BR0316482A - Processo aperfeiçoado para a preparação de indenos 1,3 substituìdos - Google Patents
Processo aperfeiçoado para a preparação de indenos 1,3 substituìdosInfo
- Publication number
- BR0316482A BR0316482A BR0316482-9A BR0316482A BR0316482A BR 0316482 A BR0316482 A BR 0316482A BR 0316482 A BR0316482 A BR 0316482A BR 0316482 A BR0316482 A BR 0316482A
- Authority
- BR
- Brazil
- Prior art keywords
- improved process
- preparing
- indenes
- substituted indenes
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C253/00—Preparation of carboxylic acid nitriles
- C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
- C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D317/30—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/45—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings
- C07C255/47—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings to carbon atoms of rings being part of condensed ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Rheumatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Addiction (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Circuit Arrangements For Discharge Lamps (AREA)
Abstract
"PROCESSO APERFEIçOADO PARA A PREPARAçãO DE INDENOS 1,3 SUBSTITUìDOS". A presente invenção refere-se a um processo aperfeiçoado para a preparação de indenos 1,3 substituídos que são intermediários úteis na síntese de compostos arila aza-policíclicos condensados como agentes para o tratamento de distúrbios neurológicos e psicológicos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US42902902P | 2002-11-25 | 2002-11-25 | |
PCT/IB2003/005121 WO2004048318A1 (en) | 2002-11-25 | 2003-11-12 | Improved process for the preparation of 1,3-substituted indenes |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0316482A true BR0316482A (pt) | 2005-10-11 |
Family
ID=32393492
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0316482-9A BR0316482A (pt) | 2002-11-25 | 2003-11-12 | Processo aperfeiçoado para a preparação de indenos 1,3 substituìdos |
Country Status (16)
Country | Link |
---|---|
US (1) | US7285686B2 (pt) |
EP (1) | EP1567483A1 (pt) |
JP (1) | JP2006507342A (pt) |
KR (1) | KR100655848B1 (pt) |
CN (1) | CN1714075A (pt) |
AR (1) | AR042205A1 (pt) |
AU (1) | AU2003278510B8 (pt) |
BR (1) | BR0316482A (pt) |
CA (1) | CA2511762A1 (pt) |
MX (1) | MXPA05005517A (pt) |
PL (1) | PL377292A1 (pt) |
RS (1) | RS20050393A (pt) |
RU (1) | RU2284319C2 (pt) |
TW (1) | TWI245756B (pt) |
WO (1) | WO2004048318A1 (pt) |
ZA (1) | ZA200503190B (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2009504852A (ja) | 2005-08-11 | 2009-02-05 | ユニバーシティ オブ マサチューセッツ ロウエル | オレフィンおよび保護または非保護のヒドロキシスチレン単位を含む共重合体を形成するための方法 |
WO2009143347A2 (en) | 2008-05-22 | 2009-11-26 | Teva Pharmaceutical Industries Ltd. | Varenicline tosylate, an intermediate in the preparation process of varenicline l-tartrate |
US20090318695A1 (en) * | 2008-06-19 | 2009-12-24 | Vinod Kumar Kansal | Processes for the preparation of varenicline and intermediates thereof |
WO2010005643A1 (en) * | 2008-07-10 | 2010-01-14 | Teva Pharmaceutical Industries Ltd. | Processes for purifying varenicline l-tartrate salt and preparing crystalline forms of varenicline l-tartrate salt |
RU2012102052A (ru) | 2009-06-22 | 2013-11-20 | Тева Фармасьютикал Индастриз Лтд. | Твердые формы солей варениклина и способы их получения |
US20160296438A1 (en) * | 2015-04-08 | 2016-10-13 | Kemin Industries, Inc. | Protective action of lutein against blue light on human skin cell lines |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6605610B1 (en) | 1997-12-31 | 2003-08-12 | Pfizer Inc | Aryl fused azapolycyclic compounds |
DK1044189T4 (en) | 1997-12-31 | 2015-03-30 | Pfizer Prod Inc | Aryl-fused fused azapolycyclic connections |
DE60225433T2 (de) * | 2001-04-20 | 2008-06-12 | Pfizer Products Inc., Groton | Verfahren zur herstellung von 1,3-substituierte indene und aryl-annellierte azapolycyclische verbindungen |
ATE402134T1 (de) | 2002-11-20 | 2008-08-15 | Pfizer Prod Inc | Methode zur herstellung von indan-1,3- dicarbonsäuren |
US20070066827A1 (en) | 2003-01-15 | 2007-03-22 | Pfizer Inc. | Process for the preparation of aryl fused polycyclic lactams |
-
2003
- 2003-11-12 PL PL377292A patent/PL377292A1/pl unknown
- 2003-11-12 BR BR0316482-9A patent/BR0316482A/pt not_active IP Right Cessation
- 2003-11-12 CA CA002511762A patent/CA2511762A1/en not_active Abandoned
- 2003-11-12 RS YUP-2005/0393A patent/RS20050393A/sr unknown
- 2003-11-12 AU AU2003278510A patent/AU2003278510B8/en not_active Ceased
- 2003-11-12 EP EP03769810A patent/EP1567483A1/en not_active Withdrawn
- 2003-11-12 JP JP2004554771A patent/JP2006507342A/ja not_active Withdrawn
- 2003-11-12 CN CNA2003801040364A patent/CN1714075A/zh active Pending
- 2003-11-12 RU RU2005115881/04A patent/RU2284319C2/ru active
- 2003-11-12 MX MXPA05005517A patent/MXPA05005517A/es active IP Right Grant
- 2003-11-12 WO PCT/IB2003/005121 patent/WO2004048318A1/en active Application Filing
- 2003-11-12 KR KR1020057009301A patent/KR100655848B1/ko not_active IP Right Cessation
- 2003-11-17 US US10/714,735 patent/US7285686B2/en not_active Expired - Fee Related
- 2003-11-24 TW TW092132907A patent/TWI245756B/zh not_active IP Right Cessation
- 2003-11-24 AR ARP030104329A patent/AR042205A1/es unknown
-
2005
- 2005-04-20 ZA ZA200503190A patent/ZA200503190B/en unknown
Also Published As
Publication number | Publication date |
---|---|
CA2511762A1 (en) | 2004-06-10 |
AU2003278510B8 (en) | 2008-07-10 |
AR042205A1 (es) | 2005-06-15 |
US7285686B2 (en) | 2007-10-23 |
RU2005115881A (ru) | 2006-02-27 |
AU2003278510A1 (en) | 2004-06-18 |
JP2006507342A (ja) | 2006-03-02 |
WO2004048318A8 (en) | 2005-05-12 |
TWI245756B (en) | 2005-12-21 |
RS20050393A (en) | 2007-12-31 |
AU2003278510B2 (en) | 2008-06-05 |
ZA200503190B (en) | 2006-07-26 |
KR100655848B1 (ko) | 2006-12-11 |
MXPA05005517A (es) | 2005-07-25 |
CN1714075A (zh) | 2005-12-28 |
US20050004379A1 (en) | 2005-01-06 |
TW200413301A (en) | 2004-08-01 |
EP1567483A1 (en) | 2005-08-31 |
KR20050087801A (ko) | 2005-08-31 |
PL377292A1 (pl) | 2006-01-23 |
RU2284319C2 (ru) | 2006-09-27 |
WO2004048318A1 (en) | 2004-06-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: application dismissed [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2160 DE 29/05/2012. |