BR112019012224A2 - compostos de benzimidazol como inibidores de c-kit - Google Patents
compostos de benzimidazol como inibidores de c-kit Download PDFInfo
- Publication number
- BR112019012224A2 BR112019012224A2 BR112019012224-9A BR112019012224A BR112019012224A2 BR 112019012224 A2 BR112019012224 A2 BR 112019012224A2 BR 112019012224 A BR112019012224 A BR 112019012224A BR 112019012224 A2 BR112019012224 A2 BR 112019012224A2
- Authority
- BR
- Brazil
- Prior art keywords
- methyl
- trifluoromethyl
- imidazol
- benzo
- ethynyl
- Prior art date
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- 102000016971 Proto-Oncogene Proteins c-kit Human genes 0.000 title claims abstract description 56
- 108010014608 Proto-Oncogene Proteins c-kit Proteins 0.000 title claims abstract description 56
- 239000003112 inhibitor Substances 0.000 title abstract description 8
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| EP4359411A1 (en) | 2021-06-23 | 2024-05-01 | Gilead Sciences, Inc. | Diacylglyercol kinase modulating compounds |
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| PE20241186A1 (es) | 2021-10-29 | 2024-06-03 | Gilead Sciences Inc | Compuestos de cd73 |
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2017
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- 2017-12-14 AU AU2017376629A patent/AU2017376629B2/en not_active Ceased
- 2017-12-14 CN CN201780085539.3A patent/CN110291081B/zh active Active
- 2017-12-14 IL IL314209A patent/IL314209A/en unknown
- 2017-12-14 WO PCT/US2017/066299 patent/WO2018112140A1/en not_active Application Discontinuation
- 2017-12-14 JP JP2019531992A patent/JP7158383B2/ja active Active
- 2017-12-14 US US16/469,535 patent/US11117883B2/en active Active
- 2017-12-14 IL IL287517A patent/IL287517B2/en unknown
- 2017-12-14 CA CA3047107A patent/CA3047107A1/en active Pending
- 2017-12-14 MA MA053150A patent/MA53150A/fr unknown
- 2017-12-14 CN CN202211731994.5A patent/CN116178343A/zh active Pending
- 2017-12-14 BR BR112019012224-9A patent/BR112019012224A2/pt not_active Application Discontinuation
- 2017-12-14 EA EA201991197A patent/EA201991197A1/ru unknown
- 2017-12-14 KR KR1020197020159A patent/KR20190092538A/ko not_active Abandoned
- 2017-12-14 MX MX2019007080A patent/MX390348B/es unknown
- 2017-12-14 CN CN202211737801.7A patent/CN116283910A/zh active Pending
-
2019
- 2019-06-12 IL IL267260A patent/IL267260B2/en unknown
- 2019-06-14 MX MX2022002581A patent/MX2022002581A/es unknown
-
2021
- 2021-08-12 US US17/400,820 patent/US20220064144A1/en not_active Abandoned
-
2022
- 2022-02-18 AU AU2022201082A patent/AU2022201082B2/en not_active Ceased
- 2022-10-11 JP JP2022163367A patent/JP2022185110A/ja active Pending
-
2024
- 2024-02-01 AU AU2024200624A patent/AU2024200624A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EA201991197A1 (ru) | 2020-01-13 |
| US20200039958A1 (en) | 2020-02-06 |
| MA53150A (fr) | 2021-05-26 |
| KR20190092538A (ko) | 2019-08-07 |
| IL287517A (en) | 2021-12-01 |
| IL314209A (en) | 2024-09-01 |
| AU2017376629B2 (en) | 2021-11-25 |
| CN110291081A (zh) | 2019-09-27 |
| CN116283910A (zh) | 2023-06-23 |
| CN110291081B (zh) | 2023-01-31 |
| MX2022002581A (es) | 2022-03-22 |
| MX2019007080A (es) | 2019-10-15 |
| IL267260A (en) | 2019-08-29 |
| AU2024200624A1 (en) | 2024-02-22 |
| CN116178343A (zh) | 2023-05-30 |
| US20220064144A1 (en) | 2022-03-03 |
| CA3047107A1 (en) | 2018-06-21 |
| AU2017376629A1 (en) | 2019-07-04 |
| JP7158383B2 (ja) | 2022-10-21 |
| JP2022185110A (ja) | 2022-12-13 |
| IL287517B1 (en) | 2024-08-01 |
| MX390348B (es) | 2025-03-20 |
| WO2018112140A1 (en) | 2018-06-21 |
| EP3555066A1 (en) | 2019-10-23 |
| AU2022201082B2 (en) | 2023-11-02 |
| IL267260B (en) | 2022-10-01 |
| JP2020503299A (ja) | 2020-01-30 |
| US11117883B2 (en) | 2021-09-14 |
| AU2022201082A1 (en) | 2022-03-10 |
| IL267260B2 (en) | 2023-02-01 |
| IL287517B2 (en) | 2024-12-01 |
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Legal Events
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| B06W | Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette] | ||
| B350 | Update of information on the portal [chapter 15.35 patent gazette] | ||
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |