BR112016024502A8 - uso de uma dose de partículas finas (fdp) de levodopa na fabricação de um medicamento - Google Patents

uso de uma dose de partículas finas (fdp) de levodopa na fabricação de um medicamento

Info

Publication number
BR112016024502A8
BR112016024502A8 BR112016024502A BR112016024502A BR112016024502A8 BR 112016024502 A8 BR112016024502 A8 BR 112016024502A8 BR 112016024502 A BR112016024502 A BR 112016024502A BR 112016024502 A BR112016024502 A BR 112016024502A BR 112016024502 A8 BR112016024502 A8 BR 112016024502A8
Authority
BR
Brazil
Prior art keywords
patient
levodopa
pdf
drug
manufacture
Prior art date
Application number
BR112016024502A
Other languages
English (en)
Portuguese (pt)
Other versions
BR112016024502A2 (pt
Inventor
Freed Martin
M Lipp Michael
P Batycky Richard
Original Assignee
Civitas Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Civitas Therapeutics Inc filed Critical Civitas Therapeutics Inc
Publication of BR112016024502A2 publication Critical patent/BR112016024502A2/pt
Publication of BR112016024502A8 publication Critical patent/BR112016024502A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Psychology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
BR112016024502A 2014-04-21 2014-04-21 uso de uma dose de partículas finas (fdp) de levodopa na fabricação de um medicamento BR112016024502A8 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2014/034778 WO2015163840A1 (en) 2014-04-21 2014-04-21 Rapid relief of motor fluctuations in parkinson's disease

Publications (2)

Publication Number Publication Date
BR112016024502A2 BR112016024502A2 (pt) 2017-08-15
BR112016024502A8 true BR112016024502A8 (pt) 2021-06-29

Family

ID=54332876

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016024502A BR112016024502A8 (pt) 2014-04-21 2014-04-21 uso de uma dose de partículas finas (fdp) de levodopa na fabricação de um medicamento

Country Status (14)

Country Link
US (2) US20170296498A1 (https=)
EP (2) EP3134077A4 (https=)
JP (1) JP2017513866A (https=)
KR (2) KR20170008754A (https=)
CN (2) CN113209055A (https=)
AU (2) AU2014391721B2 (https=)
BR (1) BR112016024502A8 (https=)
CA (1) CA2946165C (https=)
IL (2) IL309959A (https=)
MX (1) MX2016013741A (https=)
RU (1) RU2698330C2 (https=)
SG (1) SG11201608608PA (https=)
WO (1) WO2015163840A1 (https=)
ZA (1) ZA201607833B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112015010601B1 (pt) 2012-11-09 2022-07-19 Civitas Therapeutics, Inc. Composição farmacêutica e uso da composição
BR112020013749A2 (pt) * 2018-01-05 2020-12-01 Impel Neuropharma, Inc. dispensação intranasal de pó de levodopa por dispositivo olfativo de precisão
US11517548B2 (en) 2018-07-19 2022-12-06 Impel Pharmaceuticals Inc. Respiratory tract delivery of levodopa and DOPA decarboxylase inhibitor for treatment of Parkinson's Disease

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6254854B1 (en) 1996-05-24 2001-07-03 The Penn Research Foundation Porous particles for deep lung delivery
US6858199B1 (en) 2000-06-09 2005-02-22 Advanced Inhalation Research, Inc. High efficient delivery of a large therapeutic mass aerosol
US6613308B2 (en) * 2000-09-19 2003-09-02 Advanced Inhalation Research, Inc. Pulmonary delivery in treating disorders of the central nervous system
US6514482B1 (en) 2000-09-19 2003-02-04 Advanced Inhalation Research, Inc. Pulmonary delivery in treating disorders of the central nervous system
AU2003218307B8 (en) * 2002-03-20 2006-08-31 Alkermes, Inc. Pulmonary delivery for levodopa
AR044007A1 (es) * 2003-04-11 2005-08-24 Newron Pharmaceuticals Inc Metodos para el tratamiento de la enfermedad de parkinson
US8496002B2 (en) 2007-06-12 2013-07-30 Civitas Therapeutics, Inc. Powder inhaler devices
GB2454480A (en) * 2007-11-07 2009-05-13 Vectura Group Plc Pulmonary inhalation of levodopa containing compositions in the treatment of Parkinsons disease and other central nervous system disorders
MX2010014222A (es) * 2008-06-30 2011-03-29 Novartis Ag Star Combinaciones que comprenden moduladores de mglur para el tratamiento de enfermedad de parkinson.
US8399513B2 (en) * 2008-10-20 2013-03-19 Xenoport, Inc. Levodopa prodrug mesylate hydrate
TW201304822A (zh) * 2010-11-15 2013-02-01 Vectura Ltd 組成物及用途
KR20210075224A (ko) * 2012-10-22 2021-06-22 키비타스 테라퓨틱스, 인코포레이티드. 파킨슨병의 빠른 경감을 위한 레보도파 제형
US8545878B1 (en) * 2012-11-09 2013-10-01 Civitas Therapeutics, Inc. Capsules containing high doses of levodopa for pulmonary use

Also Published As

Publication number Publication date
EP3831375A1 (en) 2021-06-09
CN106659685A (zh) 2017-05-10
RU2016144340A (ru) 2018-05-22
SG11201608608PA (en) 2016-11-29
RU2016144340A3 (https=) 2018-05-22
AU2014391721A1 (en) 2016-11-03
JP2017513866A (ja) 2017-06-01
CA2946165A1 (en) 2015-10-29
KR20210144946A (ko) 2021-11-30
CN106659685B (zh) 2021-02-05
IL309959A (en) 2024-03-01
IL248445A0 (en) 2016-12-29
US20230053976A1 (en) 2023-02-23
EP3134077A4 (en) 2017-12-20
BR112016024502A2 (pt) 2017-08-15
RU2698330C2 (ru) 2019-08-26
US20170296498A1 (en) 2017-10-19
AU2020239754B2 (en) 2022-06-23
MX2016013741A (es) 2017-04-06
AU2014391721B2 (en) 2020-07-16
WO2015163840A1 (en) 2015-10-29
CA2946165C (en) 2022-10-18
EP3134077A1 (en) 2017-03-01
ZA201607833B (en) 2018-08-29
AU2020239754A1 (en) 2021-01-14
KR20170008754A (ko) 2017-01-24
CN113209055A (zh) 2021-08-06

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]
B07G Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette]

Free format text: NOTIFICACAO DE DEVOLUCAO DO PEDIDO EM FUNCAO DA REVOGACAO DO ART. 229-C DA LEI NO 9.279, DE 1996, POR FORCA DA LEI NO 14.195, DE 2021

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]