BR0214703A - Derivados de aminoacetonitrila e seu uso para controlar parasitas - Google Patents

Derivados de aminoacetonitrila e seu uso para controlar parasitas

Info

Publication number
BR0214703A
BR0214703A BR0214703-3A BR0214703A BR0214703A BR 0214703 A BR0214703 A BR 0214703A BR 0214703 A BR0214703 A BR 0214703A BR 0214703 A BR0214703 A BR 0214703A
Authority
BR
Brazil
Prior art keywords
control parasites
amino acetonitrile
acetonitrile derivatives
parasites
derivatives
Prior art date
Application number
BR0214703-3A
Other languages
English (en)
Inventor
Pierre Ducray
Thomas Goebel
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0214703A publication Critical patent/BR0214703A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/42—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/34—Nitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/24—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton
    • C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"DERIVADOS DE AMINOACETONITRILA E SEU USO PARA CONTROLAR PARASITAS". A presente invenção refere-se a novos compostos da fórmula geral em que R~ 1~, R~ 2~, X, Ar~ 1~, e Ar~ 2~ são como definido na reivindicação 1, e em quaisquer enanciómeros destes. Os ingredientes ativos tem propriedades terapêuticas vantajosas. Elas são particularmente adequadas para controlar parasitas em animais homeotérmicos.
BR0214703-3A 2001-12-06 2002-12-05 Derivados de aminoacetonitrila e seu uso para controlar parasitas BR0214703A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH22252001 2001-12-06
PCT/EP2002/013811 WO2003048112A1 (en) 2001-12-06 2002-12-05 Aminoacetonitrile derivatives and their use for controlling parasites

Publications (1)

Publication Number Publication Date
BR0214703A true BR0214703A (pt) 2004-08-31

Family

ID=4568089

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0214703-3A BR0214703A (pt) 2001-12-06 2002-12-05 Derivados de aminoacetonitrila e seu uso para controlar parasitas

Country Status (15)

Country Link
US (2) US7091371B2 (pt)
EP (1) EP1456170A1 (pt)
JP (1) JP2005511685A (pt)
KR (1) KR100648117B1 (pt)
CN (2) CN1274672C (pt)
AR (1) AR037746A1 (pt)
AU (1) AU2002358620B2 (pt)
BR (1) BR0214703A (pt)
CA (1) CA2466570A1 (pt)
CO (1) CO5590952A2 (pt)
MX (1) MXPA04005455A (pt)
RU (1) RU2293725C2 (pt)
TW (1) TWI261053B (pt)
WO (1) WO2003048112A1 (pt)
ZA (1) ZA200403577B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7705044B2 (en) * 2001-05-15 2010-04-27 Novartis Ag Benzamidoacetonitriles and their use as antiparasitics
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
JP2007513650A (ja) * 2003-11-20 2007-05-31 アンジオテック インターナショナル アーゲー 移植可能なセンサーおよび移植可能なポンプならびに瘢痕化抑制剤
US8218748B2 (en) * 2006-07-24 2012-07-10 Hewlett-Packard Development Company, L.P. Telephone call chaining
RS60858B1 (sr) * 2007-05-15 2020-10-30 Boehringer Ingelheim Animal Health Usa Inc Ariloazol-2-il cijanoetilamino jedinjenja, postupci dobijanja i postupci njihove primene
NZ592382A (en) * 2008-10-21 2013-03-28 Merial Ltd Thioamide compounds, method of making and method of using thereof
JP2012508168A (ja) * 2008-11-07 2012-04-05 ハンツマン ペトロケミカル エルエルシー ポリアミノアセトニトリル、これらの製造および使用方法
CA2945453C (en) 2008-11-14 2021-03-02 Merial, Inc. Enantiomerically enriched aryloazol-2-yl cyanoethylamino paraciticidal compounds
UA114287C2 (uk) * 2011-03-02 2017-05-25 Дзе Юніверсіті Оф Токіо Засіб для боротьби з ендопаразитами
US8710043B2 (en) 2011-06-24 2014-04-29 Amgen Inc. TRPM8 antagonists and their use in treatments
CA2839703A1 (en) 2011-06-24 2012-12-27 Amgen Inc. Trpm8 antagonists and their use in treatments
US8952009B2 (en) 2012-08-06 2015-02-10 Amgen Inc. Chroman derivatives as TRPM8 inhibitors
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
CN110407681B (zh) * 2019-08-12 2023-05-02 海南大学 一种脱氢姜酮衍生物、其制备方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3457294A (en) * 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) * 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
US5959870A (en) 1998-02-20 1999-09-28 Gamma-Metrics Real-time optimization for mix beds
US6239077B1 (en) * 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
MXPA03005701A (es) 2000-12-20 2003-10-06 Novartis Ag Compuestos organicos.

Also Published As

Publication number Publication date
CN1668580A (zh) 2005-09-14
CN1293047C (zh) 2007-01-03
CN1274672C (zh) 2006-09-13
AU2002358620A1 (en) 2003-06-17
AU2002358620B2 (en) 2006-08-31
EP1456170A1 (en) 2004-09-15
TWI261053B (en) 2006-09-01
TW200300755A (en) 2003-06-16
US20050033081A1 (en) 2005-02-10
CO5590952A2 (es) 2005-12-30
KR20050044719A (ko) 2005-05-12
CN1599716A (zh) 2005-03-23
RU2293725C2 (ru) 2007-02-20
US20060264653A1 (en) 2006-11-23
WO2003048112A1 (en) 2003-06-12
JP2005511685A (ja) 2005-04-28
ZA200403577B (en) 2006-06-28
US7091371B2 (en) 2006-08-15
CA2466570A1 (en) 2003-06-12
MXPA04005455A (es) 2005-04-19
KR100648117B1 (ko) 2006-11-24
AR037746A1 (es) 2004-12-01
RU2004120790A (ru) 2005-05-27

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2064 DE 27/07/2010.