BR112017015137A2 - compostos antiparasíticos - Google Patents

compostos antiparasíticos

Info

Publication number
BR112017015137A2
BR112017015137A2 BR112017015137-5A BR112017015137A BR112017015137A2 BR 112017015137 A2 BR112017015137 A2 BR 112017015137A2 BR 112017015137 A BR112017015137 A BR 112017015137A BR 112017015137 A2 BR112017015137 A2 BR 112017015137A2
Authority
BR
Brazil
Prior art keywords
compounds
antiparasitic compounds
relates
controlling invertebrate
pests
Prior art date
Application number
BR112017015137-5A
Other languages
English (en)
Inventor
D. Speake Jason
B. Perales Joe
Fan Weiming
Clarisse Rolland Solène
Original Assignee
Avista Pharma Solutions, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Avista Pharma Solutions, Inc. filed Critical Avista Pharma Solutions, Inc.
Publication of BR112017015137A2 publication Critical patent/BR112017015137A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Catching Or Destruction (AREA)
  • Fodder In General (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

a presente invenção refere-se aos compostos de isotiazolina de fórmula (i). os compostos são úteis para combater ou controlar as pragas de invertebrados, em particular as pragas de artrópodes e os nematoides. a invenção também se refere a um método para controlar as pragas de invertebrados por utilização destes compostos e às composições veterinárias compreendendo os ditos compostos.
BR112017015137-5A 2015-01-16 2016-01-14 compostos antiparasíticos BR112017015137A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562104364P 2015-01-16 2015-01-16
US62/104,364 2015-01-16
PCT/US2016/013358 WO2016115315A1 (en) 2015-01-16 2016-01-14 Antiparasitic compounds

Publications (1)

Publication Number Publication Date
BR112017015137A2 true BR112017015137A2 (pt) 2018-01-30

Family

ID=56406368

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112017015137-5A BR112017015137A2 (pt) 2015-01-16 2016-01-14 compostos antiparasíticos

Country Status (13)

Country Link
US (6) US9420793B2 (pt)
EP (1) EP3245209B1 (pt)
JP (2) JP2018509463A (pt)
KR (1) KR20170102359A (pt)
CN (1) CN107406458B (pt)
AU (2) AU2016206748B9 (pt)
BR (1) BR112017015137A2 (pt)
CA (1) CA2973974A1 (pt)
ES (1) ES2827477T3 (pt)
GB (3) GB2572267B (pt)
MX (2) MX370163B (pt)
RU (1) RU2017128818A (pt)
WO (1) WO2016115315A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2827477T3 (es) * 2015-01-16 2021-05-21 Avista Pharma Solutions Inc Compuestos antiparasitarios
BR112018068034A2 (pt) 2016-03-09 2019-01-08 Basf Se compostos espiro da fórmula i, composição, composição agrícola para combater pragas animais, método de combate ou controle de pragas invertebradas, método de proteção de plantas, semente e uso dos compostos
US10556909B2 (en) * 2016-05-20 2020-02-11 Avista Pharma Solutions, Inc. Synthetic process and intermediates
WO2018009751A1 (en) * 2016-07-08 2018-01-11 Avista Pharma Solutions, Inc. Antiparasitic compounds
EP3710453A1 (en) * 2017-11-16 2020-09-23 Avista Pharma Solutions, Inc. Single enantiomer antiparasitic compounds
US10239885B1 (en) * 2018-06-18 2019-03-26 Avista Pharma Solutions, Inc. Compound 1-[2-[4-(2-ethyl-6,8-dimethylimidazo[1,2-α]pyrazin-3-yl)phenyl]ethyl]-3-(p-tolylsulfonyl)urea as a prostaglandin EP4 receptor antagonist
MX2021006661A (es) * 2018-12-04 2021-07-07 Basf Se Proceso para la preparacion de 5-bromo-1,3-dicloro-2-fluoro-bencen o.
CN113024390B (zh) * 2021-02-22 2023-12-05 台州臻挚生物科技有限公司 3’,5’-二氯-2,2,2-三氟苯乙酮衍生物的合成方法

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TW200803740A (en) 2005-12-16 2008-01-16 Du Pont 5-aryl isoxazolines for controlling invertebrate pests
ES2344027T3 (es) 2006-03-10 2010-08-16 Nissan Chemical Industries, Ltd. Compuesto de isoxazolina sustituido y agente de control de plagas.
WO2008096746A1 (ja) 2007-02-06 2008-08-14 Takeda Pharmaceutical Company Limited スピロ化合物およびその用途
BRPI0810196A2 (pt) 2007-04-10 2011-12-06 Bayer Cropscience Ag inseticidas de derivados de aril isoxazolina
JP5365806B2 (ja) 2007-09-10 2013-12-11 日産化学工業株式会社 置換イソキサゾリン化合物及び有害生物防除剤
JP5365807B2 (ja) 2007-11-12 2013-12-11 日産化学工業株式会社 光学活性イソキサゾリン化合物の触媒的不斉合成方法
JP2009286773A (ja) * 2008-03-14 2009-12-10 Bayer Cropscience Ag 殺虫性縮環式アリール類
EA201100421A1 (ru) 2008-09-04 2011-10-31 Зингента Партисипейшнс Аг Инсектицидные соединения
US8362257B2 (en) 2008-09-18 2013-01-29 Nippon Soda Co., Ltd. Nitrogen-containing heterocyclic compound and pest control agent
US20110288089A1 (en) 2009-01-22 2011-11-24 Syngenta Crop Protection Llc Insecticidal compounds
BR112012020983A2 (pt) 2010-02-25 2016-11-01 Syngenta Ltd processo para a preparação de derivados isoxazolina
CA2807005C (en) 2010-08-05 2015-04-07 Ah Usa 42 Llc Isoxazoline derivatives as antiparasitic agents
AU2012226475C1 (en) 2011-03-10 2015-08-06 Zoetis Services Llc Spirocyclic isoxazoline derivatives as antiparasitic agents
WO2013037626A1 (en) * 2011-09-13 2013-03-21 Syngenta Participations Ag Isothiazoline derivatives as insecticidal compounds
RU2014131951A (ru) * 2012-02-03 2016-03-27 Зоэтис Ллс Производные дигидрофуран азетидина в качестве противопаразитарных агентов
WO2014001120A1 (en) * 2012-06-25 2014-01-03 Syngenta Participations Ag Isothiazole derivatives as insecticidal compounds
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BR112015004695A2 (pt) * 2012-09-07 2017-07-04 Zoetis Llc isoxazolinas espirocíclicas como agentes antiparasitários
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ES2827477T3 (es) * 2015-01-16 2021-05-21 Avista Pharma Solutions Inc Compuestos antiparasitarios
EP3710453A1 (en) * 2017-11-16 2020-09-23 Avista Pharma Solutions, Inc. Single enantiomer antiparasitic compounds

Also Published As

Publication number Publication date
US10342234B2 (en) 2019-07-09
US10092001B2 (en) 2018-10-09
GB2538028B (en) 2017-02-08
GB2572267A (en) 2019-09-25
GB2551214B (en) 2019-06-12
EP3245209B1 (en) 2020-07-29
US20160205936A1 (en) 2016-07-21
US9420793B2 (en) 2016-08-23
GB201620211D0 (en) 2017-01-11
US20170258089A1 (en) 2017-09-14
US20180116223A1 (en) 2018-05-03
AU2016206748B2 (en) 2019-09-05
GB201905337D0 (en) 2019-05-29
AU2016206748B9 (en) 2020-01-16
CN107406458A (zh) 2017-11-28
GB2538028A (en) 2016-11-02
EP3245209A1 (en) 2017-11-22
JP2018509463A (ja) 2018-04-05
JP2020117505A (ja) 2020-08-06
WO2016115315A1 (en) 2016-07-21
AU2019264548A1 (en) 2019-12-05
MX2017009285A (es) 2018-03-14
US9883674B2 (en) 2018-02-06
GB2572267B (en) 2020-01-01
GB2551214A (en) 2017-12-13
CA2973974A1 (en) 2016-07-21
US9686991B2 (en) 2017-06-27
RU2017128818A3 (pt) 2019-06-19
MX2019014575A (es) 2020-02-07
CN107406458B (zh) 2021-01-05
RU2017128818A (ru) 2019-02-18
US20160324156A1 (en) 2016-11-10
ES2827477T3 (es) 2021-05-21
GB201614948D0 (en) 2016-10-19
US20190000085A1 (en) 2019-01-03
MX370163B (es) 2019-12-04
EP3245209A4 (en) 2018-08-22
AU2016206748A1 (en) 2017-08-03
KR20170102359A (ko) 2017-09-08
US10772331B2 (en) 2020-09-15
US20190274305A1 (en) 2019-09-12

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2653 DE 09-11-2021 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.