KR20210043742A - 다한증 치료용 항콜린성 글리코피롤레이트 에스테르 - Google Patents
다한증 치료용 항콜린성 글리코피롤레이트 에스테르 Download PDFInfo
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- KR20210043742A KR20210043742A KR1020217010876A KR20217010876A KR20210043742A KR 20210043742 A KR20210043742 A KR 20210043742A KR 1020217010876 A KR1020217010876 A KR 1020217010876A KR 20217010876 A KR20217010876 A KR 20217010876A KR 20210043742 A KR20210043742 A KR 20210043742A
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Classifications
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
- A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
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- A—HUMAN NECESSITIES
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/205—Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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- A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
- A61K8/41—Amines
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- Chemical & Material Sciences (AREA)
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- Medicinal Chemistry (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Birds (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
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- Oil, Petroleum & Natural Gas (AREA)
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- Neurology (AREA)
- Biomedical Technology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361798073P | 2013-03-15 | 2013-03-15 | |
| US61/798,073 | 2013-03-15 | ||
| PCT/US2014/028332 WO2014144075A1 (en) | 2013-03-15 | 2014-03-14 | Anticholinergic glycopyrrolate esters for the treatment of hyperhidrosis |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| KR1020207015539A Division KR102241660B1 (ko) | 2013-03-15 | 2014-03-14 | 다한증 치료용 항콜린성 글리코피롤레이트 에스테르 |
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| KR1020197034502A Active KR102153457B1 (ko) | 2013-03-15 | 2014-03-14 | 다한증 치료용 항콜린성 글리코피롤레이트 에스테르 |
| KR1020207015539A Active KR102241660B1 (ko) | 2013-03-15 | 2014-03-14 | 다한증 치료용 항콜린성 글리코피롤레이트 에스테르 |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| KR102611847B1 (ko) * | 2023-03-27 | 2023-12-12 | 주식회사 이플라스크 | 무스카린 수용체 길항 활성을 갖는 신규한 피롤리디늄 화합물 및 이의 용도 |
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| PT2968267T (pt) * | 2013-03-15 | 2018-06-15 | Bodor Laboratories Inc | Ésteres anticolinergénicos suaves para o tratamento de hiper-hidrose |
| US20150259283A1 (en) * | 2014-03-13 | 2015-09-17 | Brickell Biotech, Inc. | Formulation for soft anticholinergic analogs |
| WO2015138700A1 (en) * | 2014-03-13 | 2015-09-17 | Bodor Laboratories, Inc. | Use of selected anticholinergic zwitterions |
| EP3290053B1 (en) * | 2015-04-30 | 2021-02-17 | Hisamitsu Pharmaceutical Co., Inc. | Topical composition comprising oxybutynin for the treatment of hyperhidrosis |
| CA3232529A1 (en) * | 2015-07-21 | 2017-01-26 | Bodor Laboratories, Inc. | Formulation for soft anticholinergic analogs |
| WO2017044412A1 (en) | 2015-09-11 | 2017-03-16 | Bodor Laboratories, Inc. | Methods and compositions for soft anticholinergic esters |
| AU2016318594A1 (en) * | 2015-09-11 | 2018-04-26 | Bodor Laboratories, Inc. | Methods and compositions for soft anticholinergic zwitterions |
| US20190224164A1 (en) * | 2016-07-01 | 2019-07-25 | Bodor Laboratories, Inc. | Compositions and methods for treatment of copd |
| TWI767507B (zh) * | 2016-07-21 | 2022-06-11 | 美商波德實驗股份有限公司 | 軟性抗膽鹼類似物之製劑 |
| KR101951021B1 (ko) | 2017-02-06 | 2019-02-22 | 주식회사 퍼슨 | 발한억제 기능을 가지는 자외선 차단 화장료 조성물 및 이를 사용한 자외선 차단제의 제조방법 |
| HUE047368T2 (hu) * | 2017-07-17 | 2020-04-28 | Dr August Wolff Gmbh & Co Kg Arzneimittel | Olaj-a-vízben emulzió |
| JP2021532112A (ja) | 2018-07-24 | 2021-11-25 | ドクトア・アウグスト・ボルフ・ゲーエムベーハー・ウント・コンパニー・カー・ゲー−アルツナイミツテル | 抗コリン性化合物の局所用エマルション |
| SG10201912063PA (en) * | 2019-12-12 | 2021-07-29 | Nat Skin Centre Singapore Pte Ltd | A pharmaceutical formulation |
| WO2021177257A1 (ja) | 2020-03-03 | 2021-09-10 | 科研製薬株式会社 | 原発性腋窩多汗症の治療方法、及びその医薬 |
| KR20220149550A (ko) | 2020-03-03 | 2022-11-08 | 가켄 세이야쿠 가부시키가이샤 | 소피로늄 브로마이드를 포함하는 의약 |
| KR20250006082A (ko) | 2022-04-14 | 2025-01-10 | 독토르. 아우구스트 볼프 게엠베하 운트 코. 카게 아르쯔네이미텔 | 중증 다한증 및 과도 발한을 치료하기 위한 항콜린성 화합물의 국소 제형 |
| EP4260852A1 (en) | 2022-04-14 | 2023-10-18 | Dr. August Wolff GmbH & Co. KG Arzneimittel | Topical formulation of an anticholinergic compound for treating severe hyperhidrosis and excessive sweating |
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| US5292530A (en) | 1991-06-02 | 1994-03-08 | Helene Curtis, Inc. | Stable anhydrous topically-active composition and suspending agent therefor |
| EP1438001A4 (en) | 2001-09-26 | 2006-03-15 | Alison B Lukacsko | COMPOSITIONS AND METHODS FOR INHIBITING ECCRINS PERSPIRATION IN HUMANS |
| US8252316B2 (en) | 2002-05-03 | 2012-08-28 | Purepharm Inc. | Method of topically applying glycopyrrolate solution using absorbent pad to reduce sweating |
| GB0428416D0 (en) | 2004-12-24 | 2005-02-02 | Novartis Ag | Organic compounds |
| GB0428418D0 (en) | 2004-12-24 | 2005-02-02 | Novartis Ag | Organic compounds |
| US7399861B2 (en) | 2005-11-10 | 2008-07-15 | Bodor Nicholas S | Soft anticholinergic esters |
| CA2627982C (en) | 2005-11-10 | 2013-09-10 | Nicholas S. Bodor | Soft anticholinergic esters |
| US8071693B2 (en) | 2006-06-22 | 2011-12-06 | Sabic Innovative Plastics Ip B.V. | Polysiloxane/polyimide copolymers and blends thereof |
| MX2010004262A (es) | 2007-10-18 | 2010-05-14 | Stiefel Res Australia Pty Ltd | Formulaciones topicas de glicopirrolato. |
| PT2968267T (pt) * | 2013-03-15 | 2018-06-15 | Bodor Laboratories Inc | Ésteres anticolinergénicos suaves para o tratamento de hiper-hidrose |
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2018
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2019
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102611847B1 (ko) * | 2023-03-27 | 2023-12-12 | 주식회사 이플라스크 | 무스카린 수용체 길항 활성을 갖는 신규한 피롤리디늄 화합물 및 이의 용도 |
| WO2024205157A1 (en) * | 2023-03-27 | 2024-10-03 | Eflask Co., Ltd. | Novel pyrrolidinium compounds having antagonistic activity against muscarinic receptors and use thereof |
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