BR112015023153A2 - utilização de um composto e composto - Google Patents

utilização de um composto e composto

Info

Publication number
BR112015023153A2
BR112015023153A2 BR112015023153A BR112015023153A BR112015023153A2 BR 112015023153 A2 BR112015023153 A2 BR 112015023153A2 BR 112015023153 A BR112015023153 A BR 112015023153A BR 112015023153 A BR112015023153 A BR 112015023153A BR 112015023153 A2 BR112015023153 A2 BR 112015023153A2
Authority
BR
Brazil
Prior art keywords
compound
hyperhidrosis
abstract
skin
hours
Prior art date
Application number
BR112015023153A
Other languages
English (en)
Portuguese (pt)
Inventor
Angulo David
S Bodor Nicholas
Original Assignee
Bodor Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50625156&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112015023153(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bodor Laboratories Inc filed Critical Bodor Laboratories Inc
Publication of BR112015023153A2 publication Critical patent/BR112015023153A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/02Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/0216Solid or semisolid forms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4906Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
    • A61K8/4913Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q15/00Anti-perspirants or body deodorants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/14Quaternary ammonium compounds, e.g. edrophonium, choline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/205Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A61K8/41Amines
    • A61K8/416Quaternary ammonium compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Birds (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
BR112015023153A 2013-03-15 2014-03-14 utilização de um composto e composto BR112015023153A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361798073P 2013-03-15 2013-03-15
PCT/US2014/028332 WO2014144075A1 (en) 2013-03-15 2014-03-14 Anticholinergic glycopyrrolate esters for the treatment of hyperhidrosis

Publications (1)

Publication Number Publication Date
BR112015023153A2 true BR112015023153A2 (pt) 2017-07-18

Family

ID=50625156

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015023153A BR112015023153A2 (pt) 2013-03-15 2014-03-14 utilização de um composto e composto

Country Status (22)

Country Link
US (5) US9220707B2 (enExample)
EP (1) EP2968267B1 (enExample)
JP (4) JP6223543B2 (enExample)
KR (4) KR20210043742A (enExample)
CN (2) CN109364066A (enExample)
AU (1) AU2014227923B2 (enExample)
BR (1) BR112015023153A2 (enExample)
CA (1) CA2904724C (enExample)
DK (1) DK2968267T3 (enExample)
ES (1) ES2673098T3 (enExample)
HK (1) HK1217177A1 (enExample)
HU (1) HUE038448T2 (enExample)
IL (1) IL241307B (enExample)
MX (1) MX363601B (enExample)
MY (1) MY192033A (enExample)
PH (1) PH12015501987A1 (enExample)
PL (1) PL2968267T3 (enExample)
PT (1) PT2968267T (enExample)
SG (1) SG11201507602SA (enExample)
TR (1) TR201808040T4 (enExample)
WO (1) WO2014144075A1 (enExample)
ZA (1) ZA201506834B (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT2968267T (pt) * 2013-03-15 2018-06-15 Bodor Laboratories Inc Ésteres anticolinergénicos suaves para o tratamento de hiper-hidrose
US20150259283A1 (en) * 2014-03-13 2015-09-17 Brickell Biotech, Inc. Formulation for soft anticholinergic analogs
WO2015138700A1 (en) * 2014-03-13 2015-09-17 Bodor Laboratories, Inc. Use of selected anticholinergic zwitterions
EP3290053B1 (en) * 2015-04-30 2021-02-17 Hisamitsu Pharmaceutical Co., Inc. Topical composition comprising oxybutynin for the treatment of hyperhidrosis
CA3232529A1 (en) * 2015-07-21 2017-01-26 Bodor Laboratories, Inc. Formulation for soft anticholinergic analogs
WO2017044412A1 (en) 2015-09-11 2017-03-16 Bodor Laboratories, Inc. Methods and compositions for soft anticholinergic esters
AU2016318594A1 (en) * 2015-09-11 2018-04-26 Bodor Laboratories, Inc. Methods and compositions for soft anticholinergic zwitterions
US20190224164A1 (en) * 2016-07-01 2019-07-25 Bodor Laboratories, Inc. Compositions and methods for treatment of copd
TWI767507B (zh) * 2016-07-21 2022-06-11 美商波德實驗股份有限公司 軟性抗膽鹼類似物之製劑
KR101951021B1 (ko) 2017-02-06 2019-02-22 주식회사 퍼슨 발한억제 기능을 가지는 자외선 차단 화장료 조성물 및 이를 사용한 자외선 차단제의 제조방법
HUE047368T2 (hu) * 2017-07-17 2020-04-28 Dr August Wolff Gmbh & Co Kg Arzneimittel Olaj-a-vízben emulzió
JP2021532112A (ja) 2018-07-24 2021-11-25 ドクトア・アウグスト・ボルフ・ゲーエムベーハー・ウント・コンパニー・カー・ゲー−アルツナイミツテル 抗コリン性化合物の局所用エマルション
SG10201912063PA (en) * 2019-12-12 2021-07-29 Nat Skin Centre Singapore Pte Ltd A pharmaceutical formulation
WO2021177257A1 (ja) 2020-03-03 2021-09-10 科研製薬株式会社 原発性腋窩多汗症の治療方法、及びその医薬
KR20220149550A (ko) 2020-03-03 2022-11-08 가켄 세이야쿠 가부시키가이샤 소피로늄 브로마이드를 포함하는 의약
KR20250006082A (ko) 2022-04-14 2025-01-10 독토르. 아우구스트 볼프 게엠베하 운트 코. 카게 아르쯔네이미텔 중증 다한증 및 과도 발한을 치료하기 위한 항콜린성 화합물의 국소 제형
EP4260852A1 (en) 2022-04-14 2023-10-18 Dr. August Wolff GmbH & Co. KG Arzneimittel Topical formulation of an anticholinergic compound for treating severe hyperhidrosis and excessive sweating
KR102611847B1 (ko) * 2023-03-27 2023-12-12 주식회사 이플라스크 무스카린 수용체 길항 활성을 갖는 신규한 피롤리디늄 화합물 및 이의 용도

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5292530A (en) 1991-06-02 1994-03-08 Helene Curtis, Inc. Stable anhydrous topically-active composition and suspending agent therefor
EP1438001A4 (en) 2001-09-26 2006-03-15 Alison B Lukacsko COMPOSITIONS AND METHODS FOR INHIBITING ECCRINS PERSPIRATION IN HUMANS
US8252316B2 (en) 2002-05-03 2012-08-28 Purepharm Inc. Method of topically applying glycopyrrolate solution using absorbent pad to reduce sweating
GB0428416D0 (en) 2004-12-24 2005-02-02 Novartis Ag Organic compounds
GB0428418D0 (en) 2004-12-24 2005-02-02 Novartis Ag Organic compounds
US7399861B2 (en) 2005-11-10 2008-07-15 Bodor Nicholas S Soft anticholinergic esters
CA2627982C (en) 2005-11-10 2013-09-10 Nicholas S. Bodor Soft anticholinergic esters
US8071693B2 (en) 2006-06-22 2011-12-06 Sabic Innovative Plastics Ip B.V. Polysiloxane/polyimide copolymers and blends thereof
MX2010004262A (es) 2007-10-18 2010-05-14 Stiefel Res Australia Pty Ltd Formulaciones topicas de glicopirrolato.
PT2968267T (pt) * 2013-03-15 2018-06-15 Bodor Laboratories Inc Ésteres anticolinergénicos suaves para o tratamento de hiper-hidrose

Also Published As

Publication number Publication date
KR20150128942A (ko) 2015-11-18
US10772867B2 (en) 2020-09-15
SG11201507602SA (en) 2015-10-29
PT2968267T (pt) 2018-06-15
EP2968267B1 (en) 2018-04-25
AU2014227923B2 (en) 2019-02-14
AU2014227923A1 (en) 2015-10-08
HK1220369A1 (en) 2017-05-05
HUE038448T2 (hu) 2018-10-29
WO2014144075A1 (en) 2014-09-18
US9492429B2 (en) 2016-11-15
IL241307B (en) 2019-07-31
MY192033A (en) 2022-07-24
CN109364066A (zh) 2019-02-22
US10383846B2 (en) 2019-08-20
HK1217177A1 (zh) 2016-12-30
JP2017105811A (ja) 2017-06-15
CN105050596A (zh) 2015-11-11
DK2968267T3 (en) 2018-06-25
JP6461214B2 (ja) 2019-01-30
CA2904724A1 (en) 2014-09-18
MX2015012072A (es) 2016-05-05
KR102153457B1 (ko) 2020-09-08
JP6223543B2 (ja) 2017-11-01
IL241307A0 (en) 2015-11-30
PL2968267T3 (pl) 2018-09-28
US9220707B2 (en) 2015-12-29
KR102050299B1 (ko) 2019-11-29
KR20210043742A (ko) 2021-04-21
JP7008988B2 (ja) 2022-01-25
MX363601B (es) 2019-03-28
JP2018115187A (ja) 2018-07-26
JP6694908B2 (ja) 2020-05-20
US20140275204A1 (en) 2014-09-18
KR102241660B1 (ko) 2021-04-19
WO2014144075A8 (en) 2015-10-15
CA2904724C (en) 2021-01-26
US20160067214A1 (en) 2016-03-10
ZA201506834B (en) 2018-12-19
US9895350B2 (en) 2018-02-20
TR201808040T4 (tr) 2018-06-21
US20190328707A1 (en) 2019-10-31
US20160310464A1 (en) 2016-10-27
JP2016517431A (ja) 2016-06-16
JP2020122002A (ja) 2020-08-13
KR20190133072A (ko) 2019-11-29
ES2673098T3 (es) 2018-06-19
PH12015501987A1 (en) 2016-01-11
EP2968267A1 (en) 2016-01-20
US20180185331A1 (en) 2018-07-05
KR20200065103A (ko) 2020-06-08

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B12B Appeal against refusal [chapter 12.2 patent gazette]