BR112022015507A2 - Processos para produzir compostos de amida, e sua forma cristalina e salina - Google Patents
Processos para produzir compostos de amida, e sua forma cristalina e salinaInfo
- Publication number
- BR112022015507A2 BR112022015507A2 BR112022015507A BR112022015507A BR112022015507A2 BR 112022015507 A2 BR112022015507 A2 BR 112022015507A2 BR 112022015507 A BR112022015507 A BR 112022015507A BR 112022015507 A BR112022015507 A BR 112022015507A BR 112022015507 A2 BR112022015507 A2 BR 112022015507A2
- Authority
- BR
- Brazil
- Prior art keywords
- amide compounds
- crystalline
- processes
- producing amide
- saline form
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/10—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
- C07D271/107—1,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with two aryl or substituted aryl radicals attached in positions 2 and 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C313/02—Sulfinic acids; Derivatives thereof
- C07C313/06—Sulfinamides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Abstract
PROCESSOS PARA PRODUZIR COMPOSTOS DE AMIDA, E SUA FORMA CRISTALINA E SALINA. São divulgados processos para produzir compostos de amida, e sua forma cristalina e salina. Neste documento, um dos compostos de amida é representado pela seguinte Fórmula (1): que é caracterizado por um padrão de difração de raios x (XRD) tendo picos em cerca de 14,2, 15,6, 16,4, 20,1, 20,5 e 21,2° ± 0,2° 2Teta.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202062985918P | 2020-03-06 | 2020-03-06 | |
PCT/US2021/020595 WO2021178486A1 (en) | 2020-03-06 | 2021-03-03 | Processes for producing amide compounds, and their crystalline and salt form |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112022015507A2 true BR112022015507A2 (pt) | 2022-09-27 |
Family
ID=77613709
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112022015507A BR112022015507A2 (pt) | 2020-03-06 | 2021-03-03 | Processos para produzir compostos de amida, e sua forma cristalina e salina |
Country Status (12)
Country | Link |
---|---|
US (1) | US20230131180A1 (pt) |
EP (1) | EP4114823A4 (pt) |
JP (1) | JP2023516082A (pt) |
KR (1) | KR20220137084A (pt) |
CN (1) | CN115052855A (pt) |
AU (2) | AU2021231787B2 (pt) |
BR (1) | BR112022015507A2 (pt) |
CA (1) | CA3170348A1 (pt) |
IL (1) | IL296041A (pt) |
MX (1) | MX2022011025A (pt) |
TW (1) | TWI787751B (pt) |
WO (1) | WO2021178486A1 (pt) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MX2013006768A (es) * | 2010-12-23 | 2013-07-22 | Pfizer | Moduladores de receptor de glucagon. |
EA023517B1 (ru) * | 2011-02-08 | 2016-06-30 | Пфайзер Инк. | Модуляторы глюкагонового рецептора |
US10882837B2 (en) * | 2017-01-24 | 2021-01-05 | Alphala Co., Ltd. | Amide compounds and use thereof |
EP3640242B1 (en) * | 2017-06-16 | 2023-04-19 | Hitgen Ltd. | Rock-inhibiting compound and uses thereof |
-
2021
- 2021-03-03 MX MX2022011025A patent/MX2022011025A/es unknown
- 2021-03-03 KR KR1020227030617A patent/KR20220137084A/ko unknown
- 2021-03-03 CN CN202180012870.9A patent/CN115052855A/zh active Pending
- 2021-03-03 EP EP21765102.5A patent/EP4114823A4/en active Pending
- 2021-03-03 AU AU2021231787A patent/AU2021231787B2/en active Active
- 2021-03-03 IL IL296041A patent/IL296041A/en unknown
- 2021-03-03 CA CA3170348A patent/CA3170348A1/en active Pending
- 2021-03-03 WO PCT/US2021/020595 patent/WO2021178486A1/en active Application Filing
- 2021-03-03 BR BR112022015507A patent/BR112022015507A2/pt unknown
- 2021-03-03 US US17/908,133 patent/US20230131180A1/en active Pending
- 2021-03-03 JP JP2022553034A patent/JP2023516082A/ja active Pending
- 2021-03-04 TW TW110107674A patent/TWI787751B/zh active
-
2023
- 2023-11-17 AU AU2023266374A patent/AU2023266374A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
AU2021231787A1 (en) | 2022-08-25 |
WO2021178486A1 (en) | 2021-09-10 |
EP4114823A4 (en) | 2024-06-19 |
MX2022011025A (es) | 2022-10-07 |
AU2021231787B2 (en) | 2023-08-17 |
US20230131180A1 (en) | 2023-04-27 |
CA3170348A1 (en) | 2021-09-10 |
CN115052855A (zh) | 2022-09-13 |
JP2023516082A (ja) | 2023-04-17 |
TW202142534A (zh) | 2021-11-16 |
EP4114823A1 (en) | 2023-01-11 |
AU2023266374A1 (en) | 2023-12-07 |
IL296041A (en) | 2022-10-01 |
TWI787751B (zh) | 2022-12-21 |
KR20220137084A (ko) | 2022-10-11 |
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