BR112012015233A2 - "processo de preparação de composto farmacêuticos e compostos intermediarios - Google Patents

"processo de preparação de composto farmacêuticos e compostos intermediarios

Info

Publication number
BR112012015233A2
BR112012015233A2 BR112012015233A BR112012015233A BR112012015233A2 BR 112012015233 A2 BR112012015233 A2 BR 112012015233A2 BR 112012015233 A BR112012015233 A BR 112012015233A BR 112012015233 A BR112012015233 A BR 112012015233A BR 112012015233 A2 BR112012015233 A2 BR 112012015233A2
Authority
BR
Brazil
Prior art keywords
compounds
preparation
pharmaceutical
intermediate compounds
pharmaceutical compounds
Prior art date
Application number
BR112012015233A
Other languages
English (en)
Inventor
Angéla Pandur
Balázs Volk
Bálint Nyulasi
Enikö Molnár
György Ruzsics
Judit Broda
József Barkóczy
József Debreczeni
Kalmán Nagy
Márta Makkay
Tamás Gregor
Tibor Mezei
Zsusanna Szentkirállyi
Original Assignee
Egis Giogyszergyar Nyilvanosan Mükodo Reszvenytarsasag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Egis Giogyszergyar Nyilvanosan Mükodo Reszvenytarsasag filed Critical Egis Giogyszergyar Nyilvanosan Mükodo Reszvenytarsasag
Publication of BR112012015233A2 publication Critical patent/BR112012015233A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
BR112012015233A 2009-12-21 2010-12-21 "processo de preparação de composto farmacêuticos e compostos intermediarios BR112012015233A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU0900794A HU229031B1 (en) 2009-12-21 2009-12-21 Process for producing prasurgel and its intermediate
PCT/HU2010/000149 WO2011077174A1 (en) 2009-12-21 2010-12-21 Process for preparing pharmaceutical compounds and intermediate compounds

Publications (1)

Publication Number Publication Date
BR112012015233A2 true BR112012015233A2 (pt) 2015-09-22

Family

ID=89989451

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012015233A BR112012015233A2 (pt) 2009-12-21 2010-12-21 "processo de preparação de composto farmacêuticos e compostos intermediarios

Country Status (8)

Country Link
US (1) US9169265B2 (pt)
EP (1) EP2516447A1 (pt)
BR (1) BR112012015233A2 (pt)
EA (1) EA023057B1 (pt)
GE (1) GEP20146163B (pt)
HU (1) HU229031B1 (pt)
UA (1) UA110608C2 (pt)
WO (1) WO2011077174A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102775422B (zh) * 2012-03-13 2014-12-31 山东新华制药股份有限公司 普拉格雷中间体的一种晶型

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2576901B1 (fr) 1985-01-31 1987-03-20 Sanofi Sa Nouveaux derives de l'acide a-(oxo-2 hexahydro-2,4,5,6,7,7a thieno (3,2-c) pyridyl-5) phenyl acetique, leur procede de preparation et leur application therapeutique
FI101150B (fi) 1991-09-09 1998-04-30 Sankyo Co Menetelmä lääkeaineina käyttökelpoisten tetrahydrotienopyridiinin johd annaisten valmistamiseksi
DE69526443T2 (de) 1994-10-07 2002-12-12 Ube Industries 2-silyloxy-tetrahydrothienopyridin, sein salz und verfahren zu seiner herstellung
RU2161282C1 (ru) 1999-05-13 2000-12-27 Багнюков Сергей Анатольевич Газовый баллончик и способ его заправки
KR101784001B1 (ko) 2006-04-04 2017-10-23 케이지 액퀴지션 엘엘씨 항혈소판제와 산 억제제를 포함하는 경구 투여용 약학 조성물
TWI392681B (zh) 2006-04-06 2013-04-11 Daiichi Sankyo Co Ltd 高純度普拉格雷及其酸加成鹽之製法
JP2007303860A (ja) 2006-05-09 2007-11-22 Fujikura Ltd 磁気デバイス
AU2008222000B2 (en) 2007-03-02 2012-06-14 Daiichi Sankyo Company, Limited Process for production of prasugrel hydrochloride having high purity
CZ302135B6 (cs) 2007-07-09 2010-11-10 Zentiva, A. S. Zpusob výroby 5-[2-cyklopropyl-1-(2-fluorfenyl)-2-oxoethyl]-4, 5, 6, 7-tetrahydrothieno[3,2-c]pyridin-2-yl acetátu (prasugrelu)
EP2205611A4 (en) * 2007-11-09 2012-02-22 Reddys Lab Ltd Dr PROCESS FOR THE PRODUCTION OF PRASUGREL AND SALTS AND POLYMERS THEREOF
WO2009066326A2 (en) 2007-11-19 2009-05-28 Msn Laboratories Limited Improved process for the preparation of prasugrel and its pharmaceutically acceptable salts
CN101177430A (zh) * 2007-12-11 2008-05-14 鲁南制药集团股份有限公司 氢化吡啶衍生物及其盐的制备方法
CN101245072B (zh) 2008-03-21 2011-03-30 上海医药工业研究院 制备普拉格雷的中间体及其制备方法
CN101245073B (zh) 2008-03-21 2011-03-23 上海医药工业研究院 一种医药中间体及其制备方法
CN101250192B (zh) 2008-03-24 2010-08-11 上海医药工业研究院 5-(α-环丙基羰基-2-氟苄基)-2-氧-2,4,5,6,7,7a-六氢噻吩并[3,2-c]吡啶的制备方法
CN101250193B (zh) 2008-03-28 2010-09-08 上海医药工业研究院 2-烷氧基-5-(α-环丙基羰基-2-氟苄基)-4,5,6,7-四氢噻吩并[3,2-c]吡啶的制备方法

Also Published As

Publication number Publication date
US9169265B2 (en) 2015-10-27
EA023057B1 (ru) 2016-04-29
EP2516447A1 (en) 2012-10-31
GEP20146163B (en) 2014-09-10
HUP0900794A2 (en) 2011-10-28
HU0900794D0 (en) 2010-03-01
EA201290535A1 (ru) 2013-05-30
HU229031B1 (en) 2013-07-29
WO2011077174A1 (en) 2011-06-30
UA110608C2 (uk) 2016-01-25
US20120330018A1 (en) 2012-12-27

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]