B2/en not_active Ceased
- 1995-12-06 EP EP95943018A patent/EP0796260B1/en not_active Expired - Lifetime
- 1995-12-06 CA CA002206965A patent/CA2206965A1/en not_active Abandoned
- 1995-12-06 AT AT95943018T patent/ATE202357T1/de not_active IP Right Cessation
- 1995-12-06 HU HU9701907A patent/HU223471B1/hu not_active IP Right Cessation
- 1995-12-06 UA UA97073588A patent/UA49815C2/uk unknown
- 1995-12-06 DE DE69521438T patent/DE69521438T2/de not_active Expired - Fee Related
- 1995-12-06 MX MX9704057A patent/MX9704057A/es not_active IP Right Cessation
- 1995-12-06 NZ NZ298639A patent/NZ298639A/xx unknown
- 1995-12-06 JP JP8517769A patent/JPH10510270A/ja not_active Withdrawn
- 1995-12-06 RU RU97111872/04A patent/RU2172316C2/ru not_active IP Right Cessation
- 1995-12-06 WO PCT/US1995/015901 patent/WO1996017845A1/en not_active Application Discontinuation
- 1995-12-06 CN CN95197475A patent/CN1085212C/zh not_active Expired - Fee Related
- 1995-12-06 PT PT95943018T patent/PT796260E/pt unknown
- 1995-12-06 ES ES95943018T patent/ES2157353T3/es not_active Expired - Lifetime
- 1995-12-06 DK DK95943018T patent/DK0796260T3/da active
- 1995-12-06 CZ CZ971720A patent/CZ172097A3/cs unknown
- 1995-12-06 KR KR1019970703753A patent/KR100380870B1/ko not_active IP Right Cessation
-
1996
- 1996-05-30 US US08/655,424 patent/US5677295A/en not_active Expired - Lifetime
-
1998
- 1998-02-20 HK HK98101335A patent/HK1002361A1/xx not_active IP Right Cessation
-
2001
- 2001-07-11 GR GR20010401062T patent/GR3036209T3/el not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
GR3036209T3 (en) | 2001-10-31 |
EP0796260B1 (en) | 2001-06-20 |
JPH10510270A (ja) | 1998-10-06 |
EP0796260A1 (en) | 1997-09-24 |
PT796260E (pt) | 2001-09-28 |
NZ298639A (en) | 1999-11-29 |
MX9704057A (es) | 1997-08-30 |
UA49815C2 (uk) | 2002-10-15 |
AU4417696A (en) | 1996-06-26 |
CN1085212C (zh) | 2002-05-22 |
DK0796260T3 (da) | 2001-09-03 |
HU223471B1 (hu) | 2004-07-28 |
HK1002361A1 (en) | 1998-08-21 |
HUT77141A (hu) | 1998-03-02 |
ATE202357T1 (de) | 2001-07-15 |
AU714120B2 (en) | 1999-12-16 |
CA2206965A1 (en) | 1996-06-13 |
DE69521438T2 (de) | 2002-05-16 |
US5563145A (en) | 1996-10-08 |
KR100380870B1 (ko) | 2003-10-04 |
DE69521438D1 (de) | 2001-07-26 |
WO1996017845A1 (en) | 1996-06-13 |
RU2172316C2 (ru) | 2001-08-20 |
US5677295A (en) | 1997-10-14 |
CZ172097A3 (cs) | 1998-01-14 |
ES2157353T3 (es) | 2001-08-16 |
CN1174554A (zh) | 1998-02-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 9A E 10A ANUIDADES. |
|
B25D | Requested change of name of applicant approved |
Owner name: WYETH (US) Free format text: ALTERADO DE: AMERICAN HOME PRODUCTS CORPORATION |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 9A E 10A ANUIDADES. |