BR112012029170A2 - fármaco antimalárico que contém ácido 5-aminolevulínico ou um derivado do mesmo como um princípio ativo - Google Patents
fármaco antimalárico que contém ácido 5-aminolevulínico ou um derivado do mesmo como um princípio ativoInfo
- Publication number
- BR112012029170A2 BR112012029170A2 BR112012029170A BR112012029170A BR112012029170A2 BR 112012029170 A2 BR112012029170 A2 BR 112012029170A2 BR 112012029170 A BR112012029170 A BR 112012029170A BR 112012029170 A BR112012029170 A BR 112012029170A BR 112012029170 A2 BR112012029170 A2 BR 112012029170A2
- Authority
- BR
- Brazil
- Prior art keywords
- derivative
- active ingredient
- antimalarial drug
- aminolevulinic acid
- drug containing
- Prior art date
Links
- 239000004480 active ingredient Substances 0.000 title abstract 3
- 239000003430 antimalarial agent Substances 0.000 title abstract 3
- ZGXJTSGNIOSYLO-UHFFFAOYSA-N 88755TAZ87 Chemical compound NCC(=O)CCC(O)=O ZGXJTSGNIOSYLO-UHFFFAOYSA-N 0.000 title abstract 2
- 229960002749 aminolevulinic acid Drugs 0.000 title abstract 2
- 201000004792 malaria Diseases 0.000 abstract 2
- 208000035473 Communicable disease Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 244000045947 parasite Species 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 230000003449 preventive effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229940124597 therapeutic agent Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
- A61K31/221—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having an amino group, e.g. acetylcholine, acetylcarnitine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/06—Aluminium, calcium or magnesium; Compounds thereof, e.g. clay
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/26—Iron; Compounds thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/30—Zinc; Compounds thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
fármaco antimalárico que contém ácido 5-aminolevulínico ou um derivado de mesmo como um princípio ativo a presente invenção refere-se a um fármaco antimalárico que é útil para a prevenção e o tratamento de doenças infecciosas causadas por parasitas causadores da malária. um agente preventivo e/ou terapêutico para malária que contém, como um princípio ativo 5-amiolevulínico (ala), um derivado do mesmo, ou um sal farmacologicamente aceitável do mesmo, é usado.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2010115721 | 2010-05-19 | ||
PCT/JP2011/002770 WO2011145343A1 (ja) | 2010-05-19 | 2011-05-18 | 5-アミノレブリン酸又はその誘導体を有効成分とする抗マラリア薬 |
Publications (2)
Publication Number | Publication Date |
---|---|
BR112012029170A2 true BR112012029170A2 (pt) | 2017-07-18 |
BR112012029170B1 BR112012029170B1 (pt) | 2020-05-19 |
Family
ID=44991461
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012029170A BR112012029170B1 (pt) | 2010-05-19 | 2011-05-18 | uso de um fármaco antimalárico que contém ácido 5-aminolevulínico ou um derivado do mesmo |
Country Status (10)
Country | Link |
---|---|
US (2) | US9089530B2 (pt) |
EP (1) | EP2572711B1 (pt) |
JP (1) | JP5582441B2 (pt) |
KR (2) | KR20120137506A (pt) |
CN (2) | CN106109455A (pt) |
AU (1) | AU2011256661B2 (pt) |
BR (1) | BR112012029170B1 (pt) |
CA (1) | CA2799491C (pt) |
NZ (1) | NZ603465A (pt) |
WO (1) | WO2011145343A1 (pt) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2012063487A1 (ja) * | 2010-11-10 | 2012-05-18 | 国立大学法人東京工業大学 | アラレマイシン又はその誘導体を有効成分とする抗マラリア薬 |
US9550073B2 (en) * | 2011-06-16 | 2017-01-24 | Sbi Pharmaceuticals Co., Ltd. | Therapeutic agent for allergic rhinitis |
JP5907357B2 (ja) | 2011-10-12 | 2016-04-26 | Sbiファーマ株式会社 | 移植臓器生着促進剤 |
HUE043511T2 (hu) * | 2012-07-13 | 2019-08-28 | Sbi Pharmaceuticals Co Ltd | Immuntoleranciát kiváltó szer |
EP3168296B1 (en) * | 2014-07-11 | 2020-09-09 | SBI Pharmaceuticals Co., Ltd. | Agent for improving normal development rate of fertilized eggs |
US10925963B2 (en) * | 2015-06-22 | 2021-02-23 | Washington University | Combination artemisinin and chemiluminescent photodynamic therapy and uses therefor |
CL2016003379A1 (es) * | 2016-12-29 | 2017-08-04 | Univ Santiago Chile | “composición que comprende ácido delta-aminolevulínico (ala) o un derivado del mismo y oxianiones y teluro o sus derivados y su uso para el control de patógenos.” |
CN109495427B (zh) * | 2017-09-12 | 2021-05-07 | 腾讯科技(深圳)有限公司 | 多媒体数据展示方法、装置、存储介质和计算机设备 |
CN108635581A (zh) * | 2018-05-23 | 2018-10-12 | 昆药集团股份有限公司 | 一种组合物及其在制备治疗肿瘤的药物中的应用 |
JP2022166334A (ja) * | 2019-09-19 | 2022-11-02 | 国立大学法人 東京大学 | 鎌状赤血球症の改善及び/又は予防剤 |
CN113952360B (zh) * | 2021-09-14 | 2023-03-10 | 上海交通大学 | 一种亚铁离子在治疗疟疾的药物中的应用 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5079262A (en) | 1989-07-28 | 1992-01-07 | Queen's University At Kingston | Method of detection and treatment of malignant and non-malignant lesions utilizing 5-aminolevulinic acid |
US5955490A (en) * | 1989-07-28 | 1999-09-21 | Queen's University At Kingston | Photochemotherapeutic method using 5-aminolevulinic acid and other precursors of endogenous porphyrins |
US6710066B2 (en) * | 1989-07-28 | 2004-03-23 | Queen's University At Kingston | Photochemotherapeutic method using 5-aminolevulinic acid and other precursors of endogenous porphyrins |
FR2777782B1 (fr) | 1998-04-22 | 2001-05-18 | Alexandre Marti | Solution pour la preparation d'une substance pharmaceutique pour le diagnostic et/ou le traitement de lesions tissulaires |
ES2464169T3 (es) | 2004-04-28 | 2014-05-30 | Cosmo Oil Co., Ltd. | Restaurador capilar |
JP5034032B2 (ja) | 2004-09-29 | 2012-09-26 | Sbiファーマ株式会社 | 腫瘍診断剤 |
US8609073B2 (en) * | 2005-03-04 | 2013-12-17 | Dusa Pharmaceuticals, Inc. | Compositions and methods for reducing photosensitivity associated with photodynamic therapy |
CA2606140C (en) | 2005-04-28 | 2011-07-19 | Cosmo Oil Co., Ltd. | External preparation for skin |
-
2011
- 2011-05-18 CN CN201610470997.6A patent/CN106109455A/zh active Pending
- 2011-05-18 JP JP2012515757A patent/JP5582441B2/ja active Active
- 2011-05-18 AU AU2011256661A patent/AU2011256661B2/en active Active
- 2011-05-18 EP EP11783280.8A patent/EP2572711B1/en active Active
- 2011-05-18 NZ NZ603465A patent/NZ603465A/xx unknown
- 2011-05-18 KR KR1020127029697A patent/KR20120137506A/ko active Application Filing
- 2011-05-18 CA CA2799491A patent/CA2799491C/en active Active
- 2011-05-18 BR BR112012029170A patent/BR112012029170B1/pt active IP Right Grant
- 2011-05-18 WO PCT/JP2011/002770 patent/WO2011145343A1/ja active Application Filing
- 2011-05-18 CN CN2011800242058A patent/CN102905702A/zh active Pending
- 2011-05-18 US US13/698,090 patent/US9089530B2/en active Active
- 2011-05-18 KR KR1020147026883A patent/KR101723834B1/ko active IP Right Grant
-
2015
- 2015-06-22 US US14/745,823 patent/US9463175B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
KR20120137506A (ko) | 2012-12-21 |
KR101723834B1 (ko) | 2017-04-06 |
CA2799491C (en) | 2015-03-17 |
AU2011256661B2 (en) | 2013-07-11 |
US20150283102A1 (en) | 2015-10-08 |
US9089530B2 (en) | 2015-07-28 |
KR20140121490A (ko) | 2014-10-15 |
EP2572711A4 (en) | 2013-11-20 |
JPWO2011145343A1 (ja) | 2013-07-22 |
US9463175B2 (en) | 2016-10-11 |
WO2011145343A1 (ja) | 2011-11-24 |
CN102905702A (zh) | 2013-01-30 |
CN106109455A (zh) | 2016-11-16 |
EP2572711A1 (en) | 2013-03-27 |
US20130108710A1 (en) | 2013-05-02 |
EP2572711B1 (en) | 2017-09-20 |
JP5582441B2 (ja) | 2014-09-03 |
CA2799491A1 (en) | 2011-11-24 |
AU2011256661A1 (en) | 2012-11-29 |
NZ603465A (en) | 2013-10-25 |
BR112012029170B1 (pt) | 2020-05-19 |
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Legal Events
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B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B07E | Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
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B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 18/05/2011, OBSERVADAS AS CONDICOES LEGAIS. |