BR112018006414A2 - processo para produzir fosfinatos - Google Patents

processo para produzir fosfinatos

Info

Publication number
BR112018006414A2
BR112018006414A2 BR112018006414-9A BR112018006414A BR112018006414A2 BR 112018006414 A2 BR112018006414 A2 BR 112018006414A2 BR 112018006414 A BR112018006414 A BR 112018006414A BR 112018006414 A2 BR112018006414 A2 BR 112018006414A2
Authority
BR
Brazil
Prior art keywords
phosphinates
produce
production
phosphorus
pharmaceutical
Prior art date
Application number
BR112018006414-9A
Other languages
English (en)
Other versions
BR112018006414B1 (pt
Inventor
Ressel Hans-Joachim
Original Assignee
Bayer Cropscience Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Aktiengesellschaft filed Critical Bayer Cropscience Aktiengesellschaft
Publication of BR112018006414A2 publication Critical patent/BR112018006414A2/pt
Publication of BR112018006414B1 publication Critical patent/BR112018006414B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/48—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
    • C07F9/4866—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof the ester moiety containing a substituent or structure which is considered as characteristic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/32—Esters thereof
    • C07F9/3205—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/3211—Esters of acyclic saturated acids which can have further substituents on alkyl
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having alternatively specified atoms bound to the phosphorus atom and not covered by a single one of groups A01N57/10, A01N57/18, A01N57/26, A01N57/34
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J27/00—Catalysts comprising the elements or compounds of halogens, sulfur, selenium, tellurium, phosphorus or nitrogen; Catalysts comprising carbon compounds
    • B01J27/14—Phosphorus; Compounds thereof
    • B01J27/16—Phosphorus; Compounds thereof containing oxygen, i.e. acids, anhydrides and their derivates with N, S, B or halogens without carriers or on carriers based on C, Si, Al or Zr; also salts of Si, Al and Zr
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/301—Acyclic saturated acids which can have further substituents on alkyl
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/32—Esters thereof
    • C07F9/3205—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/3223—Esters of cycloaliphatic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4071—Esters thereof the ester moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4075—Esters with hydroxyalkyl compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Materials Engineering (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

processo para produzir fosfinatos. a presente invenção refere-se principalmente a um processo para particularmente produzir fosfinatos (monoésteres de ácido fosfônico) e seu uso para a produção de substâncias biologicamente ativas que podem ser usadas no setor farmacêutico ou agroquímico, de preferência para a produção de aminoácidos contendo fósforo.
BR112018006414-9A 2015-09-29 2016-09-26 processo para produzir fosfinatos BR112018006414B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15187469 2015-09-29
EP15187469.0 2015-09-29
PCT/EP2016/072786 WO2017055193A1 (de) 2015-09-29 2016-09-26 Verfahren zur Herstellung von Phosphinaten

Publications (2)

Publication Number Publication Date
BR112018006414A2 true BR112018006414A2 (pt) 2018-10-09
BR112018006414B1 BR112018006414B1 (pt) 2020-11-24

Family

ID=54252056

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112018006414-9A BR112018006414B1 (pt) 2015-09-29 2016-09-26 processo para produzir fosfinatos

Country Status (11)

Country Link
US (2) US10501485B2 (pt)
EP (1) EP3356376B1 (pt)
JP (1) JP6826110B2 (pt)
KR (1) KR20180059466A (pt)
CN (1) CN108137629B (pt)
BR (1) BR112018006414B1 (pt)
ES (1) ES2754603T3 (pt)
IL (1) IL258301A (pt)
MX (1) MX2018003962A (pt)
TW (1) TWI721019B (pt)
WO (1) WO2017055193A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201840578A (zh) * 2017-02-22 2018-11-16 以色列商亞當阿甘公司 製備甲基膦酸丁基酯的方法
CN110386950A (zh) * 2019-07-18 2019-10-29 石家庄瑞凯化工有限公司 一种草铵膦铵盐的合成方法
CN111909199B (zh) * 2020-08-06 2021-09-14 浙江新安化工集团股份有限公司 一种甲基亚膦酸二乙酯精馏高沸物资源化利用的方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3914345A (en) 1971-01-08 1975-10-21 Hoechst Ag Process for the manufacture of dialkyl-phosphinic acid esters
DE2415757C2 (de) 1974-04-01 1982-10-14 Hoechst Ag, 6000 Frankfurt Verfahren zur Herstellung phosphorhaltiger Ester
DE2519192C2 (de) 1975-04-30 1983-08-04 Hoechst Ag, 6230 Frankfurt Verfahren zur Herstellung phosphorhaltiger Ester
DE2717440C2 (de) * 1976-05-17 1984-04-05 Hoechst Ag, 6230 Frankfurt Unkrautbekämpfung mit [(3-Amino-3-carboxy)-propyl-1]-methylphosphinsäure-Derivaten
DE2849003A1 (de) 1978-11-11 1980-08-21 Hoechst Ag Phosphorhaltige cyanhydrinderivate und verfahren zu ihrer herstellung
DE3146197A1 (de) 1981-11-21 1983-05-26 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung von phosphonigsaeuremonoalkylestern
DE3146196A1 (de) 1981-11-21 1983-05-26 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung phosphoniger saeuren
DE3319850C2 (de) * 1983-06-01 1985-05-09 Hoechst Ag, 6230 Frankfurt Verfahren zur Herstellung von phosphorhaltigen Cyanhydrinderivaten
US5166385A (en) 1989-03-23 1992-11-24 Hoechst Aktiengesellschaft Process for the preparation of phosphino compounds
DE3911230A1 (de) 1989-04-07 1990-10-11 Hoechst Ag Verfahren zur herstellung von alkylphosphonigsaeurediestern und/oder dialkylphosphinigsaeureestern
DE19736125A1 (de) 1997-08-20 1999-02-25 Hoechst Schering Agrevo Gmbh Verfahren zur Herstellung von Glufosinate und phosphorhaltige alpha-Aminonitrile als Zwischenprodukte
CN104892670A (zh) * 2015-05-13 2015-09-09 安徽国星生物化学有限公司 一种草铵膦及其类似物的制备方法

Also Published As

Publication number Publication date
TW201726694A (zh) 2017-08-01
US20180265529A1 (en) 2018-09-20
JP6826110B2 (ja) 2021-02-03
IL258301A (en) 2018-05-31
TWI721019B (zh) 2021-03-11
US20200079804A1 (en) 2020-03-12
US10968241B2 (en) 2021-04-06
MX2018003962A (es) 2018-06-08
ES2754603T3 (es) 2020-04-20
CN108137629A (zh) 2018-06-08
JP2018534260A (ja) 2018-11-22
WO2017055193A1 (de) 2017-04-06
BR112018006414B1 (pt) 2020-11-24
KR20180059466A (ko) 2018-06-04
EP3356376B1 (de) 2019-08-07
US10501485B2 (en) 2019-12-10
EP3356376A1 (de) 2018-08-08
CN108137629B (zh) 2020-09-01

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Legal Events

Date Code Title Description
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 26/09/2016, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 6A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2689 DE 19-07-2022 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.