BR112015010512A2 - derivados de carboxamida de 3-aminociclopentano - Google Patents

derivados de carboxamida de 3-aminociclopentano

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Publication number
BR112015010512A2
BR112015010512A2 BR112015010512A BR112015010512A BR112015010512A2 BR 112015010512 A2 BR112015010512 A2 BR 112015010512A2 BR 112015010512 A BR112015010512 A BR 112015010512A BR 112015010512 A BR112015010512 A BR 112015010512A BR 112015010512 A2 BR112015010512 A2 BR 112015010512A2
Authority
BR
Brazil
Prior art keywords
aminocyclopentane
carboxamide derivatives
inflammation
cancer
diseases
Prior art date
Application number
BR112015010512A
Other languages
English (en)
Portuguese (pt)
Inventor
Leuthner Brigitta
Tsaklakidis Christos
Czodrowski Paul
Staehle Wolfgang
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of BR112015010512A2 publication Critical patent/BR112015010512A2/pt

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    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • C—CHEMISTRY; METALLURGY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

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BR112015010512A 2012-11-16 2013-10-17 derivados de carboxamida de 3-aminociclopentano BR112015010512A2 (pt)

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US20050053631A1 (en) 2003-09-10 2005-03-10 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Method of decreasing sebum production
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KR20150085045A (ko) 2015-07-22
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IL238827A0 (en) 2015-06-30
AU2013347232A8 (en) 2015-08-06
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AR093461A1 (es) 2015-06-10
MX2015006037A (es) 2015-08-07

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