BR112017024665A2 - compostos pirazol substituídos contendo pirimidinila, preparação e aplicação dos mesmos - Google Patents

compostos pirazol substituídos contendo pirimidinila, preparação e aplicação dos mesmos

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Publication number
BR112017024665A2
BR112017024665A2 BR112017024665-1A BR112017024665A BR112017024665A2 BR 112017024665 A2 BR112017024665 A2 BR 112017024665A2 BR 112017024665 A BR112017024665 A BR 112017024665A BR 112017024665 A2 BR112017024665 A2 BR 112017024665A2
Authority
BR
Brazil
Prior art keywords
compounds containing
substituted pyrazole
preparation
application
pyrazole compounds
Prior art date
Application number
BR112017024665-1A
Other languages
English (en)
Chinese (zh)
Other versions
BR112017024665B1 (pt
Inventor
Liu Changling
Guan Aiying
Wang Junfeng
Sun Xufeng
Li Zhinian
Zhang Jinbo
Ban Lanfeng
Ma Sen
Lan Jie
Xia Xiaoli
Yang Jinlong
Original Assignee
Shenyang Sinochem Agrochemicals R&D Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shenyang Sinochem Agrochemicals R&D Co., Ltd. filed Critical Shenyang Sinochem Agrochemicals R&D Co., Ltd.
Publication of BR112017024665A2 publication Critical patent/BR112017024665A2/pt
Publication of BR112017024665B1 publication Critical patent/BR112017024665B1/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

o documento revela compostos pirazol substituídos contendo pirimidinila conforme mostrado na fórmula i: as definições de cada substituinte podem ser vistas na descrição. os compostos da presente invenção possuem um bom espectro de atividade bactericida, inseticida e acaricida e possuem bom efeito de controle em míldio do pepino, míldio do trigo, ferrugem do milho, mangra do arroz, antracnose do pepino e semelhantes. os compostos da presente invenção também mostram boa atividade inseticida.
BR112017024665-1A 2015-05-18 2016-05-17 Compostos pirazol substituídos contendo pirimidinila, preparação e aplicação dos mesmos BR112017024665B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201510252832.7 2015-05-18
CN201510252832 2015-05-18
PCT/CN2016/082291 WO2016184378A1 (zh) 2015-05-18 2016-05-17 含嘧啶的取代吡唑类化合物及其制备方法和用途

Publications (2)

Publication Number Publication Date
BR112017024665A2 true BR112017024665A2 (pt) 2018-11-06
BR112017024665B1 BR112017024665B1 (pt) 2023-02-23

Family

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Family Applications (2)

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BR122020001830-5A BR122020001830B1 (pt) 2015-05-18 2016-05-17 Compostos pirazol substituídos contendo pirimidinila, preparação e aplicação dos mesmos
BR112017024665-1A BR112017024665B1 (pt) 2015-05-18 2016-05-17 Compostos pirazol substituídos contendo pirimidinila, preparação e aplicação dos mesmos

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BR122020001830-5A BR122020001830B1 (pt) 2015-05-18 2016-05-17 Compostos pirazol substituídos contendo pirimidinila, preparação e aplicação dos mesmos

Country Status (11)

Country Link
US (1) US11008339B2 (pt)
EP (2) EP3702355B1 (pt)
CN (1) CN106167484B (pt)
AR (1) AR104658A1 (pt)
AU (1) AU2016264519B2 (pt)
BR (2) BR122020001830B1 (pt)
CA (1) CA2982206C (pt)
ES (1) ES2824119T3 (pt)
RU (1) RU2687089C2 (pt)
UA (2) UA127459C2 (pt)
WO (1) WO2016184378A1 (pt)

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EP3719015A4 (en) * 2017-11-29 2021-04-21 Shenyang Sinochem Agrochemicals R & D Co., Ltd. SUBSTITUTED PYRIMIDINE COMPOUND AND MANUFACTURING METHOD FOR ITS AND USES THEREOF
CN109836418A (zh) * 2017-11-29 2019-06-04 沈阳中化农药化工研发有限公司 取代吡唑类化合物及其制备方法和作为杀虫杀螨剂的用途
CN109836417A (zh) * 2017-11-29 2019-06-04 沈阳中化农药化工研发有限公司 取代嘧啶类化合物及其制备方法和作为杀菌剂的用途
CN109096194B (zh) * 2018-10-09 2022-02-08 湖南师范大学 一种双胍衍生物、药物组合物、制备方法和用途
CN111316992B (zh) * 2018-12-14 2021-07-20 沈阳中化农药化工研发有限公司 一种杀真菌组合物及应用
CN111316990B (zh) * 2018-12-14 2021-06-25 沈阳中化农药化工研发有限公司 杀真菌组合物及其应用
CN111316991B (zh) * 2018-12-14 2021-07-20 沈阳中化农药化工研发有限公司 杀真菌组合物及应用
CN111316987B (zh) * 2018-12-14 2021-06-29 沈阳中化农药化工研发有限公司 一种杀真菌组合物及其应用
CN117016550A (zh) * 2019-11-25 2023-11-10 沈阳中化农药化工研发有限公司 杀菌组合物及其应用
CN113512029B (zh) * 2020-04-10 2023-01-24 沈阳中化农药化工研发有限公司 含嘧啶胺的取代吡唑类化合物制备及其用途
CN113754636B (zh) * 2020-06-02 2022-10-04 湖南化工研究院有限公司 含喹唑啉的氮杂醚类化合物
CN115843810A (zh) * 2020-09-29 2023-03-28 沈阳中化农药化工研发有限公司 一种杀菌制剂及其应用
CN116831116A (zh) * 2022-03-23 2023-10-03 沈阳中化农药化工研发有限公司 一种含稳定剂的杀菌组合物制剂

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Also Published As

Publication number Publication date
AU2016264519B2 (en) 2018-06-28
CA2982206C (en) 2020-07-14
EP3702355B1 (en) 2022-01-12
AU2016264519A1 (en) 2017-12-14
CA2982206A1 (en) 2016-11-24
EP3299366A4 (en) 2018-11-21
EP3299366A1 (en) 2018-03-28
EP3702355A1 (en) 2020-09-02
UA124524C2 (uk) 2021-10-05
RU2017135214A (ru) 2019-04-10
BR122020001830B1 (pt) 2023-02-28
RU2687089C2 (ru) 2019-05-07
US11008339B2 (en) 2021-05-18
AR104658A1 (es) 2017-08-02
BR112017024665B1 (pt) 2023-02-23
US20180141961A1 (en) 2018-05-24
UA127459C2 (uk) 2023-08-30
CN106167484B (zh) 2020-03-17
RU2017135214A3 (pt) 2019-04-10
EP3299366B1 (en) 2020-09-09
WO2016184378A1 (zh) 2016-11-24
ES2824119T3 (es) 2021-05-11
CN106167484A (zh) 2016-11-30

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