BR112017018977A2 - ?composto, composição farmacêutica, métodos para tratamento de uma infecção por hepatite c ou uma condição resultante de uma infecção por hepatite c, em um hospedeiro em necessidade do mesmo e para fabricação de um medicamento direcionado para uso terapêutico para tratamento de uma infecção pelo vírus da hepatite c, uso de um composto, e, formulação farmacêutica?. - Google Patents

?composto, composição farmacêutica, métodos para tratamento de uma infecção por hepatite c ou uma condição resultante de uma infecção por hepatite c, em um hospedeiro em necessidade do mesmo e para fabricação de um medicamento direcionado para uso terapêutico para tratamento de uma infecção pelo vírus da hepatite c, uso de um composto, e, formulação farmacêutica?.

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Publication number
BR112017018977A2
BR112017018977A2 BR112017018977-1A BR112017018977A BR112017018977A2 BR 112017018977 A2 BR112017018977 A2 BR 112017018977A2 BR 112017018977 A BR112017018977 A BR 112017018977A BR 112017018977 A2 BR112017018977 A2 BR 112017018977A2
Authority
BR
Brazil
Prior art keywords
hepatitis
infection
treating
compound
host
Prior art date
Application number
BR112017018977-1A
Other languages
English (en)
Other versions
BR112017018977B1 (pt
Inventor
Sommadossi Jean-Pierre
Moussa Adel
Original Assignee
Atea Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Atea Pharmaceuticals, Inc. filed Critical Atea Pharmaceuticals, Inc.
Publication of BR112017018977A2 publication Critical patent/BR112017018977A2/pt
Publication of BR112017018977B1 publication Critical patent/BR112017018977B1/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • C07H19/20Purine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids
    • C07H19/207Purine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids the phosphoric or polyphosphoric acids being esterified by a further hydroxylic compound, e.g. flavine adenine dinucleotide or nicotinamide-adenine dinucleotide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • C07H19/20Purine radicals with the saccharide radical esterified by phosphoric or polyphosphoric acids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicinal Preparation (AREA)

Abstract

composto da estrutura: ou um sal farmaceuticamente aceitável ou composição do mesmo para o tratamento de um hospedeiro infectado com ou exposto a um vírus ou distúrbios descritos mais completamente aqui.
BR112017018977-1A 2015-03-06 2016-03-07 Compostos nucleotídicos, composição farmacêutica, e, uso de um composto BR112017018977B1 (pt)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201562129319P 2015-03-06 2015-03-06
US62/129319 2015-03-06
US201562253958P 2015-11-11 2015-11-11
US62/253958 2015-11-11
US201662276597P 2016-01-08 2016-01-08
US62/276597 2016-01-08
PCT/US2016/021276 WO2016144918A1 (en) 2015-03-06 2016-03-07 β-D-2'-DEOXY-2'α-FLUORO-2'-β-C-SUBSTITUTED-2-MODIFIED-N6-SUBSTITUTED PURINE NUCLEOTIDES FOR HCV TREATMENT

Publications (2)

Publication Number Publication Date
BR112017018977A2 true BR112017018977A2 (pt) 2018-05-22
BR112017018977B1 BR112017018977B1 (pt) 2024-03-26

Family

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Also Published As

Publication number Publication date
GEP20217282B (en) 2021-08-10
IL254111B (en) 2021-04-29
CA2978085A1 (en) 2016-09-15
UA124966C2 (uk) 2021-12-22
KR20220025914A (ko) 2022-03-03
SA517382236B1 (ar) 2022-09-07
NZ734908A (en) 2021-10-29
US20210009628A1 (en) 2021-01-14
US10239911B2 (en) 2019-03-26
PH12017501598A1 (en) 2018-02-12
JP2022088596A (ja) 2022-06-14
AU2018282469A1 (en) 2019-01-24
US20190177356A1 (en) 2019-06-13
KR20170120700A (ko) 2017-10-31
AU2016229966A8 (en) 2017-10-12
US10815266B2 (en) 2020-10-27
CA2978085C (en) 2023-01-17
US20200331956A1 (en) 2020-10-22
JP2018507261A (ja) 2018-03-15
JP6776273B2 (ja) 2020-10-28
US20200308215A1 (en) 2020-10-01
JP2021008494A (ja) 2021-01-28
GEP20247600B (en) 2024-02-26
AU2020203055B2 (en) 2021-03-25
US20180030082A1 (en) 2018-02-01
EA201791903A1 (ru) 2018-01-31
MY190867A (en) 2022-05-13
MX2017011386A (es) 2018-04-26
US20220267366A1 (en) 2022-08-25
CA3182565A1 (en) 2016-09-15
US20200331955A1 (en) 2020-10-22
KR102363946B1 (ko) 2022-02-17
IL295418A (en) 2022-10-01
IL302877A (en) 2023-07-01
CN112209980A (zh) 2021-01-12
CN107427530A (zh) 2017-12-01
CO2017010162A2 (es) 2018-01-05
EP3265102A4 (en) 2018-12-05
JP7053754B2 (ja) 2022-04-12
CN107427530B (zh) 2020-09-08
AU2018282469B2 (en) 2020-02-13
IL254111A0 (en) 2017-10-31
US10000523B2 (en) 2018-06-19
RU2764767C2 (ru) 2022-01-21
AU2023202634A1 (en) 2023-05-18
EA037098B1 (ru) 2021-02-05
US20180030081A1 (en) 2018-02-01
US10875885B2 (en) 2020-12-29
US20160257706A1 (en) 2016-09-08
AU2020203055A1 (en) 2020-05-28
AU2016229966B2 (en) 2018-09-27
HK1247829A1 (zh) 2018-10-05
SG11201706841PA (en) 2017-09-28
AU2021204022B2 (en) 2023-05-18
US12084473B2 (en) 2024-09-10
US20180282364A1 (en) 2018-10-04
RU2017133011A3 (pt) 2019-09-13
AU2021204022A1 (en) 2021-07-08
JP7532440B2 (ja) 2024-08-13
WO2016144918A1 (en) 2016-09-15
CN112209980B (zh) 2023-12-05
ZA201705852B (en) 2019-11-27
AU2016229966A1 (en) 2017-09-14
US20240002426A1 (en) 2024-01-04
US10005811B2 (en) 2018-06-26
EP3265102A1 (en) 2018-01-10
US10870672B2 (en) 2020-12-22
US9828410B2 (en) 2017-11-28
IL295418B2 (en) 2023-10-01
US10870673B2 (en) 2020-12-22
GEP20237502B (en) 2023-04-25
IL295418B1 (en) 2023-06-01
RU2017133011A (ru) 2019-04-09
MX2022015612A (es) 2023-02-13

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B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
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