BR112023025459A2 - Inibidores da tirosina quinase de bruton e métodos de uso dos mesmos - Google Patents
Inibidores da tirosina quinase de bruton e métodos de uso dos mesmosInfo
- Publication number
- BR112023025459A2 BR112023025459A2 BR112023025459A BR112023025459A BR112023025459A2 BR 112023025459 A2 BR112023025459 A2 BR 112023025459A2 BR 112023025459 A BR112023025459 A BR 112023025459A BR 112023025459 A BR112023025459 A BR 112023025459A BR 112023025459 A2 BR112023025459 A2 BR 112023025459A2
- Authority
- BR
- Brazil
- Prior art keywords
- methods
- tyrosine kinase
- kinase inhibitors
- bruton
- malignancies
- Prior art date
Links
- 102000001714 Agammaglobulinaemia Tyrosine Kinase Human genes 0.000 title abstract 2
- 108010029445 Agammaglobulinaemia Tyrosine Kinase Proteins 0.000 title abstract 2
- 229940121358 tyrosine kinase inhibitor Drugs 0.000 title abstract 2
- 239000005483 tyrosine kinase inhibitor Substances 0.000 title abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000036210 malignancy Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
- A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
nibidores da tirosina quinase de bruton e métodos de uso dos mesmos. a presente invenção refere-se ao uso de um composto da fórmula (iii) no tratamento de malignidades.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202163196843P | 2021-06-04 | 2021-06-04 | |
PCT/IB2022/055154 WO2022254371A1 (en) | 2021-06-04 | 2022-06-02 | Inhibitors of bruton's tyrosine kinase and methods of their use |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112023025459A2 true BR112023025459A2 (pt) | 2024-02-27 |
Family
ID=82214195
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112023025459A BR112023025459A2 (pt) | 2021-06-04 | 2022-06-02 | Inibidores da tirosina quinase de bruton e métodos de uso dos mesmos |
Country Status (13)
Country | Link |
---|---|
US (1) | US20230013755A1 (pt) |
EP (1) | EP4346834A1 (pt) |
JP (1) | JP2024520630A (pt) |
KR (1) | KR20240019214A (pt) |
CN (1) | CN117412753A (pt) |
AU (1) | AU2022284369A1 (pt) |
BR (1) | BR112023025459A2 (pt) |
CA (1) | CA3220015A1 (pt) |
CL (1) | CL2023003564A1 (pt) |
IL (1) | IL308951A (pt) |
MX (1) | MX2023014435A (pt) |
TW (1) | TW202317127A (pt) |
WO (1) | WO2022254371A1 (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11964976B1 (en) | 2023-09-12 | 2024-04-23 | King Faisal University | Substituted pyrido[3′,4′:4,5]pyrrolo[3,2-c][1,6]naphthyridines as CK2 inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2887697A1 (en) | 2012-10-11 | 2014-04-17 | Pharmacyclics, Inc. | Companion diagnostics for tec family kinase inhibitor therapy |
DK3179991T3 (da) * | 2014-08-11 | 2021-12-06 | Acerta Pharma Bv | Terapeutiske kombinationer af en btk-inhibitor og en bcl-2-inhibitor |
JO3794B1 (ar) | 2015-12-10 | 2021-01-31 | Janssen Pharmaceutica Nv | المركبات متعددة الحلقات كمثبطات لتيروزين كيناز بروتون |
WO2018103060A1 (en) * | 2016-12-09 | 2018-06-14 | Janssen Pharmaceutica Nv | Inhibitors of bruton's tyrosine kinase and methods of their use |
-
2022
- 2022-06-02 CA CA3220015A patent/CA3220015A1/en active Pending
- 2022-06-02 BR BR112023025459A patent/BR112023025459A2/pt unknown
- 2022-06-02 JP JP2023574315A patent/JP2024520630A/ja active Pending
- 2022-06-02 IL IL308951A patent/IL308951A/en unknown
- 2022-06-02 MX MX2023014435A patent/MX2023014435A/es unknown
- 2022-06-02 KR KR1020247000043A patent/KR20240019214A/ko unknown
- 2022-06-02 EP EP22733732.6A patent/EP4346834A1/en active Pending
- 2022-06-02 US US17/830,714 patent/US20230013755A1/en active Pending
- 2022-06-02 AU AU2022284369A patent/AU2022284369A1/en active Pending
- 2022-06-02 CN CN202280039736.2A patent/CN117412753A/zh active Pending
- 2022-06-02 WO PCT/IB2022/055154 patent/WO2022254371A1/en active Application Filing
- 2022-06-02 TW TW111120615A patent/TW202317127A/zh unknown
-
2023
- 2023-11-29 CL CL2023003564A patent/CL2023003564A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
TW202317127A (zh) | 2023-05-01 |
AU2022284369A1 (en) | 2024-01-25 |
CL2023003564A1 (es) | 2024-06-21 |
IL308951A (en) | 2024-01-01 |
WO2022254371A1 (en) | 2022-12-08 |
US20230013755A1 (en) | 2023-01-19 |
KR20240019214A (ko) | 2024-02-14 |
EP4346834A1 (en) | 2024-04-10 |
MX2023014435A (es) | 2024-03-08 |
CN117412753A (zh) | 2024-01-16 |
JP2024520630A (ja) | 2024-05-24 |
CA3220015A1 (en) | 2022-12-08 |
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