BR112016007729B1 - Forma de dosagem compreendendo (s)-3-(4-((4- (morfolinometil)benzil) óxi)-1-oxoisoindolin-2-il)piperidina-2,6- diona e kit que a compreende - Google Patents

Forma de dosagem compreendendo (s)-3-(4-((4- (morfolinometil)benzil) óxi)-1-oxoisoindolin-2-il)piperidina-2,6- diona e kit que a compreende Download PDF

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Publication number
BR112016007729B1
BR112016007729B1 BR112016007729-6A BR112016007729A BR112016007729B1 BR 112016007729 B1 BR112016007729 B1 BR 112016007729B1 BR 112016007729 A BR112016007729 A BR 112016007729A BR 112016007729 B1 BR112016007729 B1 BR 112016007729B1
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Brazil
Prior art keywords
compound
dosage form
pharmaceutically acceptable
amount
solvate
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BR112016007729-6A
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Portuguese (pt)
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BR112016007729A2 (enExample
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Darshan Parikh
Anil Menon
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Celgene Corporation
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Publication of BR112016007729B1 publication Critical patent/BR112016007729B1/pt

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
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    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
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    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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BR112016007729-6A 2013-10-08 2014-10-07 Forma de dosagem compreendendo (s)-3-(4-((4- (morfolinometil)benzil) óxi)-1-oxoisoindolin-2-il)piperidina-2,6- diona e kit que a compreende BR112016007729B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361888419P 2013-10-08 2013-10-08
US61/888,419 2013-10-08
PCT/US2014/059424 WO2015054199A1 (en) 2013-10-08 2014-10-07 Formulations of (s)-3-(4-((4-(morpholinomethyl)benzyloxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione

Publications (2)

Publication Number Publication Date
BR112016007729A2 BR112016007729A2 (enExample) 2017-08-01
BR112016007729B1 true BR112016007729B1 (pt) 2023-05-16

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CN (1) CN105899196B (enExample)
AR (1) AR100663A1 (enExample)
AU (1) AU2014332171C1 (enExample)
BR (1) BR112016007729B1 (enExample)
CA (1) CA2921436C (enExample)
CL (1) CL2016000816A1 (enExample)
CR (1) CR20160131A (enExample)
CY (1) CY1121689T1 (enExample)
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SA (1) SA516370860B1 (enExample)
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TW (1) TW201605493A (enExample)
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