BR112015006571A2 - composição farmacêutica, processo para preparar uma composição farmacêutica, uso de uma composição farmacêutica, e, método para a profilaxia ou tratamento de asma, doença pulmonar obstrutiva crônica e distúrbios respiratórios relacionados - Google Patents
composição farmacêutica, processo para preparar uma composição farmacêutica, uso de uma composição farmacêutica, e, método para a profilaxia ou tratamento de asma, doença pulmonar obstrutiva crônica e distúrbios respiratórios relacionadosInfo
- Publication number
- BR112015006571A2 BR112015006571A2 BR112015006571A BR112015006571A BR112015006571A2 BR 112015006571 A2 BR112015006571 A2 BR 112015006571A2 BR 112015006571 A BR112015006571 A BR 112015006571A BR 112015006571 A BR112015006571 A BR 112015006571A BR 112015006571 A2 BR112015006571 A2 BR 112015006571A2
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical composition
- prophylaxis
- preparing
- treatment
- respiratory disorders
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 8
- 238000004519 manufacturing process Methods 0.000 title abstract 3
- 238000011321 prophylaxis Methods 0.000 title abstract 3
- 208000023504 respiratory system disease Diseases 0.000 title abstract 3
- 238000011282 treatment Methods 0.000 title abstract 3
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 title abstract 2
- 208000006673 asthma Diseases 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000003814 drug Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 239000003380 propellant Substances 0.000 abstract 1
- LERNTVKEWCAPOY-DZZGSBJMSA-N tiotropium Chemical compound O([C@H]1C[C@@H]2[N+]([C@H](C1)[C@@H]1[C@H]2O1)(C)C)C(=O)C(O)(C=1SC=CC=1)C1=CC=CS1 LERNTVKEWCAPOY-DZZGSBJMSA-N 0.000 abstract 1
- 229940110309 tiotropium Drugs 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pulmonology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Otolaryngology (AREA)
- Emergency Medicine (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
1 / 1 resumo âcomposiãão farmacãutica, processo para preparar uma composiãão farmacãutica, uso de uma composiãão farmacãutica, e, mãtodo para a profilaxia ou tratamento de asma, doenãa pulmonar obstrutiva crãnica e distãrbios respiratãrios relacionadosâ a presente invenã§ã£o refere-se a uma composiã§ã£o farmacãªutica compreendendo tiotrã³pio, um propulsor de hidrofuoralcano (hfa) e opcionalmente um ou mais excipientes farmaceuticamente aceitã¡veis; a um processo para preparar uma composiã§ã£o farmacãªutica como esta e o uso desta na medicina, em particular para a profilaxia e tratamento de distãºrbios respiratã³rios.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN3092MU2012 | 2012-10-23 | ||
IN280MU2013 | 2013-01-31 | ||
PCT/GB2013/000454 WO2014064410A2 (en) | 2012-10-23 | 2013-10-23 | Pharmaceutical composition |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112015006571A2 true BR112015006571A2 (pt) | 2017-07-04 |
Family
ID=54261200
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015006571A BR112015006571A2 (pt) | 2012-10-23 | 2013-10-23 | composição farmacêutica, processo para preparar uma composição farmacêutica, uso de uma composição farmacêutica, e, método para a profilaxia ou tratamento de asma, doença pulmonar obstrutiva crônica e distúrbios respiratórios relacionados |
Country Status (10)
Country | Link |
---|---|
US (1) | US20150250713A1 (pt) |
JP (1) | JP2016503390A (pt) |
KR (1) | KR20150096371A (pt) |
CN (1) | CN104918604A (pt) |
AU (1) | AU2013336492A1 (pt) |
BR (1) | BR112015006571A2 (pt) |
CA (1) | CA2885767A1 (pt) |
MX (1) | MX2015003731A (pt) |
WO (1) | WO2014064410A2 (pt) |
ZA (1) | ZA201501930B (pt) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2016317040A1 (en) * | 2015-08-31 | 2018-03-29 | Mercator Medsystems, Inc. | Local administration of drugs for the treatment of asthma |
BR122020022602B1 (pt) | 2015-12-04 | 2024-03-05 | Mexichem Fluor S.A. De C.V. | Composição farmacêutica |
CN106880637B (zh) * | 2015-12-15 | 2021-01-29 | 天津金耀集团有限公司 | 一种环索奈德福莫特罗噻托溴铵复方干粉吸入剂组合物 |
CN106880635B (zh) * | 2015-12-15 | 2021-02-02 | 天津金耀集团有限公司 | 一种环索奈德福莫特罗干粉吸入剂组合物 |
CN106466322A (zh) * | 2016-08-25 | 2017-03-01 | 杭州百诚医药科技股份有限公司 | 一种以布地奈德和噻托溴铵为活性成分的复方制剂 |
WO2018051128A1 (en) | 2016-09-19 | 2018-03-22 | Mexichem Fluor S.A. De C.V. | Pharmaceutical composition |
GB2554090A (en) * | 2016-09-19 | 2018-03-28 | Mexichem Fluor Sa De Cv | Pharmaceutical compound |
US10792256B2 (en) | 2016-09-19 | 2020-10-06 | Mexichem Fluor S.A. De C.V. | Pharmaceutical composition |
UA124240C2 (uk) * | 2016-09-19 | 2021-08-11 | Мехікем Флуор С.А. Де С.В. | Фармацевтична композиція |
JP6781831B2 (ja) * | 2016-09-19 | 2020-11-04 | メキシケム フロー エセ・ア・デ・セ・ヴェ | 医薬組成物 |
CN114272238A (zh) | 2016-09-19 | 2022-04-05 | 墨西哥氟石股份公司 | 药物组合物 |
US20210275439A1 (en) * | 2018-06-07 | 2021-09-09 | Kindeva Drug Delivery L.P. | Fluticasone and vilanterol formulation and inhaler |
US20210220367A1 (en) * | 2020-01-20 | 2021-07-22 | Cai Gu Huang | Inhalable formulation of a solution containing glycopyrrolate and olodaterol hydrochloride |
CN111481550A (zh) * | 2020-05-14 | 2020-08-04 | 王兆霖 | 含有噻托溴铵和阿福特罗的药物制剂 |
CN111467498A (zh) * | 2020-05-14 | 2020-07-31 | 王兆霖 | 药物组合物制剂 |
CN113768906B (zh) * | 2021-10-25 | 2023-05-09 | 上海方予健康医药科技有限公司 | 新型糖皮质激素吸入气雾剂及药物组件 |
EP4212106A1 (en) | 2022-01-13 | 2023-07-19 | Cuantum Medical Cosmetics, S.L. | Handheld device for applying a cyanoacrylate adhesive composition |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7311894B2 (en) * | 2002-03-28 | 2007-12-25 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | HFA suspension formulations containing an anticholinergic |
DE10214263A1 (de) * | 2002-03-28 | 2003-10-16 | Boehringer Ingelheim Pharma | HFA-Suspensionsformulierungen enthaltend ein Anticholinergikum |
WO2004054580A1 (en) * | 2002-12-16 | 2004-07-01 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Tiotropium containing hfc solution formulations |
ES2259915B1 (es) | 2005-03-15 | 2007-12-16 | Laboratorio Aldo-Union, S.A. | Nueva formulacion estable de aerosoles en suspension y procedimiento de obtencion. |
WO2008152398A2 (en) * | 2007-06-14 | 2008-12-18 | Cipla Limited | Formulations for inhalation |
GB0801876D0 (en) * | 2008-02-01 | 2008-03-12 | Vectura Group Plc | Suspension formulations |
MX2011004730A (es) * | 2008-11-04 | 2011-05-30 | Cipla Ltd | Composicion farmaceutica en aerosol. |
EP2201934A1 (en) | 2008-12-23 | 2010-06-30 | CHIESI FARMACEUTICI S.p.A. | Tiotropium aerosol formulation products with improved chemical stability |
WO2011076843A2 (en) * | 2009-12-23 | 2011-06-30 | Chiesi Farmaceutici S.P.A. | Combination therapy for copd |
US20130274232A1 (en) * | 2010-07-16 | 2013-10-17 | Cipla Limited | Pharmaceutical Compositions |
WO2012093252A1 (en) * | 2011-01-06 | 2012-07-12 | Cipla Limited | Pharmaceutical composition |
-
2013
- 2013-10-23 WO PCT/GB2013/000454 patent/WO2014064410A2/en active Application Filing
- 2013-10-23 KR KR1020157007523A patent/KR20150096371A/ko not_active Application Discontinuation
- 2013-10-23 CA CA2885767A patent/CA2885767A1/en not_active Abandoned
- 2013-10-23 BR BR112015006571A patent/BR112015006571A2/pt not_active IP Right Cessation
- 2013-10-23 AU AU2013336492A patent/AU2013336492A1/en not_active Abandoned
- 2013-10-23 CN CN201380050294.2A patent/CN104918604A/zh active Pending
- 2013-10-23 MX MX2015003731A patent/MX2015003731A/es unknown
- 2013-10-23 US US14/431,561 patent/US20150250713A1/en not_active Abandoned
- 2013-10-23 JP JP2015537342A patent/JP2016503390A/ja active Pending
-
2015
- 2015-03-20 ZA ZA2015/01930A patent/ZA201501930B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CA2885767A1 (en) | 2014-05-01 |
WO2014064410A3 (en) | 2014-08-07 |
KR20150096371A (ko) | 2015-08-24 |
AU2013336492A1 (en) | 2015-04-09 |
MX2015003731A (es) | 2015-06-15 |
WO2014064410A2 (en) | 2014-05-01 |
CN104918604A (zh) | 2015-09-16 |
ZA201501930B (en) | 2016-01-27 |
WO2014064410A8 (en) | 2014-06-19 |
JP2016503390A (ja) | 2016-02-04 |
US20150250713A1 (en) | 2015-09-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |